Development and in-vitro evaluation of a colon-specific controlled release drug delivery system

Journal of Pharmacy and Pharmacology

Volumn 60, Issue 10, 2008, Pages 1297-1303

  Talukder, Rahmat M ^a   Fassihi, Reza ^b  

^a SOUTHWESTERN OKLAHOMA STATE UNIVERSITY   (United States)

^b TEMPLE UNIVERSITY   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ENZYME; HYDROXYPROPYLMETHYLCELLULOSE; MESALAZINE; MICROCRYSTALLINE CELLULOSE; PECTIN; PECTINOLYTIC ENZYME; PHOSPHATE BUFFERED SALINE; UNCLASSIFIED DRUG;

ARTICLE; COLON ABSORPTION; CONTROLLED RELEASE FORMULATION; DISSOLUTION; DRUG COATING; DRUG DELIVERY SYSTEM; DRUG DESIGN; DRUG RELEASE; DRUG SCREENING; DRUG STABILITY; DRUG TARGETING; ENTERIC COATED TABLET; INTESTINE TRANSIT TIME; PH;

EID: 52949110513     PISSN: 00223573     EISSN: None     Source Type: Journal    
DOI: 10.1211/jpp.60.10.0005     Document Type: Article

References (28)

1. Antonin, K. H., Sanno, V., Biek, P., Hastewell, J., Fox, R., Lowe, P., Mackay, M. (1992) Colonic absorption of human calcitonin in man. Clin. Sci. 83: 627-631
2. Ashford, M., Fell, T. J., Attwood, D., Woodhead, P. J. (1993) An in vitro investigation into the suitability of pH-dependent polymers for colon targeting. Int. J. Pharm. 91: 241-245
3. Basit, A. W. (2005) Advances in colonic drug delivery. Drugs 65: 1991-2007
4. Chourasia, M. K., Jain, S. K. (2003) Pharmaceutical approaches to colon targeted drug delivery systems.J. Pharm. Pharm. Sci. 6: 33-66
5. Coupe, A. J., Davis, S. S., Wilding, I. R. (1991) Variation in gastrointestinal transit of pharmaceutical dosage forms in healthy subjects. Pharm. Res. 8: 360-364
6. Davis, S. S., Hardy, J. G., Fara, J. W. (1986) Transit of pharmaceutical dosage forms through the small intestine. Gut 27: 886-892
7. Dressman, J. B., Amidon, G. L., Peppas, C., Shah, V. (1998) Dissolution testing a prognostic tool for oral drug absorption: immediate release dosage forms. Pharm. Res. 15: 11-22
8. Friend, D. R. (1991) Colon-specific drug delivery. Adv. Drug Deliv. Rev. 7: 149-199
9. Gustafsson, B. E. (1982) The physiological importance of the colonic microflora. Scand. J. Gastroenterol. 11 (Suppl.): 117-131
10. Hardy, J. G., Davis, S. S., Khosla, R., Robertson, C. S. (1988) Gastrointestinal transit of small tablets in patients with ulcerative colitis. Int. J. Pharm. 48: 79-82
11. Jamzad, S., Fassihi, R. (2006) Role of surfactant and pH on dissolution properties of fenofibrate and glipizide - a technical note. AAPS Pharm. Sci. Tech. 7: E33
12. Kaus, L. C., Fell, J.T. (1984) Effect of stress on the gastric emptying of capsules. J. Clin. Hosp. Pharm. 9: 249-251
13. Kim, H., Fassihi, R (1997) Application of binary polymer system in drug release rate modulation. 2. Influence of formulation variables and hydrodynamic conditions on release kinetics. J. Pharm. Sci. 86: 323-328
14. Moore, J. W., Flanner, H. H. (1996) Mathematical comparison of dissolution profiles. Pharm. Tech. 20: 64-74
15. Moore, W. E. C., Holdeman, L. V. (1975) Discussion of current bacteriologic investigations of the relationships between intestinal flora, diet, and colon cancer. Cancer Res. 35: 3418
16. Nyqvist, H. (1983) Saturated salt solutions for maintaining specified relative humidities. Int. J. Pharm. Tech. 4: 47-48
17. O'Donnell, P. B., McGinity, J.W. (1997) Mechanical properties of polymeric films prepared from aqueous polymeric dispersions. In: McGinity, J. B. (ed.) Aqueous polymeric coatings for pharmaceutical dosage forms. 2nd edn, Marcel Dekker, New York
18. Pillay, V., Fassihi, R. (1999) Evaluation and comparison of dissolution data derived from different modified release dosage forms: an alternative method. J. Control. Release 55: 45-55
19. Pozzi, F., Furlani, P., Gazzaniga, A., Davis, S. S., Wilding, I. R. (1994) The TIME-CLOCK System: a new oral dosage form for fast and complete release of drug after predetermined lag time. J. Control. Release 31: 99-108
20. Reddy, S. M., Sinha, V. R., Reddy, D. S. (1999) Novel oral colon-specific drug delivery systems for pharmacotherapy of peptide and nonpeptide drugs. Drugs Today 35: 537-580
21. Rohera, B. D., Parikh, N. H. (2002) Influence of type and level of water-soluble additives on drug release and surface and mechanical properties of surelease films. Pharm. Dev. Technol. 7: 421-432
22. Rubinstein, A. (1990) Microbially controlled drug delivery to the colon. Biopharm. Drug Dispos. 11: 465-475
23. Saffran, M., Kumar, G. S., Savariar, C., Burnham, J. C., Williams, F., Neckers, D. C. (1986) A new approach to the oral administration of insulin and other peptide drugs. Science 233: 1081-1084
24. Sakellariou, P., Rowe, R. C., White, J. D. (1986) An evaluation of the interaction and plasticizing efficiency of the polyethylene glycols in ethylcellulose and hydroxypropyl methylcellulose films using the torsional braid pendulum. Int. J. Pharm. 31: 55-64
25. Theeuwes, F., Guittard, G. V., Wong, G. V, Patrick. S. L. (1990) Delivery of drug to colon by oral dosage form. US Patent # 4904474
26. Tozar, N. T., Friend, D. R., Mcleod, A. D. (1995) Kinetic perspectives on colonic delivery. STP Pharma Sci. 5: 5-12
27. Van den Mooter, G. (2006) Colon drug delivery. Expert Opin. Drug Deliv. 3: 111-125
28. Youan, B. B. C. (2004) Chronotherapeutics: gimmick or clinically relevant approach to drug delivery. J. Control. Release 98: 337-353