Oxygenated chalcones and bischalcones as a new class of inhibitors of DNA topoisomerase II of malarial parasites

Medicinal Chemistry Research

Volumn 17, Issue 2-7, 2008, Pages 234-244

  Srivastava, Shalini ^a   Joshi, Shweta ^a   Singh, Alok R ^a   Yadav, Sarika ^a   Saxena, A S ^a   Ram, V J ^a   Chandra, Subhash ^a   Saxena, J K ^a  

^a CENTRAL DRUG RESEARCH INSTITUTE   (India)

Author keywords

Bischalcones; Chalcones; Chloroquine resistant strain; DNA; Plasmodium berghei; Topoisomerase inhibitors; Topoisomerases

Indexed keywords

CHALCONE DERIVATIVE; CHLOROQUINE; GYRASE INHIBITOR;

ANTIBIOTIC RESISTANCE; CONFERENCE PAPER; DRUG ACTIVITY; DRUG SYNTHESIS; ENZYME ACTIVITY; ENZYME INHIBITION; IN VITRO STUDY; IN VIVO STUDY; MALARIA; NONHUMAN; OXYGENATION; PARASITEMIA; PLASMODIUM BERGHEI; RODENT;

EID: 52949136697     PISSN: 10542523     EISSN: None     Source Type: Journal    
DOI: 10.1007/s00044-007-9057-0     Document Type: Conference Paper

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