Synthesis of 2-arylbenzimidazoles via microwave Suzuki-Miyaura reaction of unprotected 2-chlorobenzimidazoles

Tetrahedron Letters

Volumn 49, Issue 47, 2008, Pages 6667-6669

  Savall, Brad M ^a   Fontimayor, Jill R ^a  

^a JOHNSON AND JOHNSON PHARMACEUTICAL RESEARCH AND DEVELOPMENT   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

2 ARYLBENZIMIDAZOLE; 2 CHLOROBENZIMIDAZOLE; BENZIMIDAZOLE DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; CHEMICAL REACTION; MICROWAVE RADIATION; SUZUKI REACTION; SYNTHESIS;

EID: 53349162126     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.tetlet.2008.09.043     Document Type: Article

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12. 2 and dried under vacuum to yield 96 mg, 86% yield of 2-(4-methoxy-phenyl)-1H-benzimidazole.
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