Modulation of a pulsatile release drug delivery system using different swellable/rupturable materials

Drug Delivery

Volumn 14, Issue 8, 2007, Pages 539-546

  El Maradny, Hoda A ^a  

^a Alexandria University Faculty of Pharmacy   (Egypt)

Author keywords

Pulsatile Release Drug Delivery System; Rupturable Coating Substance; Swelling Materials

Indexed keywords

CROSCARMELLOSE SODIUM; DICLOFENAC; ETHYL CELLULOSE; EXCIPIENT; LACTOSE; LUDIPRESS; MICROCRYSTALLINE CELLULOSE; STA RX 1500; STARCH GLYCOLATE SODIUM; UNCLASSIFIED DRUG;

ARTICLE; DRUG COATING; DRUG DELIVERY SYSTEM; DRUG RELEASE; PRIORITY JOURNAL; SCANNING ELECTRON MICROSCOPY; TABLET COMPRESSION; TABLET FORMULATION;

CARBOXYMETHYLCELLULOSE; CELLULOSE; DELAYED-ACTION PREPARATIONS; DICLOFENAC; DRUG DELIVERY SYSTEMS; EXCIPIENTS; MICROSCOPY, ELECTRON, SCANNING; POLYVINYLS; PYRROLIDINES; STARCH; SURFACE PROPERTIES; TABLETS; TRIACETIN; WATER;

EID: 36248953831     PISSN: 10717544     EISSN: 15210464     Source Type: Journal    
DOI: 10.1080/10717540701606574     Document Type: Article

References (20)

1. Bussemer, T., and Bodmeier, R. 2001. A review of pulsatile drug delivery. Am. Pharm. Rev. 4(4):18-24.
2. Bussemer, T., Dashevsky, A., and Bodmeier, R. 2003. A pulsatile drug delivery system based on rupturable coated hard gelatin capsules. J. Control. Rel. 93:331-339.
3. Bussemer, T., Otto, L., and Bodmeier, R. 2001. Pulsatile-drug delivery systems. Crit. Rev. Ther. Drug Carrier Syst. 18(5):433-458.
4. Efentakis, M., Koligliati, S., and Vlachou, M. 2006. Design and evaluation of a dry coated drug delivery system with an impermeable cup, swellable top layer and pulsatile release. Int. J. Pharm. 311:147-156.
5. Fan, T. Y., Wei, S. L., Yan, W. W., Chen, D. B., and Li, J. 2001. An investigation of pulsatile release tablets with ethylcellulose and Eudragit L as film coating materials and cross-linked polyvinylpyrrolidone in core tablets. J. Control. Rel. 77:245-251.
6. Freichel, O. L., and Lippold, B. C. 2000. A new oral erosion controlled drug delivery system with a late burst in the release profile. Eur. J. Pharm. Biopharm. 50:345-351.
7. Karavas, E., Georgarakis, E., and Bikiaris, D. 2006a. Application of PVP/HPMC miscible blends with enhanced mucoadhesive properties for adjusting drug release in predictable pulsatile chronotherapeutics. Eur. J. Pharm. Biopharm. 64(1):115-126.
8. Karavas, E., Georgarakis, E., and Bikiaris, D. 2006b. Felodipine nanodispersions as active core for predictable pulsatile chronotherapeutics using PVP/HPMC blends as coating layer. Int. J. Pharm. 313(1-2):189-197.
9. Kr̈ogel, I., and Bodmeier, R. 1999a. Evaluation of an enzyme-containing capsular shaped pulsatile drug delivery system. Pharm. Res. 16(9):1424-1429.
10. Kr̈ogel, I., and Bodmeier, R. 1999b. Floating or pulsatile drug delivery systems based on coating effervescent cores. Int. J. Pharm. 187:175-184.
11. Lemmer, B. 1999. Chronopharmacokinetic: implications for drug treatment. J. Pharm. Pharmacol. 51:887-890.
12. Li, Y. H., and Zhu, J. B. 2002. Oral site-specific drug delivery system, World pharmacy- a branch of synthetic drug. Biochem. Drug Pharmac. 23(4):225-228.
13. Maggi, L., Conte, U., Giunchedi, P., and Colombo, P. 1993. Press-coated tablets for the sequential pulsed administration of two different drugs. Int. J. Pharm. 99:173-179.
14. Morita, R., Honda, R., and Takahashi, Y. 2000. Development of oral controlled release preparations, a PVA swelling controlled release system (SCRS); I. Design of SCRS and its release controlling factor. J. Control. Rel. 63:297-304.
15. Sangalli, M. E., Maroni, A., Zema, L., Busetti, C., Giordano, F., and Gazzaniga, A. 2001. In-vitro and in-vivo evaluation of an oral system for time and/or site-specific drug delivery. J. Control. Rel. 73:103-110.
16. Sinha, V. R., Bhinge, J. R., Kumria, R., and Kumar, M. 2006. Development of pulsatile systems for targeted drug delivery of celecoxib for prophylaxis of colorectal cancer. Drug Del. 13(3):221-225.
17. Sungthongjeen, S., Puttipipatkhachorn, S., Paeratakul, O., Dashevsky, A., and Bodmeier, R. 2004. Development of pulsatile release tablets with swelling and rupturable layers. J. Control. Rel. 95:147-159.
18. Thombre, A. G., Appel, L. E., Chidlaw, M. B., Daugherity, P. D., Dumont, F., Evans, L. A. F., and Sutton, S. C. 2004. Osmotic drug delivery using swellable-core technology. J. Control. Rel. 94:75-89.
19. Ueda, S., Ibuki, R., Kimura, S., Murata, S., Takahashi, T., Tokunaga, Y., and Hata, T. 1994. Development of a novel release system, time controlled explosion system (TES). III. Relation between lag time and membrane thickness. Chem. Pharm. Bull. 42(2):364-367.
20. Wan, L. S., and Lim, L. Y. 1992. Drug release from heat-treated polyvinyl alcohol films. Drug Dev. Ind. Pharm. 18:1895-1906.