Interactions between antiplasmodial 3,6-diamino-1′-dimethyl-9- anilinoacridine and hematin and concanamycin A

Southeast Asian Journal of Tropical Medicine and Public Health

Volumn 38, Issue 6, 2007, Pages 979-982

  Auparakkitanon, Saranya ^a   Poonchareon, Kritchai ^b   Sopitthummakhun, Kittipat ^b   Wilairat, Prapon ^b  

^a MAHIDOL UNIVERSITY   (Thailand)

^b MAHIDOL UNIVERSITY   (Thailand)

Author keywords

[No Author keywords available]

Indexed keywords

EID: 37849020756     PISSN: 01251562     EISSN: 26975718     Source Type: Journal    
DOI: None     Document Type: Article

References (10)

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3. Auparakkitanon S, Noonpakdee W, Ralph RK, Denny WA, Wilairat P. Antimalarial 9-anilinoacridine compounds directed at hematin. Antimicrobial Agents Chemother 2003; 47: 3708-12.
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5. Gamage SA, Tepsiri N, Wilairat P, et al. Synthesis and in vitro evaluation of 9-anilino-3,6-diaminoacridines active against a multidrug-resistant strain of the malaria parasite Plasmodium falciparum. J Med Chem 1994; 37: 1486-94.
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7. +-pyrophosphatase. J Biol Chem 2003; 278: 5605-12.
8. Solomonov I, Osipova M, Feldman Y, et al. Crystal nucleation, growth, and morphology of the synthetic malaria pigment β-hematin and the effect thereon by quinoline additives: the malaria pigment as a target of various antimalarial drugs. J Am Chem Soc 2007; 129: 2615-27.
9. Tilley L, Loria P, Foley M. Chloroquine and other quinoline antimalarials. In: Rosenthal PJ, ed. Antimalarial chemotherapy: mechanisms of action, resistance, and new directions in drug discovery. New Jersey: Humana Press, 2001: 87-121.
10. Trager W, Jensen JB. Human malarial parasites in continuous culture. Science 1976; 193: 673-5.