Evaluation of poly(styrene-alt-maleic anhydride)-ethanol as enteric coating material

International Journal of Pharmaceutics

Volumn 352, Issue 1-2, 2008, Pages 66-73

  Lai, Xiaolin ^a,b   Sun, Chengdong ^a,b   Tian, Hua ^a,b   Zhao, Wenjun ^a   Gao, Lin ^a  

^a XINJIANG TECHNICAL INSTITUTE OF PHYSICS AND CHEMISTRY   (China)

^b UNIVERSITY OF CHINESE ACADEMY OF SCIENCES   (China)

Author keywords

Enteric coating; Erythromycin tablets; SMA ethanol

Indexed keywords

ALCOHOL; ERYTHROMYCIN; PLASTICIZER; STYRENE MALEIC ANHYDRIDE COPOLYMER;

ARTICLE; DRUG RELEASE; DRUG SCREENING; DRUG SYNTHESIS; ENTERIC COATED TABLET; IN VITRO STUDY; MATERIAL COATING; MOISTURE; MOLECULAR WEIGHT; PH MEASUREMENT; PHYSICAL CHEMISTRY; PRIORITY JOURNAL; TENSILE STRENGTH; THERMAL ANALYSIS; TOPOGRAPHY; WATER VAPOR;

ANTI-BACTERIAL AGENTS; CHEMISTRY, PHARMACEUTICAL; DIBUTYL PHTHALATE; DRUG COMPOUNDING; ERYTHROMYCIN; ETHANOL; HYDROGEN-ION CONCENTRATION; KINETICS; MALEATES; MICROSCOPY, ELECTRON, SCANNING; MOLECULAR WEIGHT; PLASTICIZERS; POLYSTYRENES; SOLUBILITY; SURFACE PROPERTIES; TABLETS, ENTERIC-COATED; TECHNOLOGY, PHARMACEUTICAL; TENSILE STRENGTH; VOLATILIZATION; WATER;

EID: 39449089160     PISSN: 03785173     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.ijpharm.2007.10.011     Document Type: Article

References (18)

1. Baldrick P. Pharmaceutical excipient development: the need for preclinical guidance. Regul. Toxicol. Pharm. 32 (2000) 210-218
2. Dana M., Villenave J.J., and Montaudon E. Correlation entre architecture moleculaire et adhesion thermodynamique: copolymeres (anhydride maleique-co-styrene) modifies. Eur. Polym. J. 34 (1998) 1309-1313
3. Dimantov A., Greenberg M., Kesselman E., and Shimoni E. Study of high amylose corn starch as food grade enteric coating in a microcapsule model system. Innovative Food Sci. Emer. Technol. 5 (2004) 93-100
4. Guha S.K., Singh G., Srivastava A., Das H.C., Bhardwaj J.C., Mathur V., Koul V., Malhotra R.L., and Das S.K. Two-year clinical efficacy trial with dose variations of a vas deferens injectable contraceptive for the male. Contraception 58 (1998) 165-174
5. Jeonga J.-H., Byounb Y.-S., and Leea Y.-S. Poly(styrene-alt-maleic anhydride)-4-aminophenol conjugate synthesis and antibacterial activity. React. Funct. Polym. 50 (2002) 257-263
6. Kalcic I., Zorc B., and Butula I. Macromolecular prodrugs. Polymer-dopamine conjugates. Int. J. Pharm. 4 (1996) S109
7. Limmatvapirat S., Limmatvapirat C., Luangtana-anan M., Nunthanid J., Oguchi T., Tozuka Y., Yamamoto K., and Puttipipatkhachorn S. Modification of physicochemical and mechanical properties of shellac by partial hydrolysis. Int. J. Pharm. 278 (2004) 41-49
8. Maeda H. SMANCS and polymer-conjugated macromolecular drugs: advantages in cancer chemotherapy. Adv. Drug Deliver Rev. 46 (2001) 169-185
9. Patel M., Patel J.M., and Lemberger A.P. Water vapour permeation of selected cellulose ester films. J. Pharm. Sci. 53 (1964) 286-290
10. Pearnchob N., Dashevsky A., and Bodmeier R. Improvement in the disintegration of shellac-coated soft gelatin capsules in simulated intestinal fluid. J. Control Release 94 (2004) 313-321
11. Satturwar P.M., Fulzele S.V., Panyam J., Mandaogade P.M., Mundhada D.R., Gogte B.B., Labhasetwar V., and Dorle A.K. Evaluation of new rosin derivatives for pharmaceutical coating. Int. J. Pharm. 270 (2004) 27-36
12. Sethi N., Board Path., Srivastava R.K., and Singh R.K. Safety evaluation of a male injectable antifertility agent, styrene maleic anhydride, in rats. Contraception 39 (1989) 217-226
13. Sethi N., Srivastava R.K., and Singh R.K. Histological changes in the vas deferens of rats after injection of a new male antifertility agent "SMA" and its reversibility. Contraception 41 (1990) 333-339
14. Sethi N., Srivastava R.K., and Singh R.K. Male mediated teratogenic potential evaluation of new antifertility compound SMA in rabbit. Contraception 42 (1990) 215-223
15. Shulkin A., and Stover H.D.H. Microcapsules from styrene-maleic anhydride copolymers: study of morphology and release behavior. J. Membr. Sci. 209 (2002) 433-444
16. Thoma K., and Bechtold K. Influence of aqueous coatings on the stability of enteric coated pellets and tablets. Eur. J. Pharm. Biopharm. 47 (1999) 39-50
17. Utsumi I., Ida T., Takahashi T., and Sugimoto N. Water vapour transmission properties of polymeric materials. J. Pharm. Sci. 50 (1961) 592-597
18. Veronese F.M., and Morpurgo M. Bioconjugation in pharmaceutical chemistry. IL Farmaco 54 (1999) 497-516