QSAR studies on CCR2 antagonists with chiral sensitive hologram descriptors

Bioorganic and Medicinal Chemistry Letters

Volumn 18, Issue 4, 2008, Pages 1323-1330

  Nair, Pramod C ^a   Srikanth, K ^a   Sobhia, M Elizabeth ^a  

^a NATIONAL INSTITUTE OF PHARMACEUTICAL EDUCATION AND RESEARCH NIPER   (India)

Author keywords

CCR2; Chemokines; Enantiopure; Fragments; HQSAR

Indexed keywords

3 AMINO 1 CYCLOPENTANE CARBOXAMIDE; ALPHA AMINOTHIAZOLE ALPHA AMINOBUTANOIC AMIDE; BUTYRAMIDE DERIVATIVE; CHEMOKINE RECEPTOR ANTAGONIST; CHEMOKINE RECEPTOR CCR2; GLYCINAMIDE; UNCLASSIFIED DRUG;

ARTICLE; CHIRALITY; HUMAN; HUMAN CELL; PHARMACOPHORE; QUANTITATIVE STRUCTURE ACTIVITY RELATION;

AMIDES; ANIMALS; DRUG DESIGN; HOLOGRAPHY; HUMANS; INHIBITORY CONCENTRATION 50; MODELS, MOLECULAR; QUANTITATIVE STRUCTURE-ACTIVITY RELATIONSHIP; RECEPTORS, CCR2; STEREOISOMERISM;

EID: 38949111736     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2008.01.023     Document Type: Article

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