Design, synthesis and antiproliferative properties of oligomers with chromophore units linked by amide backbones

Bioorganic and Medicinal Chemistry Letters

Volumn 18, Issue 7, 2008, Pages 2440-2444

  Farrera Sinfreu, Josep ^a   Aviñó, Anna ^b,c,e   Navarro, Isabel ^d   Aymamí, Juan ^d,f   Beteta, Natàlia G ^a   Varón, Sònia ^a   Pérez Tomás, Ricardo ^g   Castillo Avila, Wilmar ^g   Eritja, Ramon ^b,c,e   Albericio, Fernando ^b,c,g   Royo, Miriam ^a,c  

^a Combinatorial Chemistry Unit ^*  (Spain)

^b INSTITUTE FOR RESEARCH IN BIOMEDICINE   (Spain)

^c BIOMATERIALES Y NANOMEDICINA CIBER BBN   (Spain)

^d Crystax Pharmaceuticals SL   (Spain)

^e INSTITUTE OF ADVANCED CHEMISTRY OF CATALONIA IQAC CSIC   (Spain)

^f UNIVERSITAT POLITÈCNICA DE CATALUNYA   (Spain)

^g UNIVERSITY OF BARCELONA   (Spain)

Author keywords

4 Aminoproline; Antiproliferative; Chromophore; Fluorescence; Ornithine; Peptide nucleic acids; Peptides; Solid phase synthesis

Indexed keywords

AMIDE; PEPTIDE; POLYMER;

ARTICLE; CHEMISTRY; CHROMATOPHORE; DRUG DESIGN; DRUG SYNTHESIS; FLUORESCENCE;

AMIDES; AMINO ACID SEQUENCE; AMINO ACIDS; ANIMALS; ANTINEOPLASTIC AGENTS; CARBOXYLIC ACIDS; CELL LINE, TUMOR; DRUG DESIGN; HUMANS; INHIBITORY CONCENTRATION 50; MICE; MOLECULAR SEQUENCE DATA; PEPTIDES; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 41349088667     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2008.02.045     Document Type: Article

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