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Volumn 58, Issue 3, 2008, Pages 257-274

Improved dissolution of a poorly water soluble drug in solid dispersions with polymeric and non-polymeric hydrophilic additives

Author keywords

Amorphous form; Dissolution rate; Irbesartan; Solid dispersion; Solubility

Indexed keywords

IRBESARTAN;

EID: 53549113334     PISSN: 13300075     EISSN: None     Source Type: Journal    
DOI: 10.2478/v10007-008-0016-1     Document Type: Article
Times cited : (39)

References (25)
  • 1
    • 0343527392 scopus 로고    scopus 로고
    • Modern bioavailability, bioequivalence and biopharmaceutics classification system. New scientific approaches to international regulatory standards
    • DOI: 10.1016/S0939-6411(00)00091-6
    • R. Lobenberg and G. L. Amidon, Modern bioavailability, bioequivalence and biopharmaceutics classification system. New scientific approaches to international regulatory standards, Eur. J. Pharm. Biopharm. 50 (2000) 3-12; DOI: 10.1016/S0939-6411(00)00091-6.
    • (2000) Eur. J. Pharm. Biopharm , vol.50 , pp. 3-12
    • Lobenberg, R.1    Amidon, G.L.2
  • 2
    • 85176822415 scopus 로고    scopus 로고
    • H. Yan, S. E. Tabibi and S. H. Yalkowsky, Solubilization of two structurally related anticancer drugs: XK-469 and PPA, J. Pharm. Sci. 95 (2006) 97-107; DOI: 10.1002/jps.20500.
    • H. Yan, S. E. Tabibi and S. H. Yalkowsky, Solubilization of two structurally related anticancer drugs: XK-469 and PPA, J. Pharm. Sci. 95 (2006) 97-107; DOI: 10.1002/jps.20500.
  • 3
    • 1042264121 scopus 로고    scopus 로고
    • Impact of solid state properties on developability assessment of drug candidates
    • DOI: 10.1016/j.addr.2003.10.007
    • L. F. Huang and W. Q. Tong, Impact of solid state properties on developability assessment of drug candidates, Adv. Drug Del. Rev. 56 (2004) 321-334; DOI: 10.1016/j.addr.2003.10.007.
    • (2004) Adv. Drug Del. Rev , vol.56 , pp. 321-334
    • Huang, L.F.1    Tong, W.Q.2
  • 4
    • 20344391910 scopus 로고    scopus 로고
    • Trends in solubility of polymorphs
    • DOI: 10.1002/jps.20302
    • M. Pudipeddi and A. T. M. Serajuddin, Trends in solubility of polymorphs, J. Pharm. Sci. 94 (2005) 929-939; DOI: 10.1002/jps.20302.
    • (2005) J. Pharm. Sci , vol.94 , pp. 929-939
    • Pudipeddi, M.1    Serajuddin, A.T.M.2
  • 5
    • 0037074108 scopus 로고    scopus 로고
    • The mechanisms of drug release from solid dispersions in water-soluble polymers
    • DOI: 10.1016/S0378-5173(01)00891-2
    • D. Q. M. Craig, The mechanisms of drug release from solid dispersions in water-soluble polymers, Int. J. Pharm. 231 (2002) 131-144; DOI: 10.1016/S0378-5173(01)00891-2.
    • (2002) Int. J. Pharm , vol.231 , pp. 131-144
    • Craig, D.Q.M.1
  • 6
    • 34548672900 scopus 로고    scopus 로고
    • A comparative assessment of solubility advantage from glassy and crystalline forms of a water-insoluble drug
    • DOI: 10.1016/j.ejps.2007.05.111
    • G. Chawla and A. K. Bansal, A comparative assessment of solubility advantage from glassy and crystalline forms of a water-insoluble drug, Eur. J. Pharm. Sci. 32 (2007) 45-57; DOI: 10.1016/j.ejps.2007.05.111.
    • (2007) Eur. J. Pharm. Sci , vol.32 , pp. 45-57
    • Chawla, G.1    Bansal, A.K.2
  • 7
    • 10844266571 scopus 로고
    • Kinetics of decomposition of irbesartan in aqueous solutions determined by high performance liquid chromatography
    • C. J. Mbah, Kinetics of decomposition of irbesartan in aqueous solutions determined by high performance liquid chromatography, Pharmazie 59 (1994) 920-922.
    • (1994) Pharmazie , vol.59 , pp. 920-922
    • Mbah, C.J.1
  • 8
    • 0036531002 scopus 로고    scopus 로고
    • Dissolution and phase transition of pharmaceutical compounds
    • DOI: 10.1016/S0022-0248(01)02282-5
    • E. Garcia, C. Hoff and S. Veesler, Dissolution and phase transition of pharmaceutical compounds, J. Crys. Growth 237-239 (2002) 2233-2239; DOI: 10.1016/S0022-0248(01)02282-5.
    • (2002) J. Crys. Growth , vol.237-239 , pp. 2233-2239
    • Garcia, E.1    Hoff, C.2    Veesler, S.3
  • 9
    • 0347995143 scopus 로고    scopus 로고
    • Phase transitions in supersaturated drug solution
    • DOI: 10.1021/op034089f
    • S. Veesler, L. Lafferrere, E. Garcia and C. Hoff, Phase transitions in supersaturated drug solution, Org. Process Res. Develop. 7 (2003) 983-989; DOI: 10.1021/op034089f.
    • (2003) Org. Process Res. Develop , vol.7 , pp. 983-989
    • Veesler, S.1    Lafferrere, L.2    Garcia, E.3    Hoff, C.4
  • 10
    • 0034886795 scopus 로고    scopus 로고
    • Physicochemical considerations in the preparation of amorphous ritonavir-poly(ethylene glycol) 8000 solid dispersions
    • DOI: 10.1002/jps.1054
    • B. Law, S. L. Krill, E. A. Schmitt, J. J. Fort, Y. Qiu, W. Wang and W. R. Porter, Physicochemical considerations in the preparation of amorphous ritonavir-poly(ethylene glycol) 8000 solid dispersions, J. Pharm. Sci. 90 (2001) 1015-1025; DOI: 10.1002/jps.1054.
    • (2001) J. Pharm. Sci , vol.90 , pp. 1015-1025
    • Law, B.1    Krill, S.L.2    Schmitt, E.A.3    Fort, J.J.4    Qiu, Y.5    Wang, W.6    Porter, W.R.7
  • 11
    • 33747033371 scopus 로고    scopus 로고
    • Development, characterization and stabilization of amorphous form of a low Tg drug
    • DOI: 10.1016/j.powtec.2006.05.012
    • V. B. Pokharkar, L. P. Mandpe, M. N. Padamwar, A. A. Ambike, K. R. Mahadik and A. Paradkar, Development, characterization and stabilization of amorphous form of a low Tg drug, Powder Technol. 167 (2006) 20-25; DOI: 10.1016/j.powtec.2006.05.012.
    • (2006) Powder Technol , vol.167 , pp. 20-25
    • Pokharkar, V.B.1    Mandpe, L.P.2    Padamwar, M.N.3    Ambike, A.A.4    Mahadik, K.R.5    Paradkar, A.6
  • 12
    • 0015124656 scopus 로고
    • Pharmaceutical applications of solid dispersion systems
    • DOI: 10.1002/jps.2600600902
    • W. L. Chiou and S. Riegelman, Pharmaceutical applications of solid dispersion systems, J. Pharm. Sci. 60 (1971) 1281-1302; DOI: 10.1002/jps.2600600902.
    • (1971) J. Pharm. Sci , vol.60 , pp. 1281-1302
    • Chiou, W.L.1    Riegelman, S.2
  • 13
    • 0031393654 scopus 로고    scopus 로고
    • Preparation and dissolution behavior of ethenzamide solid dispersions using various sugars as dispersion carriers
    • K. Danjo, T. Nakata and A. Otsuka, Preparation and dissolution behavior of ethenzamide solid dispersions using various sugars as dispersion carriers, Chem. Pharm. Bull. 45 (1997) 1840-1844.
    • (1997) Chem. Pharm. Bull , vol.45 , pp. 1840-1844
    • Danjo, K.1    Nakata, T.2    Otsuka, A.3
  • 14
    • 0035095847 scopus 로고    scopus 로고
    • Characterization of glass solutions of poorly water-soluble drugs produced by melt extrusion with hydrophilic amorphous polymers
    • DOI: 10.1211/0022357011775532
    • A. Forster, J. Hempenstall and T. Rades, Characterization of glass solutions of poorly water-soluble drugs produced by melt extrusion with hydrophilic amorphous polymers, J. Pharm. Pharmacol. 53 (2001) 303-315; DOI: 10.1211/0022357011775532.
    • (2001) J. Pharm. Pharmacol , vol.53 , pp. 303-315
    • Forster, A.1    Hempenstall, J.2    Rades, T.3
  • 15
    • 33748209143 scopus 로고    scopus 로고
    • Enhancement of dissolution profile by solid dispersion (kneading) technique
    • DOI: 10.1208/pt070368
    • A. Modi and P. Tayade, Enhancement of dissolution profile by solid dispersion (kneading) technique, AAPS PharmSciTech. 7 (2006) E1-E6; DOI: 10.1208/pt070368.
    • (2006) AAPS PharmSciTech , vol.7
    • Modi, A.1    Tayade, P.2
  • 16
    • 33746630521 scopus 로고    scopus 로고
    • Physicochemical characterization of meloxicam-mannitol binary systems
    • DOI: 10.1016/j.jpba.2006.02.055
    • P. R. Nassab, R. Rajko and P. S. Revesz, Physicochemical characterization of meloxicam-mannitol binary systems, J. Pharm. Biomed. Anal. 41 (2006) 1191-1197; DOI: 10.1016/j.jpba.2006.02.055.
    • (2006) J. Pharm. Biomed. Anal , vol.41 , pp. 1191-1197
    • Nassab, P.R.1    Rajko, R.2    Revesz, P.S.3
  • 17
    • 0041177972 scopus 로고    scopus 로고
    • Study by DSC and HSM of the oxazepam-PEG 6000 and oxazepam-D-mannitol systems: Application to the preparation of solid dispersions
    • DOI: 10.1016/S0040-6031(98)00437-7
    • M. J. Arias, J. R. Moyano and J. M. Gines, Study by DSC and HSM of the oxazepam-PEG 6000 and oxazepam-D-mannitol systems: Application to the preparation of solid dispersions, Thermochim. Acta 321 (1998) 33-41; DOI: 10.1016/S0040-6031(98)00437-7.
    • (1998) Thermochim. Acta , vol.321 , pp. 33-41
    • Arias, M.J.1    Moyano, J.R.2    Gines, J.M.3
  • 18
    • 0031845544 scopus 로고    scopus 로고
    • Thermal analysis as a screening technique in preformulation studies on picotinamide solid dosage forms
    • DOI: 10.3109/03639049809082722
    • P. Mura, M. T. Faucci, A. Manderioli, S. Furlanetto and S. Pinzauti, Thermal analysis as a screening technique in preformulation studies on picotinamide solid dosage forms, Drug Dev. Ind. Pharm. 24 (1998) 747-756; DOI: 10.3109/03639049809082722.
    • (1998) Drug Dev. Ind. Pharm , vol.24 , pp. 747-756
    • Mura, P.1    Faucci, M.T.2    Manderioli, A.3    Furlanetto, S.4    Pinzauti, S.5
  • 19
    • 0032915277 scopus 로고    scopus 로고
    • Development of a mathematical model for the water distribution in freeze-dried solids
    • DOI: 10.1023A: 1018812305562
    • H. K. Chan, K. L. Au-Yeung and I. Gonda, Development of a mathematical model for the water distribution in freeze-dried solids, Pharmacol. Res. 16 (1999) 660-665; DOI: 10.1023A: 1018812305562.
    • (1999) Pharmacol. Res , vol.16 , pp. 660-665
    • Chan, H.K.1    Au-Yeung, K.L.2    Gonda, I.3
  • 20
    • 3242706588 scopus 로고    scopus 로고
    • Phase behaviour analysis of solid dispersions of loperamide and two structurally related compounds with the polymers PVP-K30 and PVP-VA64
    • DOI: 10.1016/j.ejps.2004. 04.002
    • I. Weuts, D. Kempen, A. Decorte, G. Verreck, J. Peeters, M. Brewster and G. van den Mooter, Phase behaviour analysis of solid dispersions of loperamide and two structurally related compounds with the polymers PVP-K30 and PVP-VA64, Eur. J. Pharm. Sci. 22 (2004) 375-385; DOI: 10.1016/j.ejps.2004. 04.002.
    • (2004) Eur. J. Pharm. Sci , vol.22 , pp. 375-385
    • Weuts, I.1    Kempen, D.2    Decorte, A.3    Verreck, G.4    Peeters, J.5    Brewster, M.6    van den Mooter, G.7
  • 21
    • 0001106314 scopus 로고
    • Ideal copolymers and the second-order transitions of synthetic rubbers 1: Non-crystalline copolymers
    • M. Gordon and J. S. Taylor, Ideal copolymers and the second-order transitions of synthetic rubbers 1: Non-crystalline copolymers, J. Appl. Chem. 2 (1952) 493-498.
    • (1952) J. Appl. Chem , vol.2 , pp. 493-498
    • Gordon, M.1    Taylor, J.S.2
  • 22
    • 0031958399 scopus 로고    scopus 로고
    • Comparison of nicotinamide, ethylurea and polyethylene glycol as carriers for nifedipine solid dispersion systems
    • H. Suzuki and H. Sunada, Comparison of nicotinamide, ethylurea and polyethylene glycol as carriers for nifedipine solid dispersion systems, Chem. Pharm. Bull. 46 (1998) 482-487.
    • (1998) Chem. Pharm. Bull , vol.46 , pp. 482-487
    • Suzuki, H.1    Sunada, H.2
  • 23
    • 0036794236 scopus 로고    scopus 로고
    • Selection of suitable drug and excipient candidates to prepare glass solutions by melt extrusion for immediate release oral formulations
    • A. Forster, T. Rades and J. Hempenstall, Selection of suitable drug and excipient candidates to prepare glass solutions by melt extrusion for immediate release oral formulations, Pharm. Technol. (Europe) (2002) 27-37.
    • (2002) Pharm. Technol. (Europe , pp. 27-37
    • Forster, A.1    Rades, T.2    Hempenstall, J.3
  • 24
    • 45849111476 scopus 로고    scopus 로고
    • Dissolution rates and supersaturation behavior of amorphous repaglinide particles produced by controlled precipitation
    • DOI: 10.1166/jbn.2007.001
    • P. Sinswat, M. E. Matteucci, K. P. Johnston and R. O. Williams III, Dissolution rates and supersaturation behavior of amorphous repaglinide particles produced by controlled precipitation, J. Biomed. Nanotech. 3 (2007) 18-27; DOI: 10.1166/jbn.2007.001.
    • (2007) J. Biomed. Nanotech , vol.3 , pp. 18-27
    • Sinswat, P.1    Matteucci, M.E.2    Johnston, K.P.3    Williams III, R.O.4
  • 25
    • 0029047420 scopus 로고
    • Influence of the preparation method of solid dispersions on their dissolution rate: Study of triamterene-D-mannitol system
    • DOI: 10.1016/0378-5173(95)00026-F
    • M. J. Arias, J. M. Gines, J. R. Moyano, J. I. Perez-Martinez and A. M. Rabasco, Influence of the preparation method of solid dispersions on their dissolution rate: Study of triamterene-D-mannitol system, Int. J. Pharm. 123 (1995) 25-31; DOI: 10.1016/0378-5173(95)00026-F.
    • (1995) Int. J. Pharm , vol.123 , pp. 25-31
    • Arias, M.J.1    Gines, J.M.2    Moyano, J.R.3    Perez-Martinez, J.I.4    Rabasco, A.M.5


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.