Evaluation of the local anaesthetic activity of 3-aminobenzo[d]isothiazole derivatives using the rat sciatic nerve model

European Journal of Medicinal Chemistry

Volumn 44, Issue 2, 2009, Pages 473-481

  Geronikaki, Athina ^a   Vicini, Paola ^b   Dabarakis, Nikos ^a   Lagunin, Alexey ^c   Poroikov, Vladimir ^c   Dearden, John ^d   Modarresi, Hassan ^d   Hewitt, Mark ^d   Theophilidis, George ^a  

^a ARISTOTLE UNIVERSITY OF THESSALONIKI   (Greece)

^b UNIVERSITY OF PARMA   (Italy)

^c INSTITUTE OF BIOMEDICAL CHEMISTRY   (Russian Federation)

^d LIVERPOOL JOHN MOORES UNIVERSITY   (United Kingdom)

Author keywords

3 Aminobenzo d isothiazole derivatives; Compound action potential; In vitro; Mammalian; QSAR; Sciatic nerve

Indexed keywords

3 AMINOBENZO[D]ISOTHIAZOLE DERIVATIVE; ISOTHIAZOLE DERIVATIVE; LIDOCAINE; NITROGEN; UNCLASSIFIED DRUG;

ANIMAL TISSUE; ARTICLE; DRUG EFFECT; DRUG EFFICACY; FEMALE; MALE; NONHUMAN; PROBABILITY; RAT; SCIATIC NERVE;

ANESTHETICS, LOCAL; ANIMALS; BENZOTHIAZOLES; COMPUTER SIMULATION; LIDOCAINE; MODELS, MOLECULAR; QUANTITATIVE STRUCTURE-ACTIVITY RELATIONSHIP; RATS; SCIATIC NERVE;

EID: 60149090885     PISSN: 02235234     EISSN: 17683254     Source Type: Journal    
DOI: 10.1016/j.ejmech.2008.04.006     Document Type: Article

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