Synthesis of new substituted azetidinoyl and thiazolidinoyl-1,3,4-thiadiazino (6,5-b) indoles as promising anti-inflammatory agents

European Journal of Medicinal Chemistry

Volumn 43, Issue 11, 2008, Pages 2323-2330

  Bhati, Sudhir Kumar ^a   Kumar, Ashok ^a  

^a LLRM MEDICAL COLLEGE   (India)

Author keywords

Anti inflammatory, analgesic, ulcerogenic activities and toxicity studies; Azetidinones; Benzylidenaminoindoles; Thiazolidinones

Indexed keywords

2 ARYL 3 [5 [[(1,3,4)THIADIAZINO[6,5 B]INDOL 3 YLAMINO]METHYL] 1,3,4 THIADIAZOL 2 YL] 1,3 THIAZOLIDIN 4 ONE; 3 CHLORO 4 ARYL 1 [5 [[(1,3,4)THIADIAZINO[6,5 B]INDOL 3 YLAMINO]METHYL] 1,3,4 THIADIAZOL 2 YL]AZETIDIN 2 ONE; ANTIINFLAMMATORY AGENT; INDOLE DERIVATIVE; INDOMETACIN; N [[5 [(ARYLMETHYLENE)AMINO] 1,3,4 THIADIAZOL 2 YL]METHYL][1,3,4]THIADIAZINO[6,5 B]INDOL 3 AMINE; PHENYLBUTAZONE; UNCLASSIFIED DRUG;

ANALGESIC ACTIVITY; ANIMAL EXPERIMENT; ANTIINFLAMMATORY ACTIVITY; ARTICLE; CHEMICAL STRUCTURE; DRUG MECHANISM; DRUG SYNTHESIS; MOUSE; NONHUMAN; ULCEROGENESIS;

ANIMALS; ANTI-INFLAMMATORY AGENTS; AZA COMPOUNDS; INDOLES; INFLAMMATION; MICE; MOLECULAR STRUCTURE; STRUCTURE-ACTIVITY RELATIONSHIP; SULFHYDRYL COMPOUNDS;

EID: 54049152860     PISSN: 02235234     EISSN: 17683254     Source Type: Journal    
DOI: 10.1016/j.ejmech.2007.10.012     Document Type: Article

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