Preparation of a set of 4,5-dihydro-3H-pyrrolo[3,2-d]pyrimidin-4-ones as potential Hsp90 ligands

Tetrahedron Letters

Volumn 49, Issue 41, 2008, Pages 5965-5967

  Semeraro, Teresa ^a   Mugnaini, Claudia ^a   Corelli, Federico ^a  

^a UNIVERSITY OF SIENA   (Italy)

Author keywords

Deazapurines; Hsp90 ligands; Pyrrolo 3,2 d pyrimidin 4 ones

Indexed keywords

4,5 DIHYDRO 3H PYRROLO[3,2 D]PYRIMIDIN 4 ONE; HEAT SHOCK PROTEIN 90; LIGAND; PYRIMIDINE DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; CHEMICAL REACTION; CHEMICAL STRUCTURE; POLYMERIZATION; SYNTHESIS;

EID: 50049134595     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.tetlet.2008.07.158     Document Type: Article

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11. 2: C, 68.83; H, 6.60; N, 11.47. Found: C, 68.98; H, 6.58; N, 11.46.
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13. 4: C, 46.96; H, 4.19; N, 13.69. Found: C, 46.75; H, 4.27; N, 13.91.