Formation of shellac succinate having improved enteric film properties through dry media reaction

European Journal of Pharmaceutics and Biopharmaceutics

Volumn 70, Issue 1, 2008, Pages 335-344

  Limmatvapirat, Sontaya ^a   Panchapornpon, Danuch ^a   Limmatvapirat, Chutima ^a   Nunthanid, Jurairat ^a   Luangtana Anan, Manee ^a   Puttipipatkhachorn, Satit ^b  

^a SILPAKORN UNIVERSITY   (Thailand)

^b MAHIDOL UNIVERSITY   (Thailand)

Author keywords

Co grinding; Enteric polymer; Mechanochemistry; Shellac; Shellac succinate

Indexed keywords

CARBOXYLIC ACID DERIVATIVE; SHELLAC; SHELLAC SUCCINATE; SUCCINIC ACID DERIVATIVE; SUCCINIC ANHYDRIDE; UNCLASSIFIED DRUG;

ARTICLE; CARBON NUCLEAR MAGNETIC RESONANCE; CHEMICAL REACTION; DIFFERENTIAL SCANNING CALORIMETRY; DRUG FORMULATION; DRUG SOLUBILITY; ENTERIC COATED TABLET; ESTERIFICATION; FILM; HEATING; INFRARED SPECTROSCOPY; MECHANICS; PH; PROTON NUCLEAR MAGNETIC RESONANCE; SOLID STATE; THERMAL ANALYSIS;

CALORIMETRY, DIFFERENTIAL SCANNING; CHEMISTRY, PHARMACEUTICAL; DOSAGE FORMS; HYDROGEN-ION CONCENTRATION; MAGNETIC RESONANCE SPECTROSCOPY; PERMEABILITY; PLIABILITY; RESINS, PLANT; SOLUBILITY; SPECTROSCOPY, FOURIER TRANSFORM INFRARED; SUCCINIC ANHYDRIDES; TECHNOLOGY, PHARMACEUTICAL; TRANSITION TEMPERATURE; VOLATILIZATION; WATER;

EID: 50249117640     PISSN: 09396411     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.ejpb.2008.03.002     Document Type: Article

References (41)

1. Porter S.C. In: Lieberman H.A. (Ed). Pharmaceutical Dosage Forms: Tablet vol. 1 (1990), Marcel Dekker, New York 77-160
2. Banker G.S., and Agyilirah G.A. In: Tarcha P.J. (Ed). Polymers for Controlled Drug Delivery (1999), CRC Press, London 39-66
3. Pearnchob N., Siepmann J., and Bodmeier R. Pharmaceutical applications of shellac: moisture-protective and taste-masking coatings and extended-release matrix tablets. Drug Dev. Ind. Pharm. 29 8 (2003) 925-938
4. Pearnchob N., Dashevsky A., and Bodmeier R. Improvement in the disintegration of shellac-coated soft gelatin capsules in simulated intestinal fluid. J. Control Release 94 2-3 (2004) 313-321
5. Hogan J.E. In: Cole G., Hogan J.E., and Aulton M. (Eds). Pharmaceutical Coating Technology (1995), Taylor & Francis Books, London 409-438
6. Hogan J.E. In: Cole G., Hogan J.E., and Aulton M. (Eds). Pharmaceutical Coating Technology (1995), Taylor & Francis Books, London 6-52
7. Carstensen J.T. Advanced Pharmaceutical Solids (2001), Marcel Dekker, New York
8. Dressman J.B., and Palsson B.Ø. In: Ghebre-Sellassie I. (Ed). Multiparticulate Oral Drug Delivery (1994), Marcel Dekker, New York 285-306
9. Li X., and Vasavada R.C. In: Rowe R.C., Sheskey P.J., and Weller P.J. (Eds). Handbook of Pharmaceutical Excipients (2003), Pharmaceutical Press, London 538-540
10. Limmatvapirat S., Limmatvapirat C., Luangtana-Anan M., Nunthanid J., Oguchi T., Tozuka Y., Yamamoto K., and Puttipipatkhachorn S. Modification of physicochemical and mechanical properties of shellac by partial hydrolysis. Int. J. Pharm. 278 1 (2004) 41-49
11. Limmatvapirat S., Nunthanid J., Luangtana-anan M., and Puttipipatkhachorn S. Effect of alkali treatment on properties of native shellac and stability of hydrolyzed shellac. Pharm. Dev. Technol. 10 1 (2005) 41-46
12. Specht F., Saugested M., Waaler T., and Müller B.W. The application of shellac as an acidic polymer for enteric coating. Pharm. Tech. 10 (1998) 20-28
13. Limmatvapirat S., Limmatvapirat C., Puttipipatkhachorn S., Nuntanid J., and Luangtana-anan M. Enhanced enteric properties and stability of shellac films through composite salts formation. Eur. J. Pharm. Biopharm. 67 3 (2007) 690-698
14. Luangtana-Anan M., Limmatvapirat S., Nunthanid J., Wanawongthai C., Chalongsuk R., and Puttipipatkhachorn S. Effect of salts and plasticizers on stability of shellac film. J. Agric. Food Chem. 55 3 (2007) 687-692
15. Kokubo H., Obara S., Minemura K., and Tanaka T. Development of cellulose derivatives as novel enteric coating agents soluble at pH 3.5-4.5 and higher. Chem. Pharm. Bull. 45 8 (1997) 1350-1353
16. Kidwai M. Dry media reactions. Pure Appl. Chem. 73 1 (2001) 147-151
17. S. Mallick, S. Pattnaik, K. Swain, P.K. De, A. Saha, G. Ghoshal, A. Mondal, Formation of physically stable amorphous phase of ibuprofen by solid state milling with kaolin, Eur. J. Pharm. Sci. 8(2) 346-351.
18. Limmatvapirat S., Yonemochi E., Oguchi T., and Yamamoto K. Mechanochemical complexation between deoxycholic acid and salicylic acid. J. Incl. Phenom. 31 (1998) 367-379
19. Oguchi T., Kazama K., Fukami T., Yonemochi E., and Yamamoto K. Specific complexation of ursodeoxycholic acid with guest compounds induced by co-grinding. II. Effect of grinding temperature on the mechanochemical complexation. Bull. Chem. Soc. Jpn. 76 (2003) 515-521
20. Constabel F., and Geckeler K.E. Solvent-free self-assembly of C60 and cucurbit[7]uril using high-speed vibration milling. Tetrahedron Lett. 45 10 (2004) 2071-2073
21. USP 29, US Pharmacopeial Convention, Rockville, MD, 2006, p. 3417.
22. Sungthongjeen S., Puttipipatkhachorn S., Paeratakul O., Dashevsky A., and Bodmeier R. Development of pulsatile release tablets with swelling and rupturable layers. J. Control Release 95 2 (2004) 147-159
23. Ciper M., and Bodmeier R. Preparation and characterization of novel fast disintegrating capsules (Fastcaps) for administration in the oral cavity. Int. J. Pharm. 303 1-2 (2005) 62-71
24. Wu S.H.W., Wyatt D.M., and Adams M.W. In: McGinity J.W. (Ed). Aqueous polymeric coatings for pharmaceutical dosage forms (1997), Marcel Dekker, New York 385-418
25. Bhandari P.N., and Singhal R.S. Studies on the optimisation of preparation of succinate derivatives from corn and amaranth starches. Carbohydr. Polym. 47 3 (2002) 277-283
26. Aiedeh K., and Taha M.O. Synthesis of iron-crosslinked chitosan succinate and iron-crosslinked hydroxamated chitosan succinate and their in vitro evaluation as potential matrix materials for oral theophylline sustained-release beads. Eur. J. Pharm. Sci. 13 2 (2001) 159-168
27. Sun X.F., Sun R.C., Tomkinson J., and Baird M.S. Preparation of sugarcane bagasse hemicellulosic succinates using NBS as a catalyst. Carbohydr. Polym. 53 4 (2003) 483-495
28. Ortega-Aviles M., Vandenabeele P., Tenorio D., Murillo G., Jimenez-Reyes M., and Gutierrez N. Spectroscopic investigation of a 'Virgin of Sorrows' canvas painting: a multi-method approach. Anal. Chim. Acta 550 1-2 (2005) 164-172
29. Silverstein R.M., Bassler G.C., and Morrill T.C. Spectrometric identification of organic compounds (1991), John Wiley & Sons, Inc., New York
30. Akhgari A., Farahmand F., Afrasiabi Garekani H., Sadeghi F., and Vandamme T.F. Permeability and swelling studies on free films containing inulin in combination with different polymethacrylates aimed for colonic drug delivery. Eur. J. Pharm. Sci. 28 4 (2006) 307-314
31. Rao P.R., and Diwan P.V. Permeability studies of cellulose acetate free films for transdermal use: influence of plasticizers. Pharm. Acta Helv. 72 1 (1997) 47-51
32. Krogars K., Heinamaki J., Karjalainen M., Niskanen A., Leskela M., and Yliruusi J. Enhanced stability of rubbery amylose-rich maize starch films plasticized with a combination of sorbitol and glycerol. Int. J. Pharm. 251 1-2 (2003) 205-208
33. Liu J., and Williams R.O. Properties of heat-humidity cured cellulose acetate phthalate free films. Eur. J. Pharm. Sci. 17 1-2 (2002) 31-41
34. Shin-Etsu, Shin-Etsu AQOAT (product catalogue), 2007.
35. Shin-Etsu, HPMCP (product catalogue), 2007.
36. Heng P.W.S., Chan L.W., and Ong K.T. Influence of storage conditions and type of plasticizers on ethylcellulose and acrylate films formed from aqueous dispersions. J. Pharm. Pharm. Sci. 6 3 (2003) 334-344
37. Qussi B., and Suess W.G. The influence of different plasticizers and polymers on the mechanical and thermal properties, porosity and drug permeability of free shellac films. Drug Dev. Ind. Pharm. 32 4 (2006) 403-412
38. Qussi B., and Suess W.G. Investigation of the effect of various shellac coating compositions containing different water-soluble polymers on in vitro drug release. Drug Dev. Ind. Pharm. 31 1 (2005) 99-108
39. Aulton M.E. In: Cole G., Hogan J.E., and Aulton M. (Eds). Pharmaceutical Coating Technology (2002), Taylor & Francis Books, London 288-362
40. Wu C., and McGinity J.W. Influence of relative humidity on the mechanical and drug release properties of theophylline pellets coated with an acrylic polymer containing methylparaben as a non-traditional plasticizer. Eur. J. Pharm. Biopharm. 50 2 (2000) 277-284
41. Huang Y., Zheng L.L., Liu J., and Zhang Z.R. Synthesis and characterization of HPMC derivatives as novel duodenum-specific coating agents. Arch. Pharm. Res. 28 3 (2005) 364-369