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Volumn 600, Issue 1-3, 2008, Pages 87-92

The tachykinin NK3 receptor agonist senktide induces locomotor activity in male Mongolian gerbils

Author keywords

Antipsychotic; Aprepitant; Gerbil; Locomotor activity; MK869; Neurokinin; Osanetant; SB222200; SB223412; Senktide; SR142801; Tachykinin; Talnetant

Indexed keywords

ALPHA TOCOPHEROL; APREPITANT; HALOPERIDOL; N (ALPHA ETHYLBENZYL) 3 METHYL 2 PHENYL 4 QUINOLINECARBOXAMIDE; NEUROKININ 3 RECEPTOR; OSANETANT; RISPERIDONE; SENKTIDE; TALNETANT; VOLINANSERIN; DRUG DERIVATIVE; DRUG VEHICLE; MORPHOLINE DERIVATIVE; NEUROKININ 1 RECEPTOR; PEPTIDE FRAGMENT; SUBSTANCE P;

EID: 55949117514     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.ejphar.2008.10.011     Document Type: Article
Times cited : (12)

References (26)
  • 2
    • 0030042422 scopus 로고    scopus 로고
    • Localization of the neuromedin K receptor (NK3) in the central nervous system of the rat
    • Ding Y.Q., Shigemoto R., Takada M., Ohishi H., Nakanishi S., and Mizuno N. Localization of the neuromedin K receptor (NK3) in the central nervous system of the rat. J. Comp. Neurol. 364 (1996) 290-310
    • (1996) J. Comp. Neurol. , vol.364 , pp. 290-310
    • Ding, Y.Q.1    Shigemoto, R.2    Takada, M.3    Ohishi, H.4    Nakanishi, S.5    Mizuno, N.6
  • 3
    • 0026101943 scopus 로고
    • Injection of tachykinins and selective neurokinin receptor ligands into the substantia nigra reticulata increases striatal dopamine and 5-hydroxytryptamine metabolism
    • Humpel C., Saria A., and Regoli D. Injection of tachykinins and selective neurokinin receptor ligands into the substantia nigra reticulata increases striatal dopamine and 5-hydroxytryptamine metabolism. Eur. J. Pharmacol. 195 (1991) 107-114
    • (1991) Eur. J. Pharmacol. , vol.195 , pp. 107-114
    • Humpel, C.1    Saria, A.2    Regoli, D.3
  • 4
    • 0030593435 scopus 로고    scopus 로고
    • Electrophysiological, behavioural and biochemical evidence for activation of brain noradrenergic systems following neurokinin NK3 receptor stimulation
    • Jung M., Michaud J.C., Steinberg R., Barnouin M.C., Hayar A., Mons G., Souilhac J., Emonds-Alt X., Soubrie P., and Le Fur G. Electrophysiological, behavioural and biochemical evidence for activation of brain noradrenergic systems following neurokinin NK3 receptor stimulation. Neuroscience 74 (1996) 403-414
    • (1996) Neuroscience , vol.74 , pp. 403-414
    • Jung, M.1    Michaud, J.C.2    Steinberg, R.3    Barnouin, M.C.4    Hayar, A.5    Mons, G.6    Souilhac, J.7    Emonds-Alt, X.8    Soubrie, P.9    Le Fur, G.10
  • 5
    • 0034192260 scopus 로고    scopus 로고
    • The troubled story of tachykinins and neurokinins
    • Maggi C.A. The troubled story of tachykinins and neurokinins. Trends Pharmacol. Sci. 21 (2000) 173-175
    • (2000) Trends Pharmacol. Sci. , vol.21 , pp. 173-175
    • Maggi, C.A.1
  • 6
    • 44249084680 scopus 로고    scopus 로고
    • Me-talnetant and osanetant interact within overlapping but not identical binding pockets in the human tachykinin NK3 receptor transmembrane domains
    • Malherbe P., Bissantz C., Marcuz A., Kratzeisen C., Zenner M.T., Wettstein J.G., Ratni H., Riemer C., and Spooren W. Me-talnetant and osanetant interact within overlapping but not identical binding pockets in the human tachykinin NK3 receptor transmembrane domains. Mol. Pharmacol. 73 (2008) 1736-1750
    • (2008) Mol. Pharmacol. , vol.73 , pp. 1736-1750
    • Malherbe, P.1    Bissantz, C.2    Marcuz, A.3    Kratzeisen, C.4    Zenner, M.T.5    Wettstein, J.G.6    Ratni, H.7    Riemer, C.8    Spooren, W.9
  • 7
    • 0031768558 scopus 로고    scopus 로고
    • Activation of dopaminergic and cholinergic neurotransmission by tachykinin NK3 receptor stimulation: an in vivo microdialysis approach in guinea pig
    • Marco N., Thirion A., Mons G., Bougault I., Le Fur G., Soubrie P., and Steinberg R. Activation of dopaminergic and cholinergic neurotransmission by tachykinin NK3 receptor stimulation: an in vivo microdialysis approach in guinea pig. Neuropeptides 32 (1998) 481-488
    • (1998) Neuropeptides , vol.32 , pp. 481-488
    • Marco, N.1    Thirion, A.2    Mons, G.3    Bougault, I.4    Le Fur, G.5    Soubrie, P.6    Steinberg, R.7
  • 8
    • 0030614856 scopus 로고    scopus 로고
    • Characterization of NK3 receptors in rabbit isolated iris sphincter muscle
    • Medhurst A.D., Parsons A.A., Roberts J.C., and Hay D.W.P. Characterization of NK3 receptors in rabbit isolated iris sphincter muscle. Br. J. Pharmacol. 120 (1996) 93-101
    • (1996) Br. J. Pharmacol. , vol.120 , pp. 93-101
    • Medhurst, A.D.1    Parsons, A.A.2    Roberts, J.C.3    Hay, D.W.P.4
  • 9
    • 33846177867 scopus 로고    scopus 로고
    • NK3 receptor antagonists for the treatment of schizophrenia
    • Meltzer H., and Prus A. NK3 receptor antagonists for the treatment of schizophrenia. Drug Discov. Today Ther. Strateg. 3 (2006) 555-560
    • (2006) Drug Discov. Today Ther. Strateg. , vol.3 , pp. 555-560
    • Meltzer, H.1    Prus, A.2
  • 10
    • 2942538034 scopus 로고    scopus 로고
    • Placebo-controlled evaluation of four novel compounds for the treatment of schizophrenia and schizoaffective disorder
    • Meta-Trial Study Group
    • Meltzer H.Y., Arvanitis L., Bauer D., Rein W., and Meta-Trial Study Group. Placebo-controlled evaluation of four novel compounds for the treatment of schizophrenia and schizoaffective disorder. Am. J. Psychiatr. 161 (2004) 975-984
    • (2004) Am. J. Psychiatr. , vol.161 , pp. 975-984
    • Meltzer, H.Y.1    Arvanitis, L.2    Bauer, D.3    Rein, W.4
  • 12
    • 0026100201 scopus 로고
    • Mammalian tachykinin receptors
    • Nakanishi S. Mammalian tachykinin receptors. Annu. Rev. Neurosci. 14 (1991) 123-136
    • (1991) Annu. Rev. Neurosci. , vol.14 , pp. 123-136
    • Nakanishi, S.1
  • 13
    • 0030935824 scopus 로고    scopus 로고
    • Tachykinin neurokinin-1 and neurokinin-3 receptor-mediated responses in guinea-pig substantia nigra: an in vitro electrophysiological study
    • Nalivaiko E., Michaud J.C., Soubrie P., Le Fur G., and Feltz P. Tachykinin neurokinin-1 and neurokinin-3 receptor-mediated responses in guinea-pig substantia nigra: an in vitro electrophysiological study. Neuroscience 78 (1997) 745-757
    • (1997) Neuroscience , vol.78 , pp. 745-757
    • Nalivaiko, E.1    Michaud, J.C.2    Soubrie, P.3    Le Fur, G.4    Feltz, P.5
  • 14
    • 0029943956 scopus 로고    scopus 로고
    • Pharmacological characterization of SR 142801: a new non-peptide antagonist of the neurokinin NK-3 receptor
    • Nguyen-Le X.K., Nguyen Q.T., Gobeil F., Pheng L.H., Emonds-Alt X., Breliere J.C., and Regoli D. Pharmacological characterization of SR 142801: a new non-peptide antagonist of the neurokinin NK-3 receptor. Pharmacology 52 (1996) 283-291
    • (1996) Pharmacology , vol.52 , pp. 283-291
    • Nguyen-Le, X.K.1    Nguyen, Q.T.2    Gobeil, F.3    Pheng, L.H.4    Emonds-Alt, X.5    Breliere, J.C.6    Regoli, D.7
  • 15
    • 55949096883 scopus 로고    scopus 로고
    • Nordquist, R.E., Algeyer, B., Pauly-Evers, M., Ozmen, L., Spooren, W., submitted for publication. Pharmacological characterization of senktide-induced tail whips.
    • Nordquist, R.E., Algeyer, B., Pauly-Evers, M., Ozmen, L., Spooren, W., submitted for publication. Pharmacological characterization of senktide-induced tail whips.
  • 16
    • 55949119096 scopus 로고    scopus 로고
    • Pharmacological characterisation of senktide-induced behaviours in the guinea pig
    • Pemberton D.J., Gartlon J.E., Hill M.D.W., and Jones D.N.C. Pharmacological characterisation of senktide-induced behaviours in the guinea pig. J. Psychopharmacol. 18 (2004) A28
    • (2004) J. Psychopharmacol. , vol.18
    • Pemberton, D.J.1    Gartlon, J.E.2    Hill, M.D.W.3    Jones, D.N.C.4
  • 19
    • 0037022687 scopus 로고    scopus 로고
    • Heterologous regulation of trafficking and signaling of G protein-coupled receptors: β-Arrestin-dependent interactions between neurokinin receptors
    • Schmidlin F., Dery O., Bunnett N.W., and Grady E.F. Heterologous regulation of trafficking and signaling of G protein-coupled receptors: β-Arrestin-dependent interactions between neurokinin receptors. PNAS 99 (2002) 3324-3329
    • (2002) PNAS , vol.99 , pp. 3324-3329
    • Schmidlin, F.1    Dery, O.2    Bunnett, N.W.3    Grady, E.F.4
  • 20
    • 0028947870 scopus 로고
    • Pharmacology of tachykinin receptors on neurones in the ventral tegmental area of rat brain slices
    • Seabrook G.R., Bowery B.J., and Hill R.G. Pharmacology of tachykinin receptors on neurones in the ventral tegmental area of rat brain slices. Eur. J. Pharmacol. 273 (1995) 113-119
    • (1995) Eur. J. Pharmacol. , vol.273 , pp. 113-119
    • Seabrook, G.R.1    Bowery, B.J.2    Hill, R.G.3
  • 21
    • 55949105356 scopus 로고    scopus 로고
    • Spooren, W., 2005 (filed). NK-3 Receptor in vivo assay. EP 1829556.
    • Spooren, W., 2005 (filed). NK-3 Receptor in vivo assay. EP 1829556.
  • 22
    • 33644671816 scopus 로고    scopus 로고
    • NK3 receptor antagonists: the next generation of antipsychotics? Nat
    • Spooren W., Riemer C., and Meltzer H. NK3 receptor antagonists: the next generation of antipsychotics? Nat. Rev. Drug. Discov. 4 (2005) 967-975
    • (2005) Rev. Drug. Discov. , vol.4 , pp. 967-975
    • Spooren, W.1    Riemer, C.2    Meltzer, H.3
  • 23
    • 0023807704 scopus 로고
    • The NK-3 tachykinin receptor agonist senktide elicits 5-HT-mediated behaviour following central or peripheral administration in mice and rats
    • Stoessl A.J., Dourish C.T., and Iversen S.D. The NK-3 tachykinin receptor agonist senktide elicits 5-HT-mediated behaviour following central or peripheral administration in mice and rats. Br. J. Pharmacol. 94 (1988) 285-287
    • (1988) Br. J. Pharmacol. , vol.94 , pp. 285-287
    • Stoessl, A.J.1    Dourish, C.T.2    Iversen, S.D.3
  • 25
    • 55949129193 scopus 로고    scopus 로고
    • Swiss Academy of Medical Sciences and Swiss Academy of Sciences, 1995. Ethical Principles and Guidelines for Scientific Experiments on Animals, 2nd ed. http://www.springeronline.com/sgw/cda/pageitems/document/cda_downloaddocument/0,11996,0-0-45-137181-0,00.pdf.
    • Swiss Academy of Medical Sciences and Swiss Academy of Sciences, 1995. Ethical Principles and Guidelines for Scientific Experiments on Animals, 2nd ed. http://www.springeronline.com/sgw/cda/pageitems/document/cda_downloaddocument/0,11996,0-0-45-137181-0,00.pdf.
  • 26
    • 33847142359 scopus 로고    scopus 로고
    • Neurokinin-3 receptor-specific antagonists talnetant and osanetant show distinct mode of action in cellular Ca2+ mobilization but display similar binding kinetics and identical mechanism of binding in ligand cross-competition
    • Tian G., Wilkins D., and Scott C.W. Neurokinin-3 receptor-specific antagonists talnetant and osanetant show distinct mode of action in cellular Ca2+ mobilization but display similar binding kinetics and identical mechanism of binding in ligand cross-competition. Mol. Pharmacol. 71 (2007) 902-911
    • (2007) Mol. Pharmacol. , vol.71 , pp. 902-911
    • Tian, G.1    Wilkins, D.2    Scott, C.W.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.