Synthesis and antiproliferative activity of imidazole and imidazoline analogs for melanoma

Bioorganic and Medicinal Chemistry Letters

Volumn 18, Issue 11, 2008, Pages 3183-3187

  Chen, Jianjun ^a   Wang, Zhao ^a   Lu, Yan ^a   Dalton, James T ^b   Miller, Duane D ^a   Li, Wei ^a  

^a UNIVERSITY OF TENNESSEE HEALTH SCIENCE CENTER   (United States)

^b OHIO STATE UNIVERSITY   (United States)

Author keywords

Imidazole analogs; Imidazoline analogs; Melanoma; Structure activity relationships; Thiazolidine

Indexed keywords

IMIDAZOLE; IMIDAZOLINE DERIVATIVE; SORAFENIB; THIAZOLIDINE DERIVATIVE;

ARTICLE; DRUG ACTIVITY; DRUG SYNTHESIS; FIBROBLAST; HUMAN; MELANOMA; MELANOMA CELL; NONHUMAN;

ANTINEOPLASTIC AGENTS; CELL LINE, TUMOR; CELL PROLIFERATION; DRUG SCREENING ASSAYS, ANTITUMOR; HUMANS; IMIDAZOLES; IMIDAZOLINES; MELANOMA; STRUCTURE-ACTIVITY RELATIONSHIP; THIAZOLIDINES;

EID: 44149102682     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2008.04.073     Document Type: Article

References (26)

1. Atallah E., and Flaherty L. Curr. Treat. Options Oncol. 6 (2005) 185
2. Barth A., Wanek L.A., and Morton D.L. J. Am. Coll. Surg. 181 (1995) 193
3. Anderson C.M., Buzaid A.C., and Legha S.S. Oncol. (Williston Park) 9 (1995) 1149
4. Gogas H.J., Kirkwood J.M., and Sondak V.K. Cancer 109 (2007) 455
5. Serrone L., Zeuli M., Sega F.M., and Cognetti F. J. Exp. Clin. Cancer Res. 19 (2000) 21
6. Gray-Schopfer V., Wellbrock C., and Marais R. Nature 445 (2007) 851
7. Young A.M., Marsden J., Goodman A., Burton A., and Dunn J.A. Clin. Oncol. (R Coll. Radiol.) 13 (2001) 458
8. Mandara M., Nortilli R., Sava T., and Cetto G.L. Expert Rev. Anticancer Ther. 6 (2006) 121
9. Eggermont A.M., and Kirkwood J.M. Eur. J. Cancer 40 (2004) 1825
10. Ranson M., Hersey P., Thompson D., Beith J., McArthur G.A., Haydon A., Davis I.D., Kefford R.F., Mortimer P., Harris P.A., Baka S., Seebaran A., Sabharwal A., Watson A.J., Margison G.P., and Middleton M.R. J. Clin. Oncol. 25 (2007) 2540
11. Larkin J.M., Hughes S.A., Beirne D.A., Patel P.M., Gibbens I.M., Bate S.C., Thomas K., Eisen T.G., and Gore M.E. Br. J. Cancer 96 (2007) 44
12. Garbe C., and Eigentler T.K. Melanoma Res. 17 (2007) 117
13. Koon H.B., and Atkins M.B. Expert Rev. Anticancer Ther. 7 (2007) 79
14. Li W., Lu Y., Wang Z., Dalton J.T., and Miller D.D. Bioorg. Med. Chem. Lett. 17 (2007) 4113
15. Li W., Wang Z., Gududuru V., Zbytek B., Slominski A.T., Dalton J.T., and Miller D.D. Anticancer Res. 27 (2007) 883
16. Williams D.A., and Lemke T.L. Foye's Principles of Medicinal Chemistry. fifth ed. (2002), Lippincott Williams & Wilkins, Philadelphia
17. Anderson W.K., Bhattacharjee D., and Houston D.M. J. Med. Chem. 32 (1989) 119
18. Davis D.P., Kirk K.L., and Cohen L.A. J. Heterocyclic Chem. 19 (1982) 253
19. Gududuru V., Hurh E., Dalton J.T., and Miller D.D. J. Med. Chem. 48 (2005) 2584
20. Bergeron R.J., Wiegand J., Weimar W.R., Vinson J.R., Bussenius J., Yao G.W., and McManis J.S. J. Med. Chem. 42 (1999) 95
21. Hsu F.L., Hamada A., Booher M.E., Fuder H., Patil P.N., and Miller D.D. J. Med. Chem. 23 (1980) 1232
22. Calcinari R., Case N., Guerrato A., Milanino R., Passarella E., Perchinunno M., Tamburini B., and Sparatore F. J. Med. Chem. 24 (1981) 632
23. Wirt U., Frohlich R., and Wunsch B. Tetrahedron: Asymmetry 16 (2005) 2199
24. Sawada Y., Kayakiri H., Abe Y., Mizutani T., Inamura N., Asano M., Aramori I., Hatori C., Oku T., and Tanaka H. J. Med. Chem. 47 (2004) 2667
25. Dothager R.S., Putt K.S., Allen B.J., Leslie B.J., Nesterenko V., and Hergenrother P.J. J. Am. Chem. Soc. 127 (2005) 8686
26. Eisen T., Ahmad T., Flaherty K.T., Gore M., Kaye S., Marais R., Gibbens I., Hackett S., James M., Schuchter L.M., Nathanson K.L., Xia C., Simantov R., Schwartz B., Poulin-Costello M., O'Dwyer P.J., and Ratain M.J. Br. J. Cancer 95 (2006) 581