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Volumn 3, Issue 2, 2000, Pages 58-63

An overview of the different excipients useful for the direct compression of tablets

Author keywords

[No Author keywords available]

Indexed keywords

AMYLOPECTIN; CALCIUM PHOSPHATE DIBASIC; DRUG; EXCIPIENT; LACTOSE; LUBRICATING AGENT; MAGNESIUM STEARATE; MICROCRYSTALLINE CELLULOSE; STARCH;

EID: 0034141429     PISSN: 14615347     EISSN: None     Source Type: Journal    
DOI: 10.1016/S1461-5347(99)00237-0     Document Type: Review
Times cited : (399)

References (39)
  • 2
    • 0007196894 scopus 로고    scopus 로고
    • Direct compression characteristics of granulated Lactitol
    • 2 Armstrong, N.A. (1997) Direct compression characteristics of granulated Lactitol. Pharm.Technol. Eur. 9, 24-30
    • (1997) Pharm.Technol. Eur. , vol.9 , pp. 24-30
    • Armstrong, N.A.1
  • 3
    • 0001873133 scopus 로고
    • The production of tablets by direct compression
    • 3 Khan, K.A. and Rhodes, C.T. (1973) The production of tablets by direct compression. Can. J. Pharm. Sci. 8, 1-5
    • (1973) Can. J. Pharm. Sci. , vol.8 , pp. 1-5
    • Khan, K.A.1    Rhodes, C.T.2
  • 4
    • 0023201814 scopus 로고
    • A study of the compactibility characteristics of a direct compression and a wet granulated formulation of norfloxacin
    • 4 Katdare, A.V. and Bavitz, J.E. (1987) A study of the compactibility characteristics of a direct compression and a wet granulated formulation of norfloxacin. Drug Dev. Ind. Pharm. 13, 1047-1061
    • (1987) Drug Dev. Ind. Pharm. , vol.13 , pp. 1047-1061
    • Katdare, A.V.1    Bavitz, J.F.2
  • 5
    • 0008957011 scopus 로고
    • Criteria for assessing direct compression diluents
    • 5 Armstrong, N.A. (1986) Criteria for assessing direct compression diluents. Manuf. Chem. 57, 29-31
    • (1986) Manuf. Chem. , vol.57 , pp. 29-31
    • Armstrong, N.A.1
  • 6
    • 0007196894 scopus 로고    scopus 로고
    • Selection of excipients for direct compression tablet formulations
    • 6 Armstrong, N.A. (1998) Selection of excipients for direct compression tablet formulations. Pharm.Technol. Eur. 39, 24-30
    • (1998) Pharm.Technol. Eur. , vol.39 , pp. 24-30
    • Armstrong, N.A.1
  • 8
    • 0003005657 scopus 로고
    • A survey of current industrial practices in the formulation and manufacture of tablets and capsules
    • 8 Shangraw, R.F. and Demarest, D.A. (1993) A survey of current industrial practices in the formulation and manufacture of tablets and capsules. Pharm. Technol. 17, 32-38
    • (1993) Pharm. Technol. , vol.17 , pp. 32-38
    • Shangraw, R.F.1    Demarest, D.A.2
  • 9
    • 0019868032 scopus 로고
    • The effect of moisture content of microcrystalline cellulose on the compressional properties of some formulations
    • 9 Khan, K.A. et al. (1981) The effect of moisture content of microcrystalline cellulose on the compressional properties of some formulations. Drug. Dev. Ind. Pharm. 7, 525-538
    • (1981) Drug. Dev. Ind. Pharm. , vol.7 , pp. 525-538
    • Khan, K.A.1
  • 10
    • 84984088144 scopus 로고
    • Microcrystalline cellulose in tableting
    • 10 Reier, G.E. and Shangraw, R.F. (1966) Microcrystalline cellulose in tableting. J. Pharm. Sci. 55, 510-514
    • (1966) J. Pharm. Sci. , vol.55 , pp. 510-514
    • Reier, G.E.1    Shangraw, R.F.2
  • 11
    • 0019908451 scopus 로고
    • Effect of particle size on the compaction mechanism and tensile strength of tablets
    • 11 Mckenna, A. and McCafferty, D.F. (1982) Effect of particle size on the compaction mechanism and tensile strength of tablets. J. Pharm. Pharmacol. 34, 347-351
    • (1982) J. Pharm. Pharmacol. , vol.34 , pp. 347-351
    • Mckenna, A.1    McCafferty, D.F.2
  • 12
    • 0022478706 scopus 로고
    • The effect of the relationship between punch velocity and particle size on the compaction behaviour of materials with varying deformation mechanisms
    • 12 Roberts, R.J. and Rowe, R.C. (1986) The effect of the relationship between punch velocity and particle size on the compaction behaviour of materials with varying deformation mechanisms. J. Pharm. Pharmacol. 38, 567-571
    • (1986) J. Pharm. Pharmacol. , vol.38 , pp. 567-571
    • Roberts, R.J.1    Rowe, R.C.2
  • 13
    • 0000621207 scopus 로고
    • Comparative evaluation of excipients for direct compression
    • 13 Bolhuis, G.K. and Lerk, C.F. (1973) Comparative evaluation of excipients for direct compression, I. Pharm.Weekbl. 108, 469-481
    • (1973) I. Pharm.Weekbl. , vol.108 , pp. 469-481
    • Bolhuis, G.K.1    Lerk, C.F.2
  • 14
    • 0016204022 scopus 로고
    • Comparative evaluation of excipients for direct compression
    • 14 Lerk, C.F. et al. (1974) Comparative evaluation of excipients for direct compression, II. Pharm.Weekbl. 109, 945-955
    • (1974) II. Pharm.Weekbl. , vol.109 , pp. 945-955
    • Lerk, C.F.1
  • 15
    • 0000568058 scopus 로고    scopus 로고
    • Materials for direct compaction
    • (Alderborn, G. and Nystrom, C., eds), Marcel Dekker, New York, USA
    • 15 Bolhuis, G.K and Chowhan, Z.T. (1996) Materials for direct compaction. In Pharmaceutical Powder Compaction Technology (Alderborn, G. and Nystrom, C., eds), pp. 419-500, Marcel Dekker, New York, USA
    • (1996) Pharmaceutical Powder Compaction Technology , pp. 419-500
    • Bolhuis, G.K.1    Chowhan, Z.T.2
  • 16
    • 0008900453 scopus 로고
    • Morphology and functionality in tablet excipients for direct compression: Part II
    • 16 Shangraw, R.F. et al. (1981) Morphology and functionality in tablet excipients for direct compression: Part II. Pharm.Technol. 5, 44-60
    • (1981) Pharm.Technol. , vol.5 , pp. 44-60
    • Shangraw, R.F.1
  • 17
    • 0018132437 scopus 로고
    • Time-dependent deformation of some direct compression excipients
    • 17 Rees, J.E. and Rue, P.J. (1978) Time-dependent deformation of some direct compression excipients. J. Pharm. Pharmacol. 30, 601-607
    • (1978) J. Pharm. Pharmacol. , vol.30 , pp. 601-607
    • Rees, J.E.1    Rue, P.J.2
  • 18
    • 0016608523 scopus 로고
    • Film formation by magnesium stearate during mixing and its effect on tableting
    • 18 Bolhuis, G.K. et al. (1975) Film formation by magnesium stearate during mixing and its effect on tableting. Pharm. Weekbl. 110, 317-325
    • (1975) Pharm. Weekbl. , vol.110 , pp. 317-325
    • Bolhuis, G.K.1
  • 19
    • 0022644745 scopus 로고
    • The role of water uptake on tablet disintegration
    • 19 Van Kamp, H. V. et al. (1986) The role of water uptake on tablet disintegration. Pharm.Acta. Helv. 61, 22-29
    • (1986) Pharm.Acta. Helv. , vol.61 , pp. 22-29
    • Van Kamp, H.V.1
  • 20
    • 0017164326 scopus 로고
    • Contact angles and wetting of pharmaceutical powders
    • 20 Lerk, C.F. et al. (1976) Contact angles and wetting of pharmaceutical powders. J. Pharm. Sci. 65, 843-847
    • (1976) J. Pharm. Sci. , vol.65 , pp. 843-847
    • Lerk, C.F.1
  • 21
    • 0023009119 scopus 로고
    • Water uptake and disintegrating force measurements: Towards a general understanding of disintegration mechanisms
    • 21 Caramella, C. et al. (1986) Water uptake and disintegrating force measurements: towards a general understanding of disintegration mechanisms. Drug Dev. Ind. Pharm. 12, 1749-1766
    • (1986) Drug Dev. Ind. Pharm. , vol.12 , pp. 1749-1766
    • Caramella, C.1
  • 22
    • 0017029833 scopus 로고
    • Effect of variation in compaction force on properties of six direct compression tablet formulations
    • 22 Khan, K.A. and Rhodes, C.T. (1976) Effect of variation in compaction force on properties of six direct compression tablet formulations. J. Pharm. Sci. 65, 1835-1837
    • (1976) J. Pharm. Sci. , vol.65 , pp. 1835-1837
    • Khan, K.A.1    Rhodes, C.T.2
  • 23
    • 0015356079 scopus 로고
    • Effect of moisture on physical characteristics of tablets prepared from direct compression excipients
    • 23 Sangekar, S.A. et al. (1972) Effect of moisture on physical characteristics of tablets prepared from direct compression excipients. J. Pharm. Sci. 61, 939-944
    • (1972) J. Pharm. Sci. , vol.61 , pp. 939-944
    • Sangekar, S.A.1
  • 24
    • 0019441795 scopus 로고
    • Dicalcium phosphate dihydrate -microcrystalline cellulose systems in direct compression tableting
    • 24 Wells, J.I. and Langridge, J.R. (1981) Dicalcium phosphate dihydrate -microcrystalline cellulose systems in direct compression tableting. Int. J. Pharm.Technol. & Prod. Manuf. 2, 1-8
    • (1981) Int. J. Pharm.Technol. & Prod. Manuf. , vol.2 , pp. 1-8
    • Wells, J.I.1    Langridge, J.R.2
  • 25
    • 0031936142 scopus 로고    scopus 로고
    • Maillard reaction of lactose and fluoxetine hydrochloride, a secondary amine
    • 25 Wirth, D.D. et al. (1998) Maillard reaction of lactose and fluoxetine hydrochloride, a secondary amine. J. Pharm. Sci. 87, 31-39
    • (1998) J. Pharm. Sci. , vol.87 , pp. 31-39
    • Wirth, D.D.1
  • 26
    • 0023882740 scopus 로고
    • The evaluation of six lactose-based materials as direct compression tablet excipients
    • 26 Whiteman, M. and Yarwood, R.J. (1988) The evaluation of six lactose-based materials as direct compression tablet excipients. Drug Dev. Ind. Pharm. 14, 1023-1040
    • (1988) Drug Dev. Ind. Pharm. , vol.14 , pp. 1023-1040
    • Whiteman, M.1    Yarwood, R.J.2
  • 28
    • 0021031968 scopus 로고
    • Tableting characteristics of sorbitol
    • 28 Schmidt, P.C. (1983) Tableting characteristics of sorbitol. Pharm.Technol. 7, 65-74
    • (1983) Pharm.Technol. , vol.7 , pp. 65-74
    • Schmidt, P.C.1
  • 29
    • 0021630171 scopus 로고
    • Modification of the crystalline structure of sorbitol and its effects on tableting characteristics
    • 29 Du Ross, J.W. (1974) Modification of the crystalline structure of sorbitol and its effects on tableting characteristics. Pharm.Technol. 8, 42
    • (1974) Pharm.Technol. , vol.8 , pp. 42
    • Du Ross, J.W.1
  • 30
    • 0001647951 scopus 로고
    • Study of different crystalline forms of mannitol: Comparative behaviour under compression
    • 30 Debord, B. et al. (1987) Study of different crystalline forms of mannitol: comparative behaviour under compression. Drug Dev. Ind. Pharm. 13, 1533-1546
    • (1987) Drug Dev. Ind. Pharm. , vol.13 , pp. 1533-1546
    • Debord, B.1
  • 31
    • 0031941064 scopus 로고    scopus 로고
    • Direct compression characterisitics of granulated Lactitol
    • 31 Armstrong, N.A. (1998) Direct compression characterisitics of granulated Lactitol. Pharm.Technol. 22, 84-92
    • (1998) Pharm.Technol. , vol.22 , pp. 84-92
    • Armstrong, N.A.1
  • 32
    • 0008920064 scopus 로고    scopus 로고
    • Crystalline maltose: A direct compression pharmaceutical excipient
    • 32 Bowe, K.E. et al. (1998) Crystalline maltose: A direct compression pharmaceutical excipient. Pharm.Technol. Eur. 10, 34-40
    • (1998) Pharm.Technol. Eur. , vol.10 , pp. 34-40
    • Bowe, K.E.1
  • 33
    • 0027996978 scopus 로고
    • Evaluation of ludipress as a 'multipurpose excipient' for direct compression. Part I: Powder characteristics and tableting properties
    • 33 Schmidt, P.C. and Rubensdorfer, C.J.W. (1994) Evaluation of Ludipress as a 'multipurpose excipient' for direct compression. Part I: Powder characteristics and tableting properties. Drug Dev. Ind. Pharm. 20, 2899-2925
    • (1994) Drug Dev. Ind. Pharm. , vol.20 , pp. 2899-2925
    • Schmidt, P.C.1    Rubensdorfer, C.J.W.2
  • 34
    • 0026747303 scopus 로고
    • Evaluation of the tableting properties of a new excipient for direct compression
    • 34 Plazier-Vercammen, J.A. and Van der Bossche, H. (1992) Evaluation of the tableting properties of a new excipient for direct compression. Pharm. Ind. 54, 973-977
    • (1992) Pharm. Ind. , vol.54 , pp. 973-977
    • Plazier-Vercammen, J.A.1    Van Der Bossche, H.2
  • 35
    • 0028173275 scopus 로고
    • Pharmaceutical development of tablets of a new antineoplastic drug: Mitonafide
    • 35 Suarez, A.I.T. et al. ( 1994) Pharmaceutical development of tablets of a new antineoplastic drug: mitonafide. Pharm.Acta. Helv. 69, 101-105
    • (1994) Pharm.Acta. Helv. , vol.69 , pp. 101-105
    • Suarez, A.I.T.1
  • 36
    • 0032528373 scopus 로고    scopus 로고
    • Physicochemical comparison between microcrystalline cellulose and silicified microcrystalline cellulose
    • 36 Tobyn, M.J. et al. (1998) Physicochemical comparison between microcrystalline cellulose and silicified microcrystalline cellulose. Int. J. Pharm. 169, 183-194
    • (1998) Int. J. Pharm. , vol.169 , pp. 183-194
    • Tobyn, M.J.1
  • 37
    • 0008881119 scopus 로고    scopus 로고
    • Silicified microcrystalline cellulose (SMCC): A new class of high functionality binders for direct compression tableting
    • PT 6164, Plenum Press, New York, USA
    • 37 Sherwood, B.E. et al. (1996) Silicified microcrystalline cellulose (SMCC): a new class of high functionality binders for direct compression tableting. Proc. AAPS Conf., PT 6164, Plenum Press, New York, USA
    • (1996) Proc. AAPS Conf.
    • Sherwood, B.E.1
  • 38
    • 0033151655 scopus 로고    scopus 로고
    • Excipients as stabilisers
    • 38 Crowley, P.J. (1999) Excipients as stabilisers. Pharm. Sci.Technol.Today 2, 237-243
    • (1999) Pharm. Sci.Technol.Today , vol.2 , pp. 237-243
    • Crowley, P.J.1
  • 39
    • 0032809138 scopus 로고    scopus 로고
    • Selection of solid dosage form composition through drug-excipient compatibility testing
    • 39 Serajuddin, A.T.M. et al. (1999) Selection of solid dosage form composition through drug-excipient compatibility testing. J. Pharm. Sci. 88, 696-704
    • (1999) J. Pharm. Sci. , vol.88 , pp. 696-704
    • Serajuddin, A.T.M.1


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.