Screening for polymorphs on polymer microarrays

Journal of Combinatorial Chemistry

Volumn 10, Issue 1, 2008, Pages 24-27

  Liberski, Albert R ^a   Tizzard, Graham J ^b   Diaz Mochon, Juan J ^a   Hursthouse, Michael B ^b   Milnes, Phillip ^a   Bradley, Mark ^a  

^a UNIVERSITY OF EDINBURGH   (United Kingdom)

^b UNIVERSITY OF SOUTHAMPTON   (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

DRUG; POLYMER;

ARTICLE; CHEMISTRY; COMBINATORIAL CHEMISTRY; CRYSTALLIZATION; MICROARRAY ANALYSIS; MOLECULAR LIBRARY; RAMAN SPECTROMETRY;

COMBINATORIAL CHEMISTRY TECHNIQUES; CRYSTALLIZATION; MICROARRAY ANALYSIS; PHARMACEUTICAL PREPARATIONS; POLYMERS; SMALL MOLECULE LIBRARIES; SPECTRUM ANALYSIS, RAMAN;

EID: 38849175380     PISSN: 15204766     EISSN: None     Source Type: Journal    
DOI: 10.1021/cc700107x     Document Type: Article

References (37)

1. Morissette, S. L.; Soukasene, S.; Levinson, D.; Cima, M. J.; Almarsson, Ö. Proc. Natl. Acad. Sci. 2006, 100, 2180-2184.
2. Yu, L. X.; Furness, M. S.; Raw, A.; Woodland Outlaw, K. P.; Nashed, N. E.; Ramos, E.; Miller, S. P. F.; Adams, R. C.; Fang, F.; Patel, R. M.; Holcombe, F. O., Jr.; Chiu, Y.; Hussain, A. S Pharm. Res. 2003, 20, 531-536.
3. Yu, L. X.; Ellison, C. D.; Hussain, A. S. Predicting human oral bioavailability using in silico models. In Applications of Pharmacokinetic Principles in Drug Development; Krishna, R. Ed.; Springer: New York, 2003; pp 53-75
4. Price, C. P.; Grzesiak, A. L.; Matzger, A. J. J. Am. Chem. Soc. 2005, 127, 5512-5517.
5. Day, G. M.; Trask, A. V.; Motherwell, W. D. S.; Jones, W. Chem. Commun. 2006, 1, 54-56.
6. Vishweshwar, P.; McMahon, J. A.; Paterson, M. L.; Zawratko, M. J. J. Am. Chem. Soc. 2005, 127, 16802-16803.
7. McCrone's often quoted pronouncement is "The number of forms known for a given compound is proportional to the time and money spent in research on that compound." See: McCrone, W. C. Polymorphism. In Physics and Chemistry of the Organic Solid State; Fox, D., Ed.; John Wiley & Sons, Inc.: New York, 1965; pp. 726-767.
8. Dunitz, J. D.; Bernstein, J. Ace. Chem. Res. 1995, 28, 193-200.
9. Peterson, M. L.; Morissette, S. L.; McNulty, C.; Goldsweig, A.; Shaw, P.; LeQuesne, M.; Monagle, J.; Encina, N.; Marchionna, J.; Johnson, A.; Gonzalez-Zugasti, J.; Lemmo, A. V.; Ellis, S. J.; Cima, M. J.; Almarsson, Ö. J. Am. Chem. Soc. 2002, 124, 10958-10959.
10. Aizenberg, J.; Black, A. J.; Whitesides, G. M. J. Am. Chem. Soc. 1999, 121, 4500-4509.
11. (a) Han, Y.; Wysocki, L. M.; Thanawala, M. S.; Siegrist, T.; Aizenberg, J. Angew. Chem., Int. Ed. 2005, 44, 2386-2390.
12. (b) Ichikawa, K.; Shimomura, N.; Yamada, M.; Ohkubo, N. Chem-Eur. J. 2003, 9, 3235-3241.
13. Aizenberg, J.; Black, A. J.; Whitesides, G. M. Nature 1999, 398, 495-498.
14. Lang, M.; Grzesiak, A. L.; Matzger, A. J. J. Am. Chem. Soc. 2002, 124, 14834-14835.
15. Chan, K. L. A.; Kazarian, G. J. Comb. Chem. 2005, 185-189.
16. Cabeza, A. J. C.; Day, G. M.; Motherwell, W. D.; Jones, W. Chem. Commun. 2007, 16, 1600-1602.
17. Kogermann, K.; Aaltonen, J.; Strachan, C. J.; Pöllänen, K.; Veski, P.; Heinämäki, J.; Yliruusi, J.; Rantane, J. J. Pharm. Sci. 2007, 96, 1802-1820.
18. Wyttenbach, N.; Alsenz, J.; Grassmann, O. Pharm. Res. 2007, 24, 888-898.
19. Tian, F.; Sandler, N.; Aaltonen, J.; Lang, C.; Saville, D. J.; Gordon, K. C.; Strachan, C. J.; Rantanen, J.; Rades, T. J. Pharm. Sci. 2007, 96, 584-594.
20. Kipouros, K.; Kachrimanis, K.; Nikolakakis, I.; Tserki, V.; Malamataris, S. J. Pharm. Sci. 2006, 95, 2419-2431.
21. Rama, M. J. R.; López-Sánchez, M.; Ruiz-Medina, A.; MolinaDíaz, A.; Ayora-Caflada, M. J. Analyst 2005, 130, 1617-1623.
22. Takasuka, M.; Nakai, H. Vib. Spectrosc. 2001, 25, 197-204.
23. Karthikeyan, G.; Mohanraj, K.; Elango, K. P.; Girishkumar, K. Russ. J. Coord. Chem. 2006, 32, 380-385.
24. Göbel, A.; Thomsen, A.; Mcardell, C. S.; Joss, A.; Giger, W. Environ. Sci. Technol. 2005, 39, 3981-3989.
25. Zhang, C-L.; Wang, F.-A.; Wang, Y. J. Chem. Eng. Data 2007, 52, 1563-1566.
26. McKinnon, J. J.; Fabbiani, F. P. A.; Spackman, M. A. Cryst. Growth Des. 2007, 7, 755-769.
27. Li, H.; Stowell, J. G.; Borchardt, T. B.; Byrn, S. R. Cryst. Growth Des. 2006, 6, 2469-2474.
28. Smith, J. R.; Xu, W.; Raftery, D. 7. Phys. Chem. B 2006, 110, 7766-7776.
29. Chen, S.; Xi, H.; Yu, L. J. Am. Chem. Soc. 2005, 127, 17439-17444.
30. Dunitz, J. D.; Gavezzotti, A. Cryst. Growth Des. 2005, 5, 2180-2189.
31. Chen, S.; Guzei, I. A.; Yu, L. J. Am. Chem. Soc. 2005, 127, 9881-9885.
32. Grzesiak, A. L.; Lang, M.; Kim, K.; Matzger, A. J. J. Pharm. Sci. 2003, 92, 2260-2271.
33. Tian, F.; Zeitler, J. A.; Strachan, C. J.; Saville, D. J.; Gordon, K. C.; Rades, T. J. Pharm. Biomed. Anal. 2006, 40, 271-280.
34. Lang, M.; Kampf, J. W.; Matzger, A. J. J. Pharm. Sci. 2002, 91, 1186-1190.
35. O'Brien, L. E.; Timmins, P.; Williams, A. C.; York, P. J. Pharm. Biomed. Anal. 2004, 36, 335-340.
36. Momany, F. A.; Sessa, D. J.; Lawton, J. W.; Selling, G. W.; Hamaker, S. A. H.; Willett, J. L. J. Agric. Food Chem. 2006, 54, 543-547.
37. Morissette, S. L.; Almarsson, Ö.; Peterson, M. L.; Remenar, J. F.; Read, M. J.; Lemmo, A. V.; Ellis, S.; Cima, M. J.; Gardner, C. R. Adv. Drug Delivery Rev. 2004, 56, 275-300.