Efficient preparation of secondary aminoalcohols through a Ti(IV) reductive amination procedure. Application to the synthesis and antibacterial evaluation of new 3β-N-[hydroxyalkyl]aminosteroid derivatives

Tetrahedron

Volumn 64, Issue 19, 2008, Pages 4453-4459

  Salmi, Chanaz ^a   Loncle, Céline ^a   Letourneux, Yves ^a   Brunel, Jean Michel ^a  

^a Aix Marseille University   (France)

Author keywords

[No Author keywords available]

Indexed keywords

3 BETA N [HYDROXYBUTYL]AMINO 4 CHOLESTENE; 3 BETA N [HYDROXYETHYL]AMINO 4 CHOLESTENE; 3 BETA N [HYDROXYHEXYL]AMINO 4 CHOLESTENE; 3 BETA N [HYDROXYPENTYL]AMINO 4 CHOLESTENE; 3 BETA N [HYDROXYPROPYL]AMINO 4 CHOLESTENE; ALCOHOL DERIVATIVE; ANTIINFECTIVE AGENT; KETONE DERIVATIVE; STEROID; TITANIUM; UNCLASSIFIED DRUG;

AMINATION; ANTIBACTERIAL ACTIVITY; ARTICLE; CONTROLLED STUDY; DRUG SCREENING; DRUG STRUCTURE; DRUG SYNTHESIS; ENTEROCOCCUS FAECALIS; IN VITRO STUDY; MINIMUM INHIBITORY CONCENTRATION; NONHUMAN; PRIORITY JOURNAL; REDUCTION; STAPHYLOCOCCUS AUREUS;

ENTEROCOCCUS FAECALIS; NEGIBACTERIA; POSIBACTERIA; STAPHYLOCOCCUS AUREUS;

EID: 41549144697     PISSN: 00404020     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.tet.2008.02.055     Document Type: Article

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