Separate synthesis and evaluation of glucitol bis-phosphate and mannitol bis-phosphate, as competitive inhibitors of fructose bis-phosphate aldolases

Bioorganic and Medicinal Chemistry Letters

Volumn 18, Issue 5, 2008, Pages 1735-1737

  Mabiala Bassiloua, Charles Gabin ^a   Zwolinska, Magdalena ^a   Therisod, Helene ^b   Sygusch, Jurgen ^c   Therisod, Michel ^a  

^a UNIVERSITÉ PARIS SUD   (France)

^b INSTITUTE FOR INTEGRATIVE BIOLOGY OF THE CELL I2BC   (France)

^c UNIVERSITÉ DE MONTRÉAL   (Canada)

Author keywords

Aldolase; Enzymes inhibitors; Fructose bis phosphate; Glucitol bis phosphate; Glycolysis; Hexitol bis phosphate; Mannitol bis phosphate

Indexed keywords

FRUCTOSE BISPHOSPHATE ALDOLASE; GLUCITOL 1,6 BISPHOSPHATE; LYASE INHIBITOR; MANNITOL 1,6 BISPHOSPHATE; UNCLASSIFIED DRUG;

ARTICLE; COMPETITIVE INHIBITION; DRUG SCREENING; DRUG STRUCTURE; DRUG SYNTHESIS; ENZYME INHIBITION; INHIBITION KINETICS; STRUCTURE ANALYSIS;

EID: 40149106327     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2008.01.076     Document Type: Article

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