Release of a poorly soluble drug from cross-linked β-cyclodextrin- based polymer pellets prepared via extrusion/spheronisation

Letters in Drug Design and Discovery

Volumn 5, Issue 7, 2008, Pages 462-470

  Bon, Pierre ^a,b   Joudieh, Samer ^a   Lahiani Skiba, Malika ^a   Bounoure, Frederic ^a,b   Dechelotte, Pierre ^c   Skiba, Mohamed ^a  

^a Institut Fédératif de Recherches Multidisciplinaires Sur Les Peptides   (France)

^b In Cyclo   (France)

^c ROUEN UNIVERSITY HOSPITAL   (France)

Author keywords

Characterization; Cyclodextrins; Dissolution; Extrusion spheronisation; Nimesulide; Pellets; Polymers of cyclodextrin

Indexed keywords

ALPHA CYCLODEXTRIN; BETA CYCLODEXTRIN; CROSCARMELLOSE SODIUM; EXCIPIENT; MICROCRYSTALLINE CELLULOSE; NIMESULIDE; PHARMACEL 102; POLYESTER; POLYMER; UNCLASSIFIED DRUG;

ARTICLE; CROSS LINKING; DRUG FORMULATION; DRUG RELEASE; DRUG SOLUBILITY; INFRARED SPECTROSCOPY; LEACHING; MORPHOLOGY; PELLET EXTRUSION; POROSITY; PRIORITY JOURNAL; SCANNING ELECTRON MICROSCOPY; SPHERONIZATION; SURFACE PROPERTY;

EID: 53549121961     PISSN: 15701808     EISSN: None     Source Type: Journal    
DOI: 10.2174/157018008785909822     Document Type: Article

References (19)

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