5-Carboxamido-1,3,2-dioxaphosphorinanes, potent inhibitors of MTP

Bioorganic and Medicinal Chemistry Letters

Volumn 14, Issue 20, 2004, Pages 5067-5070

  Sulsky, Richard ^a   Robl, Jeffrey A ^a   Biller, Scott A ^a   Harrity, Thomas W ^a   Wetterau, John ^a   Connolly, Fergal ^a   Jolibois, Kern ^a   Kunselman, Lori ^a  

^a BRISTOL MYERS SQUIBB   (United States)

Author keywords

Cyclophosphonates; MTP inhibitors

Indexed keywords

1,3,2 DIOXAPHOSPHORINANE DERIVATIVE; BMS 201038; MICROSOMAL TRIGLYCERIDE TRANSFER PROTEIN INHIBITOR; PIPERIDINE; PIPERIDINE N OXIDE; UNCLASSIFIED DRUG;

ARTICLE; DRUG EFFICACY; DRUG IDENTIFICATION; DRUG POTENCY; DRUG STRUCTURE; DRUG SYNTHESIS; HEPATOMA CELL; HUMAN; HUMAN CELL; NONHUMAN;

AMIDES; ANIMALS; BENZIMIDAZOLES; CARRIER PROTEINS; CRICETINAE; CYCLIC P-OXIDES; HUMANS; MALE; STEREOISOMERISM; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 4544385608     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2004.07.069     Document Type: Article

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