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Volumn 107, Issue 2, 2008, Pages 151-158

Long-lasting anti-emetic effect of T-2328, a novel NK1 antagonist

Author keywords

Cisplatin; Emesis; Long acting; NK1

Indexed keywords

2 FLUORO 4' METHOXY 3' [[(2 PHENYL 3 PIPERIDINYL)AMINO]METHY](1,1' BIPHENYL) 4 CARBONITRILE; 5 AMINOVALERYLSUBSTANCE P [7-11][9 PROLINE 10 (N METHYLLEUCINE)]; CISPLATIN; NEUROKININ 1 RECEPTOR; NEUROKININ 1 RECEPTOR AGONIST; NEUROKININ 1 RECEPTOR ANTAGONIST; ONDANSETRON; SUBSTANCE P; T 2328;

EID: 46449084301     PISSN: 13478613     EISSN: 13478648     Source Type: Journal    
DOI: 10.1254/jphs.08027FP     Document Type: Article
Times cited : (9)

References (15)
  • 1
    • 33645111467 scopus 로고    scopus 로고
    • Emerging drugs for chemotherapy-induced emesis
    • Navari RM, Province PS. Emerging drugs for chemotherapy-induced emesis. Expert Opin Emerg Drugs. 2006;11:137-151.
    • (2006) Expert Opin Emerg Drugs , vol.11 , pp. 137-151
    • Navari, R.M.1    Province, P.S.2
  • 3
    • 21344451918 scopus 로고    scopus 로고
    • Optimising antiemetic therapy: What are the problems and how can they be overcome?
    • Aapro M. Optimising antiemetic therapy: what are the problems and how can they be overcome? Curr Med Res Opin. 2005;21:885-897.
    • (2005) Curr Med Res Opin , vol.21 , pp. 885-897
    • Aapro, M.1
  • 4
    • 0038730808 scopus 로고    scopus 로고
    • 1 receptor in the brainstem in the development of emesis
    • 1 receptor in the brainstem in the development of emesis. J Pharmacol Sci. 2003;91:87-94.
    • (2003) J Pharmacol Sci , vol.91 , pp. 87-94
    • Saito, R.1    Takano, Y.2    Kamiya, H.O.3
  • 5
    • 0029065938 scopus 로고
    • The anti-emetic effects of CP-99,994 in the ferret and the dog: Role of the NK1 receptor
    • Watson JW, Gonsalves SF, Fossa AA, McLean S, Seeger T, Obach S, et al. The anti-emetic effects of CP-99,994 in the ferret and the dog: role of the NK1 receptor. Br J Pharmacol. 1995;115:84-94.
    • (1995) Br J Pharmacol , vol.115 , pp. 84-94
    • Watson, J.W.1    Gonsalves, S.F.2    Fossa, A.A.3    McLean, S.4    Seeger, T.5    Obach, S.6
  • 7
    • 0030299823 scopus 로고    scopus 로고
    • Tachykinin NK1 receptor antagonists act centrally to inhibit emesis induced by the chemotherapeutic agent cisplatin in ferrets
    • Tattersall FD, Rycroft W, Francis B, Pearce D, Merchant K, MacLeod AM, et al. Tachykinin NK1 receptor antagonists act centrally to inhibit emesis induced by the chemotherapeutic agent cisplatin in ferrets. Neuropharmacology. 1996;35:1121-1129.
    • (1996) Neuropharmacology , vol.35 , pp. 1121-1129
    • Tattersall, F.D.1    Rycroft, W.2    Francis, B.3    Pearce, D.4    Merchant, K.5    MacLeod, A.M.6
  • 8
    • 0032476067 scopus 로고    scopus 로고
    • Anti-emetic effects of a novel NK-1 receptor antagonist HSP-117 in ferrets
    • Saito R, Suehiro Y, Ariumi H, Migita K, Hori N, Hashiguchi T, et al. Anti-emetic effects of a novel NK-1 receptor antagonist HSP-117 in ferrets. Neurosci Lett. 1998;254:169-172.
    • (1998) Neurosci Lett , vol.254 , pp. 169-172
    • Saito, R.1    Suehiro, Y.2    Ariumi, H.3    Migita, K.4    Hori, N.5    Hashiguchi, T.6
  • 9
    • 0033625089 scopus 로고    scopus 로고
    • The novel NK1 receptor antagonist MK-0869 (L-754,030) and its water soluble phosphoryl prodrug, L-758,298, inhibit acute and delayed cisplatin-induced emesis in ferrets
    • Tattersall FD, Rycroft W, Cumberbatch M, Mason G, Tye S, Williamson DJ, et al. The novel NK1 receptor antagonist MK-0869 (L-754,030) and its water soluble phosphoryl prodrug, L-758,298, inhibit acute and delayed cisplatin-induced emesis in ferrets. Neuropharmacology. 2000;39:652-663.
    • (2000) Neuropharmacology , vol.39 , pp. 652-663
    • Tattersall, F.D.1    Rycroft, W.2    Cumberbatch, M.3    Mason, G.4    Tye, S.5    Williamson, D.J.6
  • 10
    • 0347816226 scopus 로고    scopus 로고
    • The oral neurokinin-1 antagonist aprepitant for the prevention of chemotherapy-induced nausea and vomiting: A multinational, randomized, double-blind, placebo-controlled trial in patients receiving high-dose cisplatin - the Aprepitant Protocol 052 Study Group
    • Hesketh PJ, Grunberg SM, Gralla RJ, War DG, Roila F, de Wit R, et al. The oral neurokinin-1 antagonist aprepitant for the prevention of chemotherapy-induced nausea and vomiting: a multinational, randomized, double-blind, placebo-controlled trial in patients receiving high-dose cisplatin - the Aprepitant Protocol 052 Study Group. J Clin Oncol. 2003;21:4112-4119.
    • (2003) J Clin Oncol , vol.21 , pp. 4112-4119
    • Hesketh, P.J.1    Grunberg, S.M.2    Gralla, R.J.3    War, D.G.4    Roila, F.5    de Wit, R.6
  • 11
    • 0038728753 scopus 로고    scopus 로고
    • Addition of the neurokinin 1 receptor antagonist aprepitant to standard antiemetic therapy improves control of chemotherapy-induced nausea and vomiting. Results from a randomized, double-blind, placebo-controlled trial in Latin America
    • Poli-Bigelli S, Rodrigues-Pereira J, Carides AD, Julie Ma G, Eldridge K, Hipple A, et al. Addition of the neurokinin 1 receptor antagonist aprepitant to standard antiemetic therapy improves control of chemotherapy-induced nausea and vomiting. Results from a randomized, double-blind, placebo-controlled trial in Latin America. Cancer. 2003;97:3090-3098.
    • (2003) Cancer , vol.97 , pp. 3090-3098
    • Poli-Bigelli, S.1    Rodrigues-Pereira, J.2    Carides, A.D.3    Julie Ma, G.4    Eldridge, K.5    Hipple, A.6
  • 13
    • 0029658238 scopus 로고    scopus 로고
    • The action of the NK1 tachykinin receptor antagonist, CP 99,994, in antagonizing the acute and delayed emesis induced by cisplatin in the ferret
    • Rudd JA, Jordan CC, Naylor RJ. The action of the NK1 tachykinin receptor antagonist, CP 99,994, in antagonizing the acute and delayed emesis induced by cisplatin in the ferret. Br J Pharmacol. 1996;119:931-936.
    • (1996) Br J Pharmacol , vol.119 , pp. 931-936
    • Rudd, J.A.1    Jordan, C.C.2    Naylor, R.J.3
  • 14
    • 0028113481 scopus 로고
    • Differential inhibition of foot tapping and chromodacryorrhoea in gerbils by CNS penetrant and non-penetrant tachykinin NK1 receptor antagonists
    • Rupniak NM, Williams AR. Differential inhibition of foot tapping and chromodacryorrhoea in gerbils by CNS penetrant and non-penetrant tachykinin NK1 receptor antagonists. Eur J Pharmacol. 1994;265:179-183.
    • (1994) Eur J Pharmacol , vol.265 , pp. 179-183
    • Rupniak, N.M.1    Williams, A.R.2
  • 15
    • 0002709945 scopus 로고
    • The clinical approach to chemotherapy-induced emesis
    • Reynolds DJM, Andrews PLR, Davis CJ, editors, Oxford: Oxford Clinical Communications;
    • Gralla, RJ. The clinical approach to chemotherapy-induced emesis. In: Reynolds DJM, Andrews PLR, Davis CJ, editors. Serotonin and the scientific basis of anti-emetic therapy. Oxford: Oxford Clinical Communications; 1995. p. 60-67.
    • (1995) Serotonin and the scientific basis of anti-emetic therapy , pp. 60-67
    • Gralla, R.J.1


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.