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Volumn 6, Issue 18, 2008, Pages 3399-3407

Bioisosteric replacement of the pyrazole 3-carboxamide moiety of rimonabant. A novel series of oxadiazoles as CB1 cannabinoid receptor antagonists

(9) Chu, Cheng Ming a Hung, Ming Shiu a Hsieh, Min Tsang a Kuo, Chun Wei a Suja, T D a Song, Jen Shin a Chiu, Hua Hao a Chao, Yu Sheng a Shia, Kak Shan a

a NATIONAL HEALTH RESEARCH INSTITUTES (Taiwan)

Author keywords

[No Author keywords available]

Indexed keywords

ARSENIC COMPOUNDS; CHLORINE COMPOUNDS; DERIVATIVES;

BIOLOGICAL ACTIVITIES; CARBOXAMIDE; ELECTRON-WITHDRAWING GROUPS; NOVEL SERIES; OXADIAZOLE; OXADIAZOLE DERIVATIVES; OXADIAZOLES; PYRAZOLE; RECEPTOR ANTAGONISTS; RIMONABANT;

ALKYLATION;

AMIDE; CANNABINOID 1 RECEPTOR; CANNABINOID 2 RECEPTOR; PIPERIDINE DERIVATIVE; PYRAZOLE; PYRAZOLE DERIVATIVE; RIMONABANT;

ARTICLE; CELL LINE; CHEMICAL STRUCTURE; CHEMISTRY; DRUG ANTAGONISM; HUMAN; ISOMERISM; METABOLISM; STRUCTURE ACTIVITY RELATION;

AMIDES; CELL LINE; HUMANS; ISOMERISM; MOLECULAR STRUCTURE; PIPERIDINES; PYRAZOLES; RECEPTOR, CANNABINOID, CB1; RECEPTOR, CANNABINOID, CB2; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 52649148140 PISSN: 14770520 EISSN: None Source Type: Journal
DOI: 10.1039/b807648k Document Type: Article

Times cited : (17)

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