메뉴 건너뛰기




Volumn 33, Issue 11, 2008, Pages 926-931

Rivoglitazone hydrochloride. PPARγ agonist, insulin sensitizer, treatment of diabetes

Author keywords

[No Author keywords available]

Indexed keywords

BALAGLITAZONE; CI 1037; DE 101; GLITAZONE DERIVATIVE; GLUCOSE; ITRACONAZOLE; LOBEGLITAZONE; MOXIFLOXACIN; NETOGLITAZONE; PEROXISOME PROLIFERATOR ACTIVATED RECEPTOR ALPHA; PEROXISOME PROLIFERATOR ACTIVATED RECEPTOR GAMMA; PIOGLITAZONE; PLACEBO; R 106056; RIVOGLITAZONE; ROSIGLITAZONE; UNCLASSIFIED DRUG;

EID: 60549094788     PISSN: 03778282     EISSN: None     Source Type: Journal    
DOI: 10.1358/dof.2008.033.011.1278754     Document Type: Article
Times cited : (2)

References (26)
  • 1
    • 60549116014 scopus 로고    scopus 로고
    • Fujita, T, Wada, K, Oguchi, M. et al, Daiichi Sankyo Co, Ltd, Benzimidazole derivatives, their preparation and their therapeutic use. CA 2177858, EP 0745600, JP 1997295970, JP 2000001487, US 5886014
    • Fujita, T., Wada, K., Oguchi, M. et al. (Daiichi Sankyo Co., Ltd.). Benzimidazole derivatives, their preparation and their therapeutic use. CA 2177858, EP 0745600, JP 1997295970, JP 2000001487, US 5886014.
  • 2
    • 60549088742 scopus 로고    scopus 로고
    • Fujita, T, Izumi, T, Fujiwara, T, Daiichi Sankyo Co, Ltd, Hydrochloride of fused-heterocycle compound. EP 1180519, JP 2001039976, US 2002111373, US 6706746, WO 2000071540
    • Fujita, T., Izumi, T., Fujiwara, T. (Daiichi Sankyo Co., Ltd.). Hydrochloride of fused-heterocycle compound. EP 1180519, JP 2001039976, US 2002111373, US 6706746, WO 2000071540.
  • 3
    • 60549097260 scopus 로고    scopus 로고
    • Kajino, H, Miyamoto, H, Ikeuchi, Y, Sankyo Co, Ltd, Intermediate of 6-substituted-1-methyl-1-H-benzimidazole derivative and method for producing same. CA 2580973, EP 1798216, JP 2006124375, WO 2006035685
    • Kajino, H., Miyamoto, H., Ikeuchi, Y. (Sankyo Co., Ltd.). Intermediate of 6-substituted-1-methyl-1-H-benzimidazole derivative and method for producing same. CA 2580973, EP 1798216, JP 2006124375, WO 2006035685.
  • 4
    • 60549103934 scopus 로고    scopus 로고
    • Nakamura, Y, Satoh, C, Miyamoto, H, Kajino, H, Daiichi San kyo Co, Ltd, Process for producing thiazolidinedione compound and production intermediate thereof. CA 2595782, EP 1894929, JP 2006225382, US 2008103185, WO 2006078037
    • Nakamura, Y., Satoh, C., Miyamoto, H., Kajino, H. (Daiichi San kyo Co., Ltd.). Process for producing thiazolidinedione compound and production intermediate thereof. CA 2595782, EP 1894929, JP 2006225382, US 2008103185, WO 2006078037.
  • 5
    • 60549109927 scopus 로고    scopus 로고
    • Kishi, N, Nakamura, Y, Abe, N, Takebayashi, T, Sankyo Co, Ltd, Intermediates for the synthesis of benzimidazole derivatives and a process for the preparation thereof. CA 2377233, EP 1191019, JP 2001072671, US 2003008907, US 2003199580, US 6525220, US 6753347, WO 2001000570
    • Kishi, N., Nakamura, Y., Abe, N., Takebayashi, T. (Sankyo Co., Ltd.). Intermediates for the synthesis of benzimidazole derivatives and a process for the preparation thereof. CA 2377233, EP 1191019, JP 2001072671, US 2003008907, US 2003199580, US 6525220, US 6753347, WO 2001000570.
  • 6
    • 0035856920 scopus 로고    scopus 로고
    • Zimmet, P., Alberti, K.G., Shaw, J. Global and societal implications of the diabetes epidemic. Nature 201, 414(6865): 782-7.
    • Zimmet, P., Alberti, K.G., Shaw, J. Global and societal implications of the diabetes epidemic. Nature 201, 414(6865): 782-7.
  • 7
    • 0034656345 scopus 로고    scopus 로고
    • ABC of arterial and venous disease: Vascular complications of diabetes
    • Donnelly, R., Emslie-Smith, A.M., Gardner, I.D., Morris, A.D. ABC of arterial and venous disease: Vascular complications of diabetes. BMJ 2000, 320(7241): 1062-6.
    • (2000) BMJ , vol.320 , Issue.7241 , pp. 1062-1066
    • Donnelly, R.1    Emslie-Smith, A.M.2    Gardner, I.D.3    Morris, A.D.4
  • 8
    • 0842263981 scopus 로고    scopus 로고
    • The biology of peroxisome proliferator-activated receptors: Relationship with lipid metabolism and insulin sensitivity
    • Ferre, P. The biology of peroxisome proliferator-activated receptors: Relationship with lipid metabolism and insulin sensitivity. Diabetes 2004, 53(Suppl. 1): S43-50.
    • (2004) Diabetes , vol.53 , Issue.SUPPL. 1
    • Ferre, P.1
  • 14
    • 26144476955 scopus 로고    scopus 로고
    • Antidiabetic characterization of CS-011: A new thiazolidinedione with potent insulin-sensitizing activity
    • June 9-13, San Antonio, Abst 425-P
    • Araki, K., Yachi, M., Hagisawa, Y. et al. Antidiabetic characterization of CS-011: A new thiazolidinedione with potent insulin-sensitizing activity. Diabetes [60th Annu Meet Sci Sess Am Diabetes Assoc (ADA) (June 9-13, San Antonio) 2000] 2000, 49(Suppl. 1): Abst 425-P.
    • (2000) Diabetes [60th Annu Meet Sci Sess Am Diabetes Assoc (ADA) , vol.49 , Issue.SUPPL. 1
    • Araki, K.1    Yachi, M.2    Hagisawa, Y.3
  • 15
    • 60549113069 scopus 로고    scopus 로고
    • Pharmacological characterization of rivoglitazone and its enatiomers in vitro and in vivo
    • June 9-13, Washington, D.C, Abst 2093-PO
    • Ohsumi, J., Kanda, S., Matsui, Y. et al. Pharmacological characterization of rivoglitazone and its enatiomers in vitro and in vivo. 66th Annu Meet Sci Sess Am Diabetes Assoc (ADA) (June 9-13, Washington, D.C.) 2006, Abst 2093-PO.
    • (2006) 66th Annu Meet Sci Sess Am Diabetes Assoc (ADA)
    • Ohsumi, J.1    Kanda, S.2    Matsui, Y.3
  • 16
    • 60549102511 scopus 로고    scopus 로고
    • Potent antidiabetic effects of rivoglitazone, a novel PPARγ agonist, in obese diabetic rodent models
    • Sept 17-21, Amsterdam, Abst 0854
    • Ohsumi, J., Kanda, S., Tanaka, J. et al. Potent antidiabetic effects of rivoglitazone, a novel PPARγ agonist, in obese diabetic rodent models. 43rd Annu Meet Eur Assoc Study Diabetes (EASD) (Sept 17-21, Amsterdam) 2007, Abst 0854.
    • (2007) 43rd Annu Meet Eur Assoc Study Diabetes (EASD)
    • Ohsumi, J.1    Kanda, S.2    Tanaka, J.3
  • 17
    • 60549104450 scopus 로고    scopus 로고
    • The effect of rivoglitazone (Rivo) on expression of genes targeted by PPARα and those implicated in cardiac function
    • Abst 2193-PO
    • Kanda, S., Tanaka, J., Takahashi, K., Nakashima, R., Ohsumi, J. The effect of rivoglitazone (Rivo) on expression of genes targeted by PPARα and those implicated in cardiac function. Diabetes 2006, 55(Suppl. 1): Abst 2193-PO.
    • (2006) Diabetes , vol.55 , Issue.SUPPL. 1
    • Kanda, S.1    Tanaka, J.2    Takahashi, K.3    Nakashima, R.4    Ohsumi, J.5
  • 18
    • 4244016877 scopus 로고    scopus 로고
    • The antidiabetic effect of CI-1037/CS011, a new thiazolidinedione
    • Abst 496-P
    • Pulaski, J.T., Davis, J.A., Yuille, K., Johnson, J.H. The antidiabetic effect of CI-1037/CS011, a new thiazolidinedione. Diabetes 2000, 49(Suppl. 1): Abst 496-P.
    • (2000) Diabetes , vol.49 , Issue.SUPPL. 1
    • Pulaski, J.T.1    Davis, J.A.2    Yuille, K.3    Johnson, J.H.4
  • 19
    • 57449101797 scopus 로고    scopus 로고
    • Single and multiple dose pharmacokinetics and pharmacodynamics of rivoglitazone (CS-011) in healthy male volunteers
    • Sept 17-19, Cambridge, Abst 37
    • Walker, J.R., Triscari, J., Dmuchowski, C.F. et al. Single and multiple dose pharmacokinetics and pharmacodynamics of rivoglitazone (CS-011) in healthy male volunteers. 35th Annu Meet Am Coll Clin Pharmacol (ACCP) (Sept 17-19, Cambridge) 2006, Abst 37.
    • (2006) 35th Annu Meet Am Coll Clin Pharmacol (ACCP)
    • Walker, J.R.1    Triscari, J.2    Dmuchowski, C.F.3
  • 20
    • 60549117160 scopus 로고    scopus 로고
    • A single-dose, food-effect and relative bioavailability study of tablet and oral formulations of rivoglitazone in healthy volunteers
    • Abst 48
    • Walker, J.R., Yoshioka, S., Izumi, T. et al. A single-dose, food-effect and relative bioavailability study of tablet and oral formulations of rivoglitazone in healthy volunteers. J Clin Pharmacol 2008, 48(9): Abst 48.
    • (2008) J Clin Pharmacol , vol.48 , Issue.9
    • Walker, J.R.1    Yoshioka, S.2    Izumi, T.3
  • 21
    • 60549091052 scopus 로고    scopus 로고
    • Thorough QTC study with rivoglitazone confirms no exposure-QTC response predicted by PK/PD modelling of pooled phase I/II ECG data
    • Abst 49
    • Walker, J.R., Rohatagi, S., Salazar, D.E. et al. Thorough QTC study with rivoglitazone confirms no exposure-QTC response predicted by PK/PD modelling of pooled phase I/II ECG data. J Clin Pharmacol 2008, 48(9): Abst 49.
    • (2008) J Clin Pharmacol , vol.48 , Issue.9
    • Walker, J.R.1    Rohatagi, S.2    Salazar, D.E.3
  • 22
    • 60549098481 scopus 로고    scopus 로고
    • The effects of rivoglitazone (PPARγ agonist) on adiponectin in healthy subjects
    • June 9-13, Washington, D.C, Abst 570-P
    • Triscari, J., Dmuchowski, C. The effects of rivoglitazone (PPARγ agonist) on adiponectin in healthy subjects. 66th Annu Meet Sci Sess Am Diabetes Assoc (ADA) (June 9-13, Washington, D.C.) 2006, Abst 570-P.
    • (2006) 66th Annu Meet Sci Sess Am Diabetes Assoc (ADA)
    • Triscari, J.1    Dmuchowski, C.2
  • 23
    • 60549089857 scopus 로고    scopus 로고
    • A randomized, multiple-dose, placebo-controlled comparative study of rivoglitazone (Rivo, CS-011) and open-label pioglitazone (Pio) in patients with type 2 diabetes (T2DM)
    • June 6-10, San Francisco, Abst 437-P
    • Truitt, K., Chou, H.S., Wang, A., Walker, J.R., Rosenstock, J. A randomized, multiple-dose, placebo-controlled comparative study of rivoglitazone (Rivo, CS-011) and open-label pioglitazone (Pio) in patients with type 2 diabetes (T2DM). Diabetes [68th Annu Meet Sci Sess Am Diabetes Assoc (ADA) (June 6-10, San Francisco) 2008] 2008, 57(Suppl. 1): Abst 437-P.
    • (2008) Diabetes [68th Annu Meet Sci Sess Am Diabetes Assoc (ADA) , vol.57 , Issue.SUPPL. 1
    • Truitt, K.1    Chou, H.S.2    Wang, A.3    Walker, J.R.4    Rosenstock, J.5
  • 24
    • 60549090646 scopus 로고    scopus 로고
    • Glucose levels in type 2 diabetes treated for 6 weeks with rivoglitazone HCI (CS-011)
    • Abst 571-P
    • Triscari, J., Dmuchowski, C., Isaacsohn, J. Glucose levels in type 2 diabetes treated for 6 weeks with rivoglitazone HCI (CS-011). Diabetes 2006, 55(Suppl. 1): Abst 571-P.
    • (2006) Diabetes , vol.55 , Issue.SUPPL. 1
    • Triscari, J.1    Dmuchowski, C.2    Isaacsohn, J.3
  • 25
    • 60549105412 scopus 로고    scopus 로고
    • Chou, H.S., Wang, A., Walker, J.R., Truitt, K., Rosenstock, J. A randomized, placebo-controlled, 26-week dose response study of rivoglitazone (RIVO, CS-011) versus pioglitazone (PIO) in patients with type 2 diabetes (T2DM). Diabetes [68th Annu Meet Sci Sess Am Diabetes Assoc (ADA) (June 6-10, San Francisco) 2008] 2008, 57(Suppl. 1): Abst 304-OR.
    • Chou, H.S., Wang, A., Walker, J.R., Truitt, K., Rosenstock, J. A randomized, placebo-controlled, 26-week dose response study of rivoglitazone (RIVO, CS-011) versus pioglitazone (PIO) in patients with type 2 diabetes (T2DM). Diabetes [68th Annu Meet Sci Sess Am Diabetes Assoc (ADA) (June 6-10, San Francisco) 2008] 2008, 57(Suppl. 1): Abst 304-OR.
  • 26
    • 57449085287 scopus 로고    scopus 로고
    • The steady-state pharmacokinetics of rivoglitazone (CS-011) are not affected by coadministration of the potent CYP3A4 inhibitor itraconazole
    • March 21-24, Anaheim, Abst Pl-84
    • Walker, J.R., Dmuchowski, C.F., Izumi, T., Samata, N., Mathew, P., Salazar, D.E. The steady-state pharmacokinetics of rivoglitazone (CS-011) are not affected by coadministration of the potent CYP3A4 inhibitor itraconazole. Clin Pharmacol Ther [Annu Meet Am Soc Clin Pharmacol Ther (ASCPT) (March 21-24, Anaheim) 2007] 2007, 81(Suppl. 1): Abst Pl-84.
    • (2007) Clin Pharmacol Ther [Annu Meet Am Soc Clin Pharmacol Ther (ASCPT) , vol.81 , Issue.SUPPL. 1
    • Walker, J.R.1    Dmuchowski, C.F.2    Izumi, T.3    Samata, N.4    Mathew, P.5    Salazar, D.E.6


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.