Structure-activity relationship studies of permeability modulating peptide AT-1002

Bioorganic and Medicinal Chemistry Letters

Volumn 18, Issue 16, 2008, Pages 4584-4586

  Li, Min ^a   Oliver, Ed ^a   Kitchens, Kelly M ^a   Vere, John ^a   Alkan, Sefik S ^a   Tamiz, Amir P ^a  

^a Alba Therapeutics Corporation   (United States)

Author keywords

Drug delivery; Paracellular permeability; Peptide; Structure activity relationship studies

Indexed keywords

AT 1002; CYSTEINE; PEPTIDE DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; CONTROLLED STUDY; DRUG PENETRATION; DRUG STABILITY; HUMAN; HUMAN CELL; MODULATION; STRUCTURE ACTIVITY RELATION;

AMINO ACIDS; BIOLOGICAL TRANSPORT; CACO-2 CELLS; CELL SURVIVAL; CHEMISTRY, PHARMACEUTICAL; CHROMATOGRAPHY, HIGH PRESSURE LIQUID; CYSTEINE; DRUG DELIVERY SYSTEMS; DRUG DESIGN; HUMANS; MODELS, CHEMICAL; OLIGOPEPTIDES; PEPTIDES; PERMEABILITY; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 48649099527     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2008.07.028     Document Type: Article

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