메뉴 건너뛰기




Volumn 352, Issue 1-2, 2008, Pages 104-114

Comparison between lipolysis and compendial dissolution as alternative techniques for the in vitro characterization of α-tocopherol self-emulsified drug delivery systems (SEDDS)

Author keywords

Dissolution; Griseofulvin; Lipolysis; Optimization; SEDDS

Indexed keywords

ALPHA TOCOPHEROL; LABRASOL; OCTANOIC ACID; POLYSORBATE 80;

EID: 39549095134     PISSN: 03785173     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.ijpharm.2007.10.023     Document Type: Article
Times cited : (27)

References (32)
  • 1
    • 16644367240 scopus 로고    scopus 로고
    • Influence of decreasing solvent polarity (1,4-dioxane/water mixtures) on the acid-base and copper(II)-binding properties of guanosine 5′-diphosphate
    • Bianchi E.M., Griesser R., and Sigel H. Influence of decreasing solvent polarity (1,4-dioxane/water mixtures) on the acid-base and copper(II)-binding properties of guanosine 5′-diphosphate. Helv. Chim. Acta 88 (2005) 406-425
    • (2005) Helv. Chim. Acta , vol.88 , pp. 406-425
    • Bianchi, E.M.1    Griesser, R.2    Sigel, H.3
  • 2
    • 0014147113 scopus 로고
    • Partition of lipid between emulsified oil and micellar phases of glyceride-bile salt dispersion
    • Borgström B. Partition of lipid between emulsified oil and micellar phases of glyceride-bile salt dispersion. J. Lipid Res. 8 (1967) 598-608
    • (1967) J. Lipid Res. , vol.8 , pp. 598-608
    • Borgström, B.1
  • 3
    • 0026586447 scopus 로고
    • Self-emulsifying drug delivery systems: formulation and biopharmaceutic evaluation of an investigational lipophilic compound
    • Charman S.A., Charman W.N., Rogge M.C., Wilson T.D., Dutko F.J., and Pouton C.W. Self-emulsifying drug delivery systems: formulation and biopharmaceutic evaluation of an investigational lipophilic compound. Pharm. Res. 9 (1992) 87-93
    • (1992) Pharm. Res. , vol.9 , pp. 87-93
    • Charman, S.A.1    Charman, W.N.2    Rogge, M.C.3    Wilson, T.D.4    Dutko, F.J.5    Pouton, C.W.6
  • 4
    • 0029562489 scopus 로고
    • Lipid microemulsions for improving drug dissolution and oral absorption: physical and biopharmaceutical aspects
    • Constantinides P.P. Lipid microemulsions for improving drug dissolution and oral absorption: physical and biopharmaceutical aspects. Pharm. Res. 12 (1995) 1561-1572
    • (1995) Pharm. Res. , vol.12 , pp. 1561-1572
    • Constantinides, P.P.1
  • 5
    • 0027301116 scopus 로고
    • An investigation into the physico-chemical properties of self-emulsifying systems using low frequency dielectric spectroscopy, surface tension measurements and particle size analysis
    • Craig D.Q.M., Lievens H.S.R., Pitt K.G., and Storey D.E. An investigation into the physico-chemical properties of self-emulsifying systems using low frequency dielectric spectroscopy, surface tension measurements and particle size analysis. Int. J. Pharm. 96 (1993) 147-155
    • (1993) Int. J. Pharm. , vol.96 , pp. 147-155
    • Craig, D.Q.M.1    Lievens, H.S.R.2    Pitt, K.G.3    Storey, D.E.4
  • 6
    • 51249180332 scopus 로고
    • The static dielectric constant of solutions of water inn-alcohols at 15, 25, 35, and 45°C
    • D'Aprano A., Donato D.I., and Caponetti E. The static dielectric constant of solutions of water inn-alcohols at 15, 25, 35, and 45°C. J. Sol. Chem. 8 (1979) 135-146
    • (1979) J. Sol. Chem. , vol.8 , pp. 135-146
    • D'Aprano, A.1    Donato, D.I.2    Caponetti, E.3
  • 7
    • 23444458748 scopus 로고    scopus 로고
    • The development and characterisation of triglyceride-based 'spontaneous' multiple emulsions
    • Devani M.J., Ashford M., and Craig D.Q. The development and characterisation of triglyceride-based 'spontaneous' multiple emulsions. Int. J. Pharm. 300 (2005) 76-88
    • (2005) Int. J. Pharm. , vol.300 , pp. 76-88
    • Devani, M.J.1    Ashford, M.2    Craig, D.Q.3
  • 8
    • 33845919075 scopus 로고    scopus 로고
    • Hard gelatin and hypromellose (HPMC) capsules: estimation of rupture time by real-time dissolution spectroscopy
    • El-Malah Y., and Nazzal S. Hard gelatin and hypromellose (HPMC) capsules: estimation of rupture time by real-time dissolution spectroscopy. Drug Dev. Ind. Pharm. 33 (2007) 27-34
    • (2007) Drug Dev. Ind. Pharm. , vol.33 , pp. 27-34
    • El-Malah, Y.1    Nazzal, S.2
  • 9
    • 34247536339 scopus 로고    scopus 로고
    • Morphological observations on a lipid-based drug delivery system during in vitro digestion
    • Fatouros D.G., Bergenstahl B., and Mullertz A. Morphological observations on a lipid-based drug delivery system during in vitro digestion. Eur. J. Pharm. Sci. 31 (2007) 85-94
    • (2007) Eur. J. Pharm. Sci. , vol.31 , pp. 85-94
    • Fatouros, D.G.1    Bergenstahl, B.2    Mullertz, A.3
  • 10
    • 0032498581 scopus 로고    scopus 로고
    • Physicochemical characterization and evaluation of microemulsion system for oral delivery of cyclosporin A
    • Gao Z.G., Choi H.G., Shin H.J., Park K.M., Lim S.J., Hwang K.J., and Kim C.K. Physicochemical characterization and evaluation of microemulsion system for oral delivery of cyclosporin A. Int. J. Pharm. 161 (1998) 75-86
    • (1998) Int. J. Pharm. , vol.161 , pp. 75-86
    • Gao, Z.G.1    Choi, H.G.2    Shin, H.J.3    Park, K.M.4    Lim, S.J.5    Hwang, K.J.6    Kim, C.K.7
  • 11
    • 0034601204 scopus 로고    scopus 로고
    • Self-dispersing lipid formulations for improving oral absorption of lipophilic drugs
    • Gershanik T., and Benita S. Self-dispersing lipid formulations for improving oral absorption of lipophilic drugs. Eur. J. Pharm. Biopharm. 50 (2000) 179-188
    • (2000) Eur. J. Pharm. Biopharm. , vol.50 , pp. 179-188
    • Gershanik, T.1    Benita, S.2
  • 12
    • 0016296842 scopus 로고
    • Measurement of the 'spontaneity' of self-emulsifiable oils
    • Groves M.J., and Mustafa R.M.A. Measurement of the 'spontaneity' of self-emulsifiable oils. J. Pharm. Pharmacol. 26 (1974) 671-681
    • (1974) J. Pharm. Pharmacol. , vol.26 , pp. 671-681
    • Groves, M.J.1    Mustafa, R.M.A.2
  • 13
    • 1842684453 scopus 로고    scopus 로고
    • Self-emulsifying drug delivery systems (SEDDS) for improved oral delivery of lipophilic drugs
    • Gursoy R.N., and Benita S. Self-emulsifying drug delivery systems (SEDDS) for improved oral delivery of lipophilic drugs. Biomed. Pharmacother. 58 (2004) 173-182
    • (2004) Biomed. Pharmacother. , vol.58 , pp. 173-182
    • Gursoy, R.N.1    Benita, S.2
  • 14
    • 0031914282 scopus 로고    scopus 로고
    • Lipid-based delivery systems for improving the bioavailability and lymphatic transport of a poorly water-soluble LTB4 inhibitor
    • Hauss D.J., Fogal S.E., Ficorilli J.V., Price C.A., Roy T., Jayaraj A.A., and Keirns J.J. Lipid-based delivery systems for improving the bioavailability and lymphatic transport of a poorly water-soluble LTB4 inhibitor. J. Pharm. Sci. 87 (1998) 164-169
    • (1998) J. Pharm. Sci. , vol.87 , pp. 164-169
    • Hauss, D.J.1    Fogal, S.E.2    Ficorilli, J.V.3    Price, C.A.4    Roy, T.5    Jayaraj, A.A.6    Keirns, J.J.7
  • 15
    • 0343963156 scopus 로고    scopus 로고
    • Improved bioavailability of vitamin E with a self-emulsifying formulation
    • Julianto T., Yuen K.H., and Noor A.M. Improved bioavailability of vitamin E with a self-emulsifying formulation. Int. J. Pharm. 200 (2000) 53-57
    • (2000) Int. J. Pharm. , vol.200 , pp. 53-57
    • Julianto, T.1    Yuen, K.H.2    Noor, A.M.3
  • 16
    • 1242291941 scopus 로고    scopus 로고
    • Drug solubilization behavior during in vitro digestion of suspension formulations of poorly water-soluble drugs in triglyceride lipids
    • Kaukonen A.M., Boyd B.J., Charman W.N., and Porter C.J. Drug solubilization behavior during in vitro digestion of suspension formulations of poorly water-soluble drugs in triglyceride lipids. Pharm. Res. 21 (2004) 254-260
    • (2004) Pharm. Res. , vol.21 , pp. 254-260
    • Kaukonen, A.M.1    Boyd, B.J.2    Charman, W.N.3    Porter, C.J.4
  • 17
    • 1242292226 scopus 로고    scopus 로고
    • Drug solubilization behavior during in vitro digestion of simple triglyceride lipid solution formulations
    • Kaukonen A.M., Boyd B.J., Porter C.J., and Charman W.N. Drug solubilization behavior during in vitro digestion of simple triglyceride lipid solution formulations. Pharm. Res. 21 (2004) 245-253
    • (2004) Pharm. Res. , vol.21 , pp. 245-253
    • Kaukonen, A.M.1    Boyd, B.J.2    Porter, C.J.3    Charman, W.N.4
  • 18
    • 0032103706 scopus 로고    scopus 로고
    • Formulation design and bioavailability assessment of lipidic self-emulsifying formulations of halofantrine
    • Khoo S.M., Humberstone A.J., Porter C.J.H., Edwards G.A., and Charman W.N. Formulation design and bioavailability assessment of lipidic self-emulsifying formulations of halofantrine. Int. J. Pharm. 167 (1998) 155-164
    • (1998) Int. J. Pharm. , vol.167 , pp. 155-164
    • Khoo, S.M.1    Humberstone, A.J.2    Porter, C.J.H.3    Edwards, G.A.4    Charman, W.N.5
  • 19
    • 0030728789 scopus 로고    scopus 로고
    • Pharmacokinetic cyclosporine A profiles under long-term neoral treatment in renal transplant recipients: does fat intake still matter?
    • Klauser R.M., Irschik H., Kletzmayr J., Sturm I., Brunner W., Woloszczuk W., and Kovarik J. Pharmacokinetic cyclosporine A profiles under long-term neoral treatment in renal transplant recipients: does fat intake still matter?. Transplant. Proc. 29 (1997) 3137-3140
    • (1997) Transplant. Proc. , vol.29 , pp. 3137-3140
    • Klauser, R.M.1    Irschik, H.2    Kletzmayr, J.3    Sturm, I.4    Brunner, W.5    Woloszczuk, W.6    Kovarik, J.7
  • 21
    • 0343051926 scopus 로고    scopus 로고
    • Influence of lipolysis on drug absorption from the gastrointestinal tract
    • MacGregor K.J., and Embleton J.K. Influence of lipolysis on drug absorption from the gastrointestinal tract. Adv. Drug Deliv. Rev. 25 (1997) 33-46
    • (1997) Adv. Drug Deliv. Rev. , vol.25 , pp. 33-46
    • MacGregor, K.J.1    Embleton, J.K.2
  • 22
    • 0036212425 scopus 로고    scopus 로고
    • Preparation and characterization of coenzyme Q10-Eudragit solid dispersion
    • Nazzal S., Guven N., Reddy I.K., and Khan M.A. Preparation and characterization of coenzyme Q10-Eudragit solid dispersion. Drug Dev. Ind. Pharm. 28 (2002) 49-57
    • (2002) Drug Dev. Ind. Pharm. , vol.28 , pp. 49-57
    • Nazzal, S.1    Guven, N.2    Reddy, I.K.3    Khan, M.A.4
  • 23
    • 0037142237 scopus 로고    scopus 로고
    • Optimization of a self-nanoemulsified tablet dosage form of Ubiquinone using response surface methodology: effect of formulation ingredients
    • Nazzal S., Nutan M., Palamakula A., Shah R., Zaghloul A.A., and Khan M.A. Optimization of a self-nanoemulsified tablet dosage form of Ubiquinone using response surface methodology: effect of formulation ingredients. Int. J. Pharm. 240 (2002) 103-114
    • (2002) Int. J. Pharm. , vol.240 , pp. 103-114
    • Nazzal, S.1    Nutan, M.2    Palamakula, A.3    Shah, R.4    Zaghloul, A.A.5    Khan, M.A.6
  • 24
    • 0037139412 scopus 로고    scopus 로고
    • Preparation and in vitro characterization of a eutectic based semisolid self-nanoemulsified drug delivery system (SNEDDS) of ubiquinone: mechanism and progress of emulsion formation
    • Nazzal S., Smalyukh I.I., Lavrentovich O.D., and Khan M.A. Preparation and in vitro characterization of a eutectic based semisolid self-nanoemulsified drug delivery system (SNEDDS) of ubiquinone: mechanism and progress of emulsion formation. Int. J. Pharm. 235 (2002) 247-265
    • (2002) Int. J. Pharm. , vol.235 , pp. 247-265
    • Nazzal, S.1    Smalyukh, I.I.2    Lavrentovich, O.D.3    Khan, M.A.4
  • 25
    • 0035478436 scopus 로고    scopus 로고
    • In vitro assessment of oral lipid based formulations
    • Porter C.J., and Charman W.N. In vitro assessment of oral lipid based formulations. Adv. Drug Deliv. Rev. 50 (2001) S127-S147
    • (2001) Adv. Drug Deliv. Rev. , vol.50
    • Porter, C.J.1    Charman, W.N.2
  • 26
    • 1942498896 scopus 로고    scopus 로고
    • Use of in vitro lipid digestion data to explain the in vivo performance of triglyceride-based oral lipid formulations of poorly water-soluble drugs: studies with halofantrine
    • Porter C.J., Kaukonen A.M., Taillardat-Bertschinger A., Boyd B.J., O'Connor J.M., Edwards G.A., and Charman W.N. Use of in vitro lipid digestion data to explain the in vivo performance of triglyceride-based oral lipid formulations of poorly water-soluble drugs: studies with halofantrine. J. Pharm. Sci. 93 (2004) 1110-1121
    • (2004) J. Pharm. Sci. , vol.93 , pp. 1110-1121
    • Porter, C.J.1    Kaukonen, A.M.2    Taillardat-Bertschinger, A.3    Boyd, B.J.4    O'Connor, J.M.5    Edwards, G.A.6    Charman, W.N.7
  • 27
    • 4344578729 scopus 로고    scopus 로고
    • Susceptibility to lipase-mediated digestion reduces the oral bioavailability of danazol after administration as a medium-chain lipid-based microemulsion formulation
    • Porter C.J., Kaukonen A.M., Boyd B.J., Edwards G.A., and Charman W.N. Susceptibility to lipase-mediated digestion reduces the oral bioavailability of danazol after administration as a medium-chain lipid-based microemulsion formulation. Pharm. Res. 21 (2004) 1405-1412
    • (2004) Pharm. Res. , vol.21 , pp. 1405-1412
    • Porter, C.J.1    Kaukonen, A.M.2    Boyd, B.J.3    Edwards, G.A.4    Charman, W.N.5
  • 28
    • 0033805858 scopus 로고    scopus 로고
    • Lipid formulations for oral administration of drugs: non-emulsifying, self-emulsifying and 'self-microemulsifying' drug delivery systems
    • Pouton C.W. Lipid formulations for oral administration of drugs: non-emulsifying, self-emulsifying and 'self-microemulsifying' drug delivery systems. Eur. J. Pharm. Sci. 11 (2000) S93-S98
    • (2000) Eur. J. Pharm. Sci. , vol.11
    • Pouton, C.W.1
  • 29
    • 33751014029 scopus 로고    scopus 로고
    • Formulation of poorly water-soluble drugs for oral administration: physicochemical and physiological issues and the lipid formulation classification system
    • Pouton C.W. Formulation of poorly water-soluble drugs for oral administration: physicochemical and physiological issues and the lipid formulation classification system. Eur. J. Pharm. Sci. 29 (2006) 278-287
    • (2006) Eur. J. Pharm. Sci. , vol.29 , pp. 278-287
    • Pouton, C.W.1
  • 30
    • 33744787859 scopus 로고    scopus 로고
    • Examination of the impact of a range of Pluronic surfactants on the in-vitro solubilisation behavior and oral bioavailability of lipidic formulations of atovaquone
    • Sek L., Boyd B.J., Charman W.N., and Porter C.J. Examination of the impact of a range of Pluronic surfactants on the in-vitro solubilisation behavior and oral bioavailability of lipidic formulations of atovaquone. J. Pharm. Pharmacol. 58 (2006) 809-820
    • (2006) J. Pharm. Pharmacol. , vol.58 , pp. 809-820
    • Sek, L.1    Boyd, B.J.2    Charman, W.N.3    Porter, C.J.4
  • 31
    • 33748290093 scopus 로고    scopus 로고
    • Preparation and evaluation of self-microemulsifying drug delivery systems (SMEDDS) containing atorvastatin
    • Shen H., and Zhong M. Preparation and evaluation of self-microemulsifying drug delivery systems (SMEDDS) containing atorvastatin. J. Pharm. Pharmacol. 58 (2006) 1183-1191
    • (2006) J. Pharm. Pharmacol. , vol.58 , pp. 1183-1191
    • Shen, H.1    Zhong, M.2
  • 32
    • 3543106201 scopus 로고    scopus 로고
    • Influence of lipolysis and droplet size on tocotrienol absorption from self-emulsifying formulations
    • Yap S.P., and Yuen K.H. Influence of lipolysis and droplet size on tocotrienol absorption from self-emulsifying formulations. Int. J. Pharm. 281 (2004) 67-78
    • (2004) Int. J. Pharm. , vol.281 , pp. 67-78
    • Yap, S.P.1    Yuen, K.H.2


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.