α,α-cyclopentaneglycine dipeptides capped with biaryls as tachykinin NK2 receptor antagonists

ChemMedChem

Volumn 3, Issue 7, 2008, Pages 1048-1060

  Porcelloni, Marina ^a   D'Andrea, Piero ^a   Rossi, Cristina ^a   Sisto, Alessandro ^a   Ettorre, Alessandro ^a   Madami, Andrea ^a   Altamura, Maria ^b   Giuliani, Sandro ^b   Meini, Stefania ^b   Fattori, Daniela ^a  

^a Chemistry Department   (Italy)

^b Chemistry and Pharmacology Departments   (Italy)

Author keywords

GPCRs; NK2; Peptides; Receptors; Tachykinin

Indexed keywords

BENZOTHIOPHENE; BIPHENYL DERIVATIVE; CYCLOPENTANE DERIVATIVE; DIPEPTIDE; DRUG DERIVATIVE; GLYCINE; NEUROKININ 2 RECEPTOR; THIOPHENE DERIVATIVE;

ANIMAL; ARTICLE; BINDING COMPETITION; CELL MEMBRANE; CHEMISTRY; COLON; DRUG ANTAGONISM; DRUG EFFECT; GUINEA PIG; METABOLISM; MUSCLE CONTRACTION; PHYSIOLOGY; SYNTHESIS;

ANIMALS; BINDING, COMPETITIVE; BIPHENYL COMPOUNDS; CELL MEMBRANE; COLON; CYCLOPENTANES; DIPEPTIDES; GLYCINE; GUINEA PIGS; MUSCLE CONTRACTION; RECEPTORS, NEUROKININ-2; THIOPHENES;

EID: 48649108713     PISSN: 18607179     EISSN: 18607187     Source Type: Journal    
DOI: 10.1002/cmdc.200800018     Document Type: Article

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