Synthesis and antitubercular activity of a series of hydrazone and nitrovinyl analogs derived from heterocyclic aldehydes

Journal of Enzyme Inhibition and Medicinal Chemistry

Volumn 24, Issue 1, 2009, Pages 117-124

  Sonar, Vijayakumar N ^a   Crooks, Peter A ^a  

^a Division of Pharmacy Practice and Science   (United States)

Author keywords

3 nitrovinylindoles; Antitubercular activity; Benzo b thiophene 3 hydrazones; Indole 3 hydrazones; Thiophene 3 hydrazones

Indexed keywords

1 BENZYL 3 (2 METHYL 2 NITROVINYL) 1H INDOLE; 1 BENZYL 3 (2 NITROVINYL) 1H INDOLE; 2 METHYL 3 (2 METHYL 2 NITROVINYL) 1H INDOLE; 2 METHYL 3 (2 NITROVINYL) 1H INDOLE; 2 PHENYL 3 (2 METHYL 2 NITROVINYL) 1H INDOLE; 2 PHENYL 3 (2 NITROVINYL) 1H INDOLE; ALDEHYDE DERIVATIVE; HYDRAZONE DERIVATIVE; INDOLE DERIVATIVE; N (2,5 DICHLOROPHENYL) N' (1H INDOL 3 YLMETHYLENE)HYDRAZINE; N (2,5 DICHLOROPHENYL) N' THIOPHEN 3 YLMETHYLENE HYDRAZINE; N BENZO[B]THIOPHEN 3 YLMETHYLENE N' (2,5 DICHLOROPHENYL)HYDRAZINE; N METHYL N PHENYL N' THIOPHEN 3 YLMETHYLENE HYDRAZINE; N METHYL N' (2 METHYL 1H INDOL 3 YLMETHYLENE) N PHENYLHYDRAZINE; N' (1H INDOL 3 YLMETHYLENE) N METHYL N PHENYLHYDRAZINE; N' (1H INDOL 3 YLMETHYLENE) N,N DIMETHYLHYDRAZINE; N' BENZO[B]THIOPHEN 3 YLMETHYLENE N METHYL N PHENYLHYDRAZINE; N,N DIMETHYL N' (2 METHYL 1H INDOL 3 YLMETHYLENE)HYDRAZINE; N,N' BIS(1 METHYL 1H INDOL 3 YLMETHYLENE)HYDRAZINE; N,N' BIS(2 METHYL 1H INDOL 3 YLMETHYLENE)HYDRAZINE; TUBERCULOSTATIC AGENT; UNCLASSIFIED DRUG;

ANTIBACTERIAL ACTIVITY; ARTICLE; BACTERIUM CULTURE; CONTROLLED STUDY; CULTURE MEDIUM; DOSE RESPONSE; DRUG SCREENING; DRUG SYNTHESIS; IC 50; MINIMUM INHIBITORY CONCENTRATION; MYCOBACTERIUM TUBERCULOSIS; NONHUMAN; PRIORITY JOURNAL; STRUCTURE ACTIVITY RELATION;

ALDEHYDES; ANTITUBERCULAR AGENTS; DOSE-RESPONSE RELATIONSHIP, DRUG; HYDRAZONES; INHIBITORY CONCENTRATION 50; MICROBIAL SENSITIVITY TESTS; MYCOBACTERIUM TUBERCULOSIS; VINYL COMPOUNDS;

MYCOBACTERIUM TUBERCULOSIS;

EID: 58949100447     PISSN: 14756366     EISSN: 14756374     Source Type: Journal    
DOI: 10.1080/14756360801915526     Document Type: Article

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