Squash inhibitors: From structural motifs to macrocyclic knottins

Current Protein and Peptide Science

Volumn 5, Issue 5, 2004, Pages 341-349

  Chiche, Laurent ^a   Heitz, Annie ^a   Gelly, Jean Christophe ^a   Gracy, Jérôme ^a   Chau, Pham T T ^b   Ha, Phan T ^b   Hernandez, Jean François ^c   Le Nguyen, Dung ^d  

^a CNRS   (France)

^b VIETNAM NATIONAL UNIVERSITY   (Viet Nam)

^c UNIVERSITÉ DE MONTPELLIER   (France)

^d HÔPITAL ARNAUD DE VILLENEUVE   (France)

Author keywords

Disulfide bridges; Drug design; Inhibitor cystine knots; Knottins; Macrocyclic proteins; Serine proteinases; Squash inhibitors; Structural motifs

Indexed keywords

AMYLASE INHIBITOR; CONOTOXIN; CYCLOPEPTIDE; CYSTINE; GURMARIN; KALATA B1; MACROCYCLIC COMPOUND; SERINE PROTEINASE INHIBITOR; TRYPSIN INHIBITOR; TRYPSIN INHIBITOR I; TRYPSIN INHIBITOR II; UNCLASSIFIED DRUG;

AMINO TERMINAL SEQUENCE; BETA SHEET; CARBOXY TERMINAL SEQUENCE; CUCUMBER; DISULFIDE BOND; DRUG ACTIVITY; DRUG DETERMINATION; DRUG ISOLATION; DRUG POTENCY; DRUG STABILITY; DRUG STRUCTURE; DRUG SYNTHESIS; MOMORDICA; NONHUMAN; PROTEIN MOTIF; REVIEW; SPECIES DIFFERENCE; VIET NAM;

AMINO ACID SEQUENCE; CUCURBITA; CYCLIZATION; DRUG DESIGN; HUMANS; MOLECULAR SEQUENCE DATA; PROTEIN FOLDING; PROTEINS; SERINE PROTEINASE INHIBITORS;

ANIMALIA; CUCURBITACEAE; FUNGI; MOMORDICA; MOMORDICA COCHINCHINENSIS;

EID: 4444318429     PISSN: 13892037     EISSN: None     Source Type: Journal    
DOI: 10.2174/1389203043379477     Document Type: Review

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