Estimation of relative microscopic affinity constants of agonists for the active state of the receptor in functional studies on M 2 and M 2 muscarinic receptors

Molecular Pharmacology

Volumn 75, Issue 2, 2009, Pages 381-396

  Tran, John A ^a   Chang, Alexander ^a   Matsui, Minoru ^b   Ehlert, Frederick J ^a,c  

^a UNIVERSITY OF CALIFORNIA   (United States)

^b CHIBA INSTITUTE OF SCIENCE   (Japan)

^c UNIVERSITY OF CALIFORNIA   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

1 (2 CHLOROETHYL) 4 DIPHENYLACETOXYPIPERIDINE; [4 [(3 CHLOROPHENYL)CARBAMOYLOXY] 2 BUTYNYL]TRIMETHYLAMMONIUM; ADRENALIN; ANTIBIOTIC G 418; ARECOLINE; ATROPINE; BETHANECHOL; CARBACHOL; CYCLIC AMP; FORSKOLIN; ISOBUTYLMETHYLXANTHINE; MUSCARINIC M2 RECEPTOR; MUSCARINIC M3 RECEPTOR; OXOTREMORINE; OXOTREMORINE M; PILOCARPINE; TETRODOTOXIN;

ANIMAL CELL; ANIMAL TISSUE; ARTICLE; CHO CELL; CONTROLLED STUDY; DRUG RECEPTOR BINDING; ILEUM; KNOCKOUT MOUSE; MALE; MATHEMATICAL MODEL; MOUSE; NONHUMAN; PREDICTION; PRIORITY JOURNAL; RECEPTOR AFFINITY;

ANIMALS; CHO CELLS; CRICETINAE; CRICETULUS; FEMALE; HUMANS; MALE; MICE; PHYSICAL PROCESSES; PROTEIN INTERACTION DOMAINS AND MOTIFS; RECEPTOR, MUSCARINIC M2; RECEPTOR, MUSCARINIC M3;

EID: 59449084824     PISSN: 0026895X     EISSN: 15210111     Source Type: Journal    
DOI: 10.1124/mol.108.051276     Document Type: Article

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