메뉴 건너뛰기




Volumn 21, Issue 2, 2008, Pages 113-120

Formulation development and optimization of ibuprofen tablets by direct compression method

Author keywords

Direct compression; Ibuprofen; Independent variables; Optimization; Response variables

Indexed keywords

CROSPOVIDONE; DILUENT; DISINTEGRATING AGENT; IBUPROFEN; LUBRICATING AGENT; MAGNESIUM STEARATE; MICROCRYSTALLINE CELLULOSE; CELLULOSE; NONSTEROID ANTIINFLAMMATORY AGENT; POVIDONE; STEARIC ACID; STEARIC ACID DERIVATIVE;

EID: 44449171518     PISSN: 1011601X     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article
Times cited : (47)

References (43)
  • 1
    • 23944512870 scopus 로고    scopus 로고
    • Nitro-arginine methyl ester, a non-selective inhibitor of nitric oxide synthase reduces ibuprofen-induced gastric mucosal injury in the rat
    • DOI 10.1007/s10620-005-2908-y
    • Abraham P and KI KD (2005). Nitro-arginine methyl ester, a non-selective inhibitor of nitric oxide synthase reduces Ibuprofen-induced gastric mucosal injury in the rat. Dig. Dis., 50(9): 1632-1640. (Pubitemid 41203655)
    • (2005) Digestive Diseases and Sciences , vol.50 , Issue.9 , pp. 1632-1640
    • Abraham, P.1    Indirani, K.2    Desigamani, K.3
  • 2
    • 22544452289 scopus 로고    scopus 로고
    • Lippincott Williams And Wilkins, A Wolters Kluwer company, Philadelphia, Baltimore
    • th ed., Lippincott Williams And Wilkins, A Wolters Kluwer company, Philadelphia, Baltimore, pp.227-259.
    • (2005) th Ed. , pp. 227-259
    • Allen, L.V.1    Popvich, N.G.2    Ansel, H.C.3
  • 3
    • 70349845026 scopus 로고    scopus 로고
    • Swarbrick J and Boylan JC (editors). Marcel Dekker, Inc., New York, Basel
    • nd edn., Vol.03, Marcel Dekker, Inc., New York, Basel, p.2723.
    • (2002) nd Edn. , vol.3 , pp. 2723
    • Armstrong, N.A.1
  • 4
    • 0034817174 scopus 로고    scopus 로고
    • The prediction, morphology, and mechanical properties of the polymorphs of paracetamol
    • DOI 10.1021/ja0102787
    • Beyer T, Day GM and Price SL (2001). The prediction, morphology and mechanical properties of the polymorphs of Paracetamol. J. Am. Chem. Soc., 123: 5086-5094. (Pubitemid 32905664)
    • (2001) Journal of the American Chemical Society , vol.123 , Issue.21 , pp. 5086-5094
    • Beyer, T.1    Day, G.M.2    Price, S.L.3
  • 5
    • 84869626104 scopus 로고    scopus 로고
    • Shargel L, Mutnick AH, Souney PF and Swanson LN (editors). Lippincott Williams and Wilkins A Wolters Kluwer Company, Philadelphia, Baltimore, New York
    • th ed. Lippincott Williams and Wilkins A Wolters Kluwer Company, Philadelphia, Baltimore, New York, p.63.
    • (2001) th Ed. , pp. 63
    • Block, L.H.1    Yu, A.B.C.2
  • 6
    • 0025946401 scopus 로고
    • Optimization of tablet formulation based on starch/lactose granulation for use in tropical countries
    • Bos CE, Bolhius GK and Lerk CF (1991). Optimization of tablet formulation based on starch/lactose granulation for use in tropical countries. Drug Dev. Ind. Pharm., 17(17): 2373-2389.
    • (1991) Drug Dev. Ind. Pharm. , vol.17 , Issue.17 , pp. 2373-2389
    • Bos, C.E.1    Bolhius, G.K.2    Lerk, C.F.3
  • 7
    • 0004206781 scopus 로고    scopus 로고
    • The Stationary Office, London, A358
    • British Pharmacopoeia (2004).The Stationary Office, London, pp.2499, A358.
    • (2004) British Pharmacopoeia , pp. 2499
  • 8
    • 0016211743 scopus 로고
    • Dissolution of Lithium and Magnesium from Lithium carbonate capsules containing Magnesium stearate
    • Caldwell HC (1974). Dissolution of Lithium and Magnesium from Lithium carbonate capsules containing Magnesium stearate. J. Pharm. Sci., 63: 770-773.
    • (1974) J. Pharm. Sci. , vol.63 , pp. 770-773
    • Caldwell, H.C.1
  • 9
    • 70349529703 scopus 로고    scopus 로고
    • Optimization of hydrochlorothiazide tablets
    • Ceshel GC, Maffei P and Badiello R (1999). Optimization of hydrochlorothiazide tablets. Drug Dev. Ind. Pharm., 25(11): 1187-11176
    • (1999) Drug Dev. Ind. Pharm. , vol.25 , Issue.11 , pp. 1187-11176
    • Ceshel, G.C.1    Maffei, P.2    Badiello, R.3
  • 10
    • 0026477593 scopus 로고
    • The effect of two lubricants (Magnesium stearate and Pruv) in the formation of tablets of four anti-ulcer agents/ by means of direct compression
    • Garcia- Marquez MA, Munoz A and Jimenez-Castellanos MR (1992). The effect of two lubricants (Magnesium stearate and Pruv) in the formation of tablets of four anti-ulcer agents/ by means of direct compression. Pharm Acta Helv., 67(2): 50-56.
    • (1992) Pharm Acta Helv. , vol.67 , Issue.2 , pp. 50-56
    • Garcia-Marquez, M.A.1    Munoz, A.2    Jimenez-Castellanos, M.R.3
  • 11
    • 0033159805 scopus 로고    scopus 로고
    • Manufacture of Lithium carbonate tablets using direct compression
    • Gazikolovic E, Obrenovic D and Nidzovic Z (1999). Manufacture of Lithium carbonate tablets using direct compression. Vojnosanit. Preg., 56(4): 389-392.
    • (1999) Vojnosanit. Preg. , vol.56 , Issue.4 , pp. 389-392
    • Gazikolovic, E.1    Obrenovic, D.2    Nidzovic, Z.3
  • 12
    • 27444436820 scopus 로고    scopus 로고
    • A review of Co-processed Directly compressible excipients
    • Gohel MC (2005). A review of Co-processed Directly compressible excipients. J. Pharm. Sci., 8(1): 76-93.
    • (2005) J. Pharm. Sci. , vol.8 , Issue.1 , pp. 76-93
    • Gohel, M.C.1
  • 13
    • 0036025245 scopus 로고    scopus 로고
    • Power of experimental design studies for the validation of pharmaceutical processes: Case study of a multilayer tablet manufacturing process
    • DOI 10.1081/DDC-120005630
    • Goutte F, Guemguem F, Dragan C, Vergnault G and Wehrle P (2002). Power of experimental design studies for the validation of pharmaceutical processes: case study of a multilayer tablet manufacturing process. Drug Dev. Ind. Pharm., 28(7): 841-848. (Pubitemid 34977802)
    • (2002) Drug Development and Industrial Pharmacy , vol.28 , Issue.7 , pp. 841-848
    • Goutte, F.1    Guemguem, F.2    Dragan, C.3    Vergnault, G.4    Wehrle, P.5
  • 14
    • 70349540434 scopus 로고
    • Pharmaceutical Development
    • Griffin JP, Grady JO and Wells FO editors. Greystone Books Ltd., Caulside Drive, Antrim, N. Ireland
    • Halbert G W (1993). Pharmaceutical Development. In: Griffin JP, Grady JO and Wells FO editors. The Text Book of Pharmaceutical Medicine. Greystone Books Ltd., Caulside Drive, Antrim, N. Ireland, pp.39- 40.
    • (1993) The Text Book of Pharmaceutical Medicine , pp. 39-40
    • Halbert, G.W.1
  • 15
    • 84869633734 scopus 로고    scopus 로고
    • Rowe RY, Sheskey PJ, Weller PJ (editors). Pharmaceutical Press, London, Chicago
    • th ed., Pharmaceutical Press, London, Chicago, pp.183-184.
    • (2003) th Ed. , pp. 183-184
    • He, X.1    Kibbe, A.H.2
  • 16
    • 0000426725 scopus 로고    scopus 로고
    • Interface between Monoclinic Crystalline Cellulose and Water: Break down of the oddf even duplicity
    • Hernier AP and Teleman O (1997). Interface between Monoclinic Crystalline Cellulose and Water: Break down of the oddf even duplicity. Langmuir, 13: 511-518.
    • (1997) Langmuir , vol.13 , pp. 511-518
    • Hernier, A.P.1    Teleman, O.2
  • 17
    • 0026799820 scopus 로고
    • Effect of commercial and high purity Magnesium stearate on in vitro dissolution of Paracetamol DC tablets
    • Hussain MSH, York P and Timmins P (1992). Effect of commercial and high purity Magnesium stearate on in vitro dissolution of Paracetamol DC tablets. Int. J. Pharm., 78: 203-207.
    • (1992) Int. J. Pharm. , vol.78 , pp. 203-207
    • Hussain, M.S.H.1    York, P.2    Timmins, P.3
  • 18
    • 0026001231 scopus 로고
    • Comperative microbial contamination levels in wet granulation and direct compression methods of tablet production
    • Ibrahim and Olurinola (1991). Comperative microbial contamination levels in wet granulation and direct compression methods of tablet production. Pharm. Acta. Helv., 66: 293-301.
    • (1991) Pharm. Acta. Helv. , vol.66 , pp. 293-301
    • Ibrahim1    Olurinola2
  • 19
    • 0034141429 scopus 로고    scopus 로고
    • An overview of the different excipients useful for the direct compression of tablets
    • DOI 10.1016/S1461-5347(99)00237-0, PII S1461534799002370
    • Jivraj M, Martini LG and Thomson CM (2000). An overview of different excipients useful for the direct compression of tablets. Pharm. Sci. Technol., 3(2): 58-63. (Pubitemid 30101632)
    • (2000) Pharmaceutical Science and Technology Today , vol.3 , Issue.2 , pp. 58-63
    • Jivraj, M.1    Martini, L.G.2    Thomson, C.M.3
  • 20
    • 0030317019 scopus 로고    scopus 로고
    • Pharmaceutical granulation and tablet formulation using neural networks
    • Kesavan JG and Peck GE (1996). Pharmaceutical granulation and tablet formulation using neural networks. Pharm. Dev. Technol., 1(4): 391-404.
    • (1996) Pharm. Dev. Technol. , vol.1 , Issue.4 , pp. 391-404
    • Kesavan, J.G.1    Peck, G.E.2
  • 21
    • 33745502024 scopus 로고    scopus 로고
    • Zero-order release of aspirin, theophylline and atenolol in water from novel methylcellulose glutarate matrix tablets
    • DOI 10.1016/j.ijpharm.2006.03.020, PII S0378517306002316
    • Khairuzzaman A, Ahmed SU, Savva M and Patel NK (2006). Zero-order release of Aspirin, Theophylline and Atenolol in water from novel Methylcellulose glutarate matrix tablets. Int. J. Pharm., 318(1-2): 15-21. (Pubitemid 43963298)
    • (2006) International Journal of Pharmaceutics , vol.318 , Issue.1-2 , pp. 15-21
    • Khairuzzaman, A.1    Ahmed, S.U.2    Savva, M.3    Patel, N.K.4
  • 23
    • 0346560087 scopus 로고
    • Effect of certain formulation factors on dissolution rate of the active ingredient III: Tablet Lubricants
    • Levy G and Gumtow RH (1963). Effect of certain formulation factors on dissolution rate of the active ingredient III: tablet Lubricants. J Pharm Sci., 52: 1139-1144.
    • (1963) J Pharm Sci. , vol.52 , pp. 1139-1144
    • Levy, G.1    Gumtow, R.H.2
  • 24
    • 0037074121 scopus 로고    scopus 로고
    • The impact of low levels of amorphous material (<5%) on the blending characteristics of a direct compression formulation
    • DOI 10.1016/S0378-5173(01)00880-8, PII S0378517301008808
    • Mackin L, Sartnurak S, Thomas I, and Moore S (2002). The impact of low levels of amorphous material (<5%) on the blending characteristics of a direct compression formulation. Int J Pharm., 231(2): 213-226. (Pubitemid 34033680)
    • (2002) International Journal of Pharmaceutics , vol.231 , Issue.2 , pp. 213-226
    • Mackin, L.1    Sartnurak, S.2    Thomas, I.3    Moore, S.4
  • 25
    • 33748437092 scopus 로고    scopus 로고
    • Optimization of poorly compactable drug tablets manufactured by direct compression using the mixture experimental design
    • DOI 10.1016/j.ijpharm.2006.05.034, PII S0378517306004157
    • Martinello T, Kaneko TM, Velasco MVR, Taqueda MVS and Consiglieri VO (2006). Optimization of poorly compactable drug tablets manufactured by direct compression using the mixture experimental design. Int. J. Pharm., 322 (1-2): 87-95. (Pubitemid 44339597)
    • (2006) International Journal of Pharmaceutics , vol.322 , Issue.1-2 , pp. 87-95
    • Martinello, T.1    Kaneko, T.M.2    Velasco, M.V.R.3    Taqueda, M.E.S.4    Consiglieri, V.O.5
  • 26
    • 4344651533 scopus 로고    scopus 로고
    • Particle interaction of lubricated or unlubricated binary mixtures according to their particle size and densification mechanism
    • DOI 10.1016/j.farmac.2004.04.003, PII S0014827X04000904
    • Martino PD, Joiris E and Martelli S (2004). Particle interaction of lubricated or un lubricated binary mixtures according to their particle size and densification mechanism II. Farmaco., 59(9): 747-758. (Pubitemid 39150038)
    • (2004) Farmaco , vol.59 , Issue.9 , pp. 747-758
    • Di Martino, P.1    Joiris, E.2    Martelli, S.3
  • 27
    • 0037391798 scopus 로고    scopus 로고
    • Forty years of Ibuprofen use
    • Moore N (2003). Forty years of Ibuprofen use. Int. J. Clin. Pract. 135(Suppl.): 28-31.
    • (2003) Int. J. Clin. Pract. , vol.135 , Issue.SUPPL. , pp. 28-31
    • Moore, N.1
  • 28
    • 0035320918 scopus 로고    scopus 로고
    • Celecoxib and Rofecoxib. The role of COX-2 inhibitors in dental practice
    • Moore PA and Hersh EV (2001). Celecoxib and Rofecoxib. The role of COX-2 inhibitors in dental practice. J Am Dent Assoc. 132(4): 451-456.
    • (2001) J Am Dent Assoc , vol.132 , Issue.4 , pp. 451-456
    • Moore, P.A.1    Hersh, E.V.2
  • 29
    • 0022999373 scopus 로고
    • Evaluation of microcrystalline cellulose as a glidant
    • Omray A and Omray P (1986). Evaluation of microcrystalline cellulose as a glidant. Indian J. Pharm. Sci., 48: 20-22.
    • (1986) Indian J. Pharm. Sci. , vol.48 , pp. 20-22
    • Omray, A.1    Omray, P.2
  • 32
    • 0007274685 scopus 로고
    • Maintaining product uniformity and uninterrupted flow to direct-compression tableting press
    • Prescott JK and Hossfield RJ (1994). Maintaining product uniformity and uninterrupted flow to direct-compression tableting press. Pharmaceutical technology, 18 (6): 99-114.
    • (1994) Pharmaceutical Technology , vol.18 , Issue.6 , pp. 99-114
    • Prescott, J.K.1    Hossfield, R.J.2
  • 33
    • 0036805062 scopus 로고    scopus 로고
    • Ibuprofen crystals with optimized properties
    • Rasenack N and Muller BW (2002). Ibuprofen crystals with optimized properties. Int. J. Pham., 245(Suppl 1-2): 9-24.
    • (2002) Int. J. Pham. , vol.245 , Issue.SUPPL. 1-2 , pp. 9-24
    • Rasenack, N.1    Muller, B.W.2
  • 34
    • 0003634042 scopus 로고
    • Rawlins EA editor Bailliere Tindall, London
    • th ed., Bailliere Tindall, London, pp. 289-290.
    • (1995) th Ed. , pp. 289-290
  • 36
    • 0000441553 scopus 로고
    • Liberman HA, Lachman L and Schwartz JB editors. Mercel Dekker, Inc., New York
    • Shangraw RF (1989). In: Liberman HA, Lachman L and Schwartz JB editors. Pharmaceutical Dosage Forms: Tablets, Vol.01 , Mercel Dekker, Inc., New York, pp.109-164.
    • (1989) Pharmaceutical Dosage Forms: Tablets , vol.1 , pp. 109-164
    • Shangraw, R.F.1
  • 38
    • 1842832428 scopus 로고    scopus 로고
    • Preparation of antipyretic analgesic by direct compression and its evaluation
    • Terashita K and Imamura K (2002). Preparation of antipyretic analgesic by direct compression and its evaluation. Chem. Pharm. Bull. (Tokyo). 50(12): 1542-1549.
    • (2002) Chem. Pharm. Bull. (Tokyo) , vol.50 , Issue.12 , pp. 1542-1549
    • Terashita, K.1    Imamura, K.2
  • 39
    • 24744436587 scopus 로고    scopus 로고
    • Evaluation of hexagonal boron nitride as a new tablet lubricant
    • DOI 10.1081/PDT-65684
    • Turkoglu M, Sahin I and San T (2005). Evaluation of hexagonal boron nitride as a new tablet lubricant. Pharm. Dev. Technol., 10(3): 381-388. (Pubitemid 41291475)
    • (2005) Pharmaceutical Development and Technology , vol.10 , Issue.3 , pp. 381-388
    • Turkoglu, M.1    Sahin, I.2    San, T.3
  • 40
    • 70349543860 scopus 로고    scopus 로고
    • (USP 27 NF 22) convention INC.
    • United State Pharmacopoeia 2005. (USP 27 NF 22) convention INC., pp.2308-2309.
    • (2005) United State Pharmacopoeia , pp. 2308-2309
  • 41
    • 34447621596 scopus 로고    scopus 로고
    • Fatality after deliberate ingestion of sustained-release ibuprofen: A case report
    • DOI 10.1186/cc4850
    • Wood DM, Monaghan J, Streete P, Jones AL and Dargan PI (2006). Fatality after deliberate ingestion of sustained- release Ibuprofen; a case report. Critical Care. 10:R44. (Pubitemid 47086798)
    • (2006) Critical Care , vol.10 , Issue.2
    • Wood, D.M.1    Monaghan, J.2    Streete, P.3    Jones, A.L.4    Ivor Dargan, P.5
  • 42
    • 33644837469 scopus 로고    scopus 로고
    • Comparative Study of Different Formulations of Atenolol
    • Yasmeen R, Shoaib MH and Khalid H (2005). Comparative Study of Different Formulations of Atenolol. Pak. J. Pharm Sci., 18(1): 49.
    • (2005) Pak. J. Pharm Sci. , vol.18 , Issue.1 , pp. 49
    • Yasmeen, R.1    Shoaib, M.H.2    Khalid, H.3
  • 43
    • 23144448736 scopus 로고    scopus 로고
    • Physical properties and compact analysis of commonly used direct compression binders
    • Zhang Y, Law Y and Chakrabarti S (2003). Physical Properties and Compact Analysis of Commonly Used Direct Compression Binders. AAPS Pharm. Sci. Tech., 4(4): 1-11. (Pubitemid 41086186)
    • (2003) AAPS PharmSciTech , vol.4 , Issue.4 , pp. 62
    • Zhang, Y.1    Law, Y.2    Chakrabarti, S.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.