Novel insight into inhibitor binding of highly symmetric HIV-1 protease

ChemBioChem

Volumn 9, Issue 6, 2008, Pages 874-878

  Wollmann, Jörg ^a   Baumert, Christiane ^a   Erlenkamp, German ^a   Sippl, Wolfgang ^a   Hilgeroth, Andreas ^a  

^a MARTIN LUTHER UNIVERSITY HALLE WITTENBERG   (Germany)

Author keywords

Binding region; Ligand docking; Medicinal chemistry; Structure activity relationships; Symmetric structure

Indexed keywords

1,4 DIHYDROPYRIDINE; A 98881; ANTIVIRUS AGENT; PROTEINASE; PROTEINASE INHIBITOR; UNCLASSIFIED DRUG;

ARTICLE; BINDING AFFINITY; CONTROLLED STUDY; DRUG PROTEIN BINDING; DRUG STRUCTURE; DRUG SYNTHESIS; ENZYME ACTIVE SITE; HUMAN IMMUNODEFICIENCY VIRUS 1; HYDROGEN BOND; MOLECULAR DOCKING; NONHUMAN; PRIORITY JOURNAL; STRUCTURE ACTIVITY RELATION; BINDING SITE; CHEMICAL MODEL; CHEMISTRY; KINETICS; METABOLISM;

HUMAN IMMUNODEFICIENCY VIRUS 1;

BINDING SITES; HIV PROTEASE; HIV PROTEASE INHIBITORS; KINETICS; MODELS, CHEMICAL;

EID: 44049093824     PISSN: 14394227     EISSN: 14397633     Source Type: Journal    
DOI: 10.1002/cbic.200700646     Document Type: Article

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