Synthesis, structure and biological activity of pseudopeptidic macrolides based on an amino alcohol

European Journal of Medicinal Chemistry

Volumn 43, Issue 1, 2008, Pages 19-24

  Lv, Jian ^a   Liu, Tingting ^b   Wang, Yongmei ^a  

^a NANKAI UNIVERSITY   (China)

^b SHENYANG PHARMACEUTICAL UNIVERSITY   (China)

Author keywords

Amino alcohol; Antibacterial activity; Antifungal activity; Hemolytic activity; Pseudopeptidic macrolides

Indexed keywords

AMINOALCOHOL; AMPHOTERICIN B; CHLORAMPHENICOL; FLUCONAZOLE; MACROLIDE; PSEUDOPEPTIDE;

ANTIBACTERIAL ACTIVITY; ANTIFUNGAL ACTIVITY; ARTICLE; ASPERGILLUS FLAVUS; ASPERGILLUS NIGER; BACILLUS SUBTILIS; BIOLOGICAL ACTIVITY; CANDIDA ALBICANS; CONTROLLED STUDY; CRYPTOCOCCUS NEOFORMANS; DRUG CYTOTOXICITY; DRUG STRUCTURE; DRUG SYNTHESIS; ESCHERICHIA COLI; HEMOLYSIS; HUMAN; HUMAN CELL; MINIMUM INHIBITORY CONCENTRATION; NONHUMAN; PSEUDOMONAS AERUGINOSA; SACCHAROMYCES CEREVISIAE; STAPHYLOCOCCUS AUREUS; STRUCTURE ACTIVITY RELATION; X RAY DIFFRACTION;

AMINO ALCOHOLS; ANTI-INFECTIVE AGENTS; CRYSTALLOGRAPHY, X-RAY; FUNGI; GRAM-NEGATIVE BACTERIA; GRAM-POSITIVE BACTERIA; HEMOLYSIS; MACROLIDES; MICROBIAL SENSITIVITY TESTS; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 38149140965     PISSN: 02235234     EISSN: 17683254     Source Type: Journal    
DOI: 10.1016/j.ejmech.2007.03.011     Document Type: Article

References (19)

1. Minassian B., Huczko E., Washo T., Bonner D., and Fung-Tomc J. Clin. Microbiol. Infect. 9 (2003) 1250
2. Ostrosky-Zeichner L., Rex J.H., Pappas P.G., Hamill R.J., Larsen R.A., Horowitz H.W., Powderly W.G., Hyslop N., Kauffman C.A., Cleary J., Mangino J.E., and Lee J. Antimicrob. Agents Chemother. 47 (2003) 3149
3. Pfaller M.A., Diekema D.J., Messer S.A., Boyken L., Hollis R.J., and Jones R.N. Diagn. Microbiol. Infect. Dis. 48 (2004) 101
4. Rees J.R., Pinner R.W., Hajjeh R.A., Brandt M.E., and Reingold A.L. Clin. Infect. Dis. 27 (1998) 1138
5. Hegde V.R., Patel M.G., Gullo V.P., Ganguly A.K., Sarre O., Puar M.S., and Mcphail A.T. J. Am. Chem. Soc. 112 (1990) 6403
6. De Lucca A.J., and Walsh T.J. Antimicrob. Agents Chemother. 43 (1999) 1
7. Uchida K., Yokota N., and Yamaguchi H. Int. J. Antimicrob. Agents 18 (2001) 167
8. Roxburgh C.J. Tetrahedron 51 (1995) 9767
9. Frensch V.K., and Vögtle F. Tetrahedron Lett. 18 (1977) 2573
10. Kuroda T., Imashiro R., and Seki M. J. Org. Chem. 65 (2000) 4213
11. Groves J.T., and Viski P. J. Org. Chem. 55 (1990) 3628
12. Helgson R.C., Koga K., Timko J.M., and Cram D.J. J. Am. Chem. Soc. 95 (1973) 3021
13. Gasparrini F., Misiti D., Villani C., Borchardt A., Burger M.T., and Still W.C. J. Org. Chem. 60 (1995) 4314
14. Breslow R., Czarnik A.W., Lauer M., Leppkes R., Winkler J., and Zimmerman S. J. Am. Chem. Soc. 108 (1986) 1969
15. Zhao H., and Hua W. J. Org. Chem. 65 (2000) 2933
16. Gao M.Zh., Gao J., Xu Z.L., and Zingaro R.A. Tetrahedron Lett. 43 (2002) 5001
17. Jiang M., Dalgarno S., Kilner C.A., Halcrow M.A., and Kee T.P. Polyhedron 20 (2001) 2151
18. Reference Method for Broth Dilution Susceptibility Testing of Yeasts: Approved Standard. NCCLS document M27A (1997), National Committee for Clinical Laboratory Standards, Wayne, PA
19. Reference Method for Broth Dilution Susceptibility Testing of Filamentous Fungi: Approved Standard. NCCLS document M38-A (2002), National Committee for Clinical Laboratory Standards, Wayne, PA