Discovery of novel and long acting muscarinic acetylcholine receptor antagonists

Journal of Medicinal Chemistry

Volumn 51, Issue 16, 2008, Pages 4866-4869

  Jin, Jian ^a,b   Wang, Yonghui ^a   Shi, Dongchuan ^a   Wang, Feng ^a   Davis, Roderick S ^a   Jin, Qi ^a   Fu, Wei ^a   Foley, James J ^a   Webb, Edward F ^a   Dehaas, Chris J ^a   Berlanga, Manuela ^a   Burman, Miriam ^a   Sarau, Henry M ^a   Morrow, Dwight M ^a   Rao, Parvathi ^a   Kallal, Lorena A ^a   Moore, Michael L ^a   Rivero, Ralph A ^a   Palovich, Michael ^a   Salmon, Michael ^a   Belmonte, Kristen E ^a   Busch Petersen, Jakob ^a   more..

^a GLAXOSMITHKLINE   (United States)

^b University of North Carolina   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

MUSCARINIC RECEPTOR BLOCKING AGENT; QUATERNARY AMMONIUM DERIVATIVE;

ANIMAL EXPERIMENT; ANIMAL MODEL; ARTICLE; BRONCHOSPASM; CHRONIC OBSTRUCTIVE LUNG DISEASE; CONTROLLED STUDY; DRUG ACTIVITY; DRUG POTENCY; DRUG SELECTIVITY; GUINEA PIG; HIGH THROUGHPUT SCREENING; IN VIVO STUDY; MOUSE; NONHUMAN; RAT; SINGLE DRUG DOSE;

ANIMALS; BICYCLO COMPOUNDS, HETEROCYCLIC; BRONCHOCONSTRICTION; DRUG EVALUATION, PRECLINICAL; GUINEA PIGS; MICE; MUSCARINIC ANTAGONISTS; PHENYLUREA COMPOUNDS; QUATERNARY AMMONIUM COMPOUNDS; RATS; TYROSINE;

EID: 50249177032     PISSN: 00222623     EISSN: None     Source Type: Journal    
DOI: 10.1021/jm800634k     Document Type: Article

References (18)

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