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58149158463
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U.S. Patent 6,420,359
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(a) Simoneau, B. U.S. Patent 6,420,359, 2002.
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Simoneau, B.1
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14444278761
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(b) Klunder, J. M.; Hoermann, M.; Cywin, C. L.; David, E.; Brickwood, J. R.; Schwartz, R.; Barringer, K. J.; Pauletti, D.; Shih, C.-K.; Erickson, D. A.; Sorge, C. L.; Joseph, D. P.; Hattox, S. E.; Adams, J.; Grob, P. M. J. Med. Chem. 1998, 41, 2960.
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58149176346
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(d) Beaulieu, P. L.; Duceppe, J.-S.; Haché, B. Synthesis 2002, 4, 528.
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Beaulieu, P.L.1
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5
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58149170742
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(a) Knochel, P.; Bonnet, V.; Mongin, F.; Trécourt, F.; Breton, G.; Marsais, F.; Quéguiner, G. Synlett 2002, 6, 1008.
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Knochel, P.1
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Breton, G.5
Marsais, F.6
Quéguiner, G.7
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6
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0038606694
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10, 1349. For a very similar finding see
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(b) Trécourt, F.; Breton, G.; Bonnet, V.; Mongin, F.; Marsais, F.; Quéguiner, G. Tetrahedron 2000, 56 (10), 1349. For a very similar finding see:
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Tetrahedron
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Trécourt, F.1
Breton, G.2
Bonnet, V.3
Mongin, F.4
Marsais, F.5
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8644283612
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(c) Pierrat, P.; Gros, P.; Fort, Y. Synlett 2004, 13, 2319.
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Pierrat, P.1
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Fort, Y.3
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37049088928
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(a) Fleming, L; Henning, R.; Parker, D. C.; Plaut, H. E.; Sanderson, P. E. J. I Chem. Soc., Perkin Trans. 1 1995, 317.
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11
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0002437012
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JAI Press: Greenwich, CT
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(d) Tamao, K. Advances in Silicon Chemistry; JAI Press: Greenwich, CT, 1996; Vol. 3, pp 1-62.
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Tamao, K.1
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3643127470
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Fleming, I.; Henning, R.; Plaut, H. J. Chem Soc., Chem. Commun. 1984, 29 See also ref 5a.
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(b) Fleming, I.; Henning, R.; Plaut, H. J. Chem Soc., Chem. Commun. 1984, 29 See also ref 5a.
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14
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85026866359
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(a) Kabalka, G. W.; Maddox, J. T.; Shoup, T. Org. Synth. 1996, 73, 116.
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Org. Synth
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Kabalka, G.W.1
Maddox, J.T.2
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0000995951
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(b) Kabalka, G. W.; Shoup, T. M.; Goudagon, N. M. J. Org. Chem. 1989, 54, 5930.
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Kabalka, G.W.1
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0033997284
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(b) Buchwald, S. L.; Fox, J. M.; Huang, X.; Chieffi, A. J. Am. Chem, Soc. 2000, 122, 1360.
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Buchwald, S.L.1
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Chieffi, A.4
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58149160491
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Buchwald, S. L.; Old, D. W.; Wolfe, J. P.; Palucki, M.; Kamikawa, K. U.S. Patent 6,307,087, CAN 135: 318588, 2001.
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(c) Buchwald, S. L.; Old, D. W.; Wolfe, J. P.; Palucki, M.; Kamikawa, K. U.S. Patent 6,307,087, CAN 135: 318588, 2001.
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20
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58149165583
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Hartwig, J. F.; Hamann, B. C. U.S. Patent 6,057,456, CAN 132:293568, 2000.
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(d) Hartwig, J. F.; Hamann, B. C. U.S. Patent 6,057,456, CAN 132:293568, 2000.
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21
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58149162255
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Hartwig, J. F.; Kawatsura, M. U.S. Patent 6,072,073, CAN 133:30376, 2000.
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(e) Hartwig, J. F.; Kawatsura, M. U.S. Patent 6,072,073, CAN 133:30376, 2000.
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22
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58149143535
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Busacca, C. A.; Eriksson, M. C.; Kim, J.-Y. U.S. Patent 6,759,533, CAN 140:59670, 2004.
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(f) Busacca, C. A.; Eriksson, M. C.; Kim, J.-Y. U.S. Patent 6,759,533, CAN 140:59670, 2004.
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25
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85078346696
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(a) Uno, M.; Seto, K.; Ueda, W.; Masuda, M.; Takahashi, S. Synthesis 1985, 506.
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Synthesis
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Uno, M.1
Seto, K.2
Ueda, W.3
Masuda, M.4
Takahashi, S.5
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26
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58149155215
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(b) Yamanaka, H.; Sakamoto, T.; Katoh, E.; Kondo, Y. Chem. Pharm. Bull. 1988, 36, 1664.
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Chem. Pharm. Bull
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Yamanaka, H.1
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0000583866
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(c) Yamanaka, H.; Sakamoto, T.; Katoh, E.; Kondo, Y. Heterocycles 1988, 27, 1353.
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Heterocycles
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Yamanaka, H.1
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0025071072
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(d) Yamanaka, H.; Sakamoto, T.; Katoh, E.; Kondo, Y. Chem. Pharm. Bull. 1990, 38, 1513.
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Kondo, Y.4
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29
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58149172457
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Yamanaka, H.; Sakamoto, T.; Kondo, Y.; Suginome, T.; Ohba, S. Synthesis 1.99.1, 552.
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(e) Yamanaka, H.; Sakamoto, T.; Kondo, Y.; Suginome, T.; Ohba, S. Synthesis 1.99.1, 552.
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30
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0001660401
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For a review see
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(f) Sakamoto, T.; Kondo, Y.; Masumoto, K. Heterocycles 1993, 36, 2509 For a review see:
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(1993)
Heterocycles
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Sakamoto, T.1
Kondo, Y.2
Masumoto, K.3
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31
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0037060980
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(g) Prim, D.; Campagne, J.-M.; Joseph, D.; Andrioletti, B. Tetrahedron 2002, 58, 2041.
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Tetrahedron
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Prim, D.1
Campagne, J.-M.2
Joseph, D.3
Andrioletti, B.4
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32
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0036532342
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Beletskaya, I. P.; Kashin, A. N.; Mitin, A. V.; Wife, R. Tetrahedron Lett. 2002, 43, 2539.
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Tetrahedron Lett
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Beletskaya, I.P.1
Kashin, A.N.2
Mitin, A.V.3
Wife, R.4
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33
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58149153521
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2 led to acid 17 in high yield.
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2 led to acid 17 in high yield.
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34
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0033888943
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For recent examples, see: a
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For recent examples, see: (a) Mannekens, E.; Tourwe, D.; Lubell, W. D. Synthesis 2000, 9, 1214.
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Synthesis
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Mannekens, E.1
Tourwe, D.2
Lubell, W.D.3
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35
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0034044940
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(b) Springer, D. M.; Luh, B.-Y.; Branson, J. J.; McElhone, K. E.; Mansuri, M. M.; Gregor, K. R.; Nettleton, D. O.; Stanley, P. L.; Tramposch, K. M. Bioorg. Med. Chem. 2000, 8, 1087.
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Bioorg. Med. Chem
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Springer, D.M.1
Luh, B.-Y.2
Branson, J.J.3
McElhone, K.E.4
Mansuri, M.M.5
Gregor, K.R.6
Nettleton, D.O.7
Stanley, P.L.8
Tramposch, K.M.9
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37
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0031081369
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(b) Silverman, R. B.; Lu, X.; Blomquist, G. D.; Ding, C. Z.; Yang, S. Bioorg. Med Chem. 1997, 5, 297.
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Silverman, R.B.1
Lu, X.2
Blomquist, G.D.3
Ding, C.Z.4
Yang, S.5
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38
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58149160493
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In situ React-IR might be suitable for monitoring this hydrolysis as well
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(c) In situ React-IR might be suitable for monitoring this hydrolysis as well.
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40
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85008486032
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(b) Periasamy, M.; Prasad, A. S. B.; Kanth, J. V. B. Tetrahedron 1992, 48, 4623.
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Tetrahedron
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Periasamy, M.1
Prasad, A.S.B.2
Kanth, J.V.B.3
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41
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58149150317
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Meyers, A. L; Dickman, D. A.; Smith, G. A.; Gawley, R. E. Organic Syntheses; Wiley & Sons: New York, 1990; Collect. VII, p 530.
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(c) Meyers, A. L; Dickman, D. A.; Smith, G. A.; Gawley, R. E. Organic Syntheses; Wiley & Sons: New York, 1990; Collect. Vol. VII, p 530.
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43
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0037043490
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For a possible explanation, see: a
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For a possible explanation, see: (a) Houk, K. N.; Washington, I. Org. Lett. 2002, 4, 2661.
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(2002)
Org. Lett
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Houk, K.N.1
Washington, I.2
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46
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24944508104
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(c) Kaneko, C.; Okuda, W.; Karasawa, Y.; Somei, M. Chem. Lett. 1980, 547.
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Chem. Lett
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Kaneko, C.1
Okuda, W.2
Karasawa, Y.3
Somei, M.4
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47
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58149148629
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See Experimental Section
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See Experimental Section.
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48
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58149148628
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Busacca, C. A.; Cerreta, M.; Varsolona, R.; Smoliga, J.; Lorenz, J. Vitous, J. U.S. Patent 7,309,700, CAN 1.43:35331.0, 2007.
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Busacca, C. A.; Cerreta, M.; Varsolona, R.; Smoliga, J.; Lorenz, J. Vitous, J. U.S. Patent 7,309,700, CAN 1.43:35331.0, 2007.
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