A high-throughput ligand competition binding assay for the androgen receptor and other nuclear receptors

Journal of Biomolecular Screening

Volumn 14, Issue 1, 2009, Pages 43-48

  Féau, Clémentine ^a   Arnold, Leggy A ^a   Kosinski, Aaron ^a   Guy, R Kiplin ^a  

^a ST JUDE CHILDREN S RESEARCH HOSPITAL   (United States)

Author keywords

Androgen receptor; Endocrine disrupting chemicals; High throughput screening; Nuclear receptors; Scintillation proximity assay

Indexed keywords

2 CHLORO 5 NITROBENZANILIDE; ANDROGEN RECEPTOR; ANDROSTANOLONE; ARACHIDONIC ACID; BICALUTAMIDE; CELL NUCLEUS RECEPTOR; CYPROTERONE ACETATE; DEXAMETHASONE; ENDOCRINE DISRUPTOR; ESTRADIOL; FLUTAMIDE; HYDROXYFLUTAMIDE; LINOLEIC ACID; METRIBOLONE; NICKEL; PEROXISOME PROLIFERATOR ACTIVATED RECEPTOR GAMMA; PROGESTERONE; ROSIGLITAZONE; THYROID HORMONE RECEPTOR ALPHA; THYROID HORMONE RECEPTOR BETA; TROGLITAZONE;

ARTICLE; AUTOANALYSIS; BINDING AFFINITY; CHEMICAL LABELING; COST; DRUG RECEPTOR BINDING; FLUORESCENCE; HIGH THROUGHPUT SCREENING; HORMONE BINDING; IC 50; ISOTOPE LABELING; LIGAND BINDING; MATERIAL COATING; PRIORITY JOURNAL; PROTEIN EXPRESSION; PROTEIN PURIFICATION; RADIOASSAY; RECEPTOR BINDING; REPRODUCIBILITY; SCINTILLATION;

ANDROGENS; BINDING, COMPETITIVE; LIGANDS; RADIOLIGAND ASSAY; RECEPTORS, ANDROGEN; RECEPTORS, CYTOPLASMIC AND NUCLEAR;

EID: 58849147947     PISSN: 10870571     EISSN: 1552454X     Source Type: Journal    
DOI: 10.1177/1087057108326662     Document Type: Article

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