Synthesis and activity of 1-(3-amino-1-phenylpropyl)indolin-2-ones: A new class of selective norepinephrine reuptake inhibitors

Bioorganic and Medicinal Chemistry Letters

Volumn 18, Issue 18, 2008, Pages 4929-4931

  McComas, Casey C ^a   Vu, An T ^a   Mahaney, Paige E ^a   Cohn, Stephen T ^a   Fensome, Andrew ^a   Marella, Michael A ^a   Nogle, Lisa ^a   Trybulski, Eugene J ^a   Ye, Fei ^a   Zhang, Puwen ^a   Alfinito, Peter ^a   Bray, Jenifer ^a   Johnston, Grace ^a   Koury, Elizabeth ^a   Deecher, Darlene C ^a  

^a PFIZER INC   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

DOPAMINE TRANSPORTER; FLUOXETINE; INDOLE DERIVATIVE; NORADRENALIN; NORADRENALIN UPTAKE INHIBITOR; SEROTONIN TRANSPORTER;

ANIMAL CELL; ARTICLE; BINDING AFFINITY; CONTROLLED STUDY; DRUG ACTIVITY; DRUG BINDING; DRUG STRUCTURE; DRUG SYNTHESIS; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; HUMAN; HUMAN CELL; NONHUMAN;

HUMANS; INDOLES; MOLECULAR STRUCTURE; NEUROTRANSMITTER UPTAKE INHIBITORS; NOREPINEPHRINE; STEREOISOMERISM; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 51349157965     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2008.08.060     Document Type: Article

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