Pharmacological characterization of sr 142801: A new non-peptide antagonist of the neurokinin nk-3 receptor

Pharmacology

Volumn 52, Issue 5, 1996, Pages 283-291

  Nguyen Le, X K ^a   Nguyen, Q T ^a   Gobeil, F ^a   Pheng, L H ^a   Emonds Alt, X ^a   Breliere J C ^b   Regoli, D ^a  

^a UNIVERSITÉ DE SHERBROOKE   (Canada)

^b SANOFI   (France)

Author keywords

NK 3 receptor antagonist; Smooth muscle; SR 142801

Indexed keywords

3 (2 METHOXYBENZYLAMINO) 2 PHENYLPIPERIDINE; NEUROKININ 1 RECEPTOR; NEUROKININ 2 RECEPTOR; NEUROKININ 3 RECEPTOR; NEUROKININ 3 RECEPTOR ANTAGONIST; OSANETANT; SAREDUTANT;

ANIMAL TISSUE; ARTICLE; BINDING AFFINITY; BLADDER; CAVA VEIN; DRUG RECEPTOR BINDING; GUINEA PIG; HAMSTER; HUMAN; HUMAN TISSUE; ILEUM; NONHUMAN; PORTAL VEIN; PRIORITY JOURNAL; PULMONARY ARTERY; RABBIT; RAT;

ANIMALS; BINDING, COMPETITIVE; CEREBRAL CORTEX; CHO CELLS; CRICETINAE; ENDOTHELIUM, VASCULAR; GUINEA PIGS; HUMANS; MESOCRICETUS; MUSCLE RELAXATION; MUSCLE, SMOOTH; MUSCLE, SMOOTH, VASCULAR; PIPERIDINES; RABBITS; RATS; RATS, SPRAGUE-DAWLEY; RECEPTORS, NEUROKININ-3;

EID: 0029943956     PISSN: 00317012     EISSN: 14230313     Source Type: Journal    
DOI: 10.1159/000139393     Document Type: Article

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