Synthesis of symmetrical C- and pseudo-symmetrical O-linked disaccharide analogs for arabinosyltransferase inhibitory activity in Mycobacterium tuberculosis

Bioorganic and Medicinal Chemistry Letters

Volumn 17, Issue 16, 2007, Pages 4527-4530

  Pathak, Ashish K ^a   Pathak, Vibha ^a   Riordan, James R ^a   Suling, William J ^a   Gurcha, Sudagar S ^b   Besra, Gurdyal S ^b   Reynolds, Robert C ^a  

^a SOUTHERN RESEARCH INSTITUTE   (United States)

^b UNIVERSITY OF BIRMINGHAM   (United Kingdom)

Author keywords

Disaccharides; Glycosyltransferases; Inhibitors; Tuberculosis

Indexed keywords

ANTIINFECTIVE AGENT; ARABINOFURANOSE; ARABINOSE; BACTERIAL ENZYME; DISACCHARIDE; GALACTOFURANOSE; RHAMNOPYRANOSE; UNCLASSIFIED DRUG;

ARTICLE; COLORIMETRY; DILUTION; DRUG SYNTHESIS; IN VITRO STUDY; MYCOBACTERIUM AVIUM; MYCOBACTERIUM TUBERCULOSIS; PROTEIN DETERMINATION; PROTEIN STRUCTURE;

ANTITUBERCULAR AGENTS; DISACCHARIDES; MYCOBACTERIUM TUBERCULOSIS; PENTOSYLTRANSFERASES;

MYCOBACTERIUM AVIUM; MYCOBACTERIUM TUBERCULOSIS;

EID: 34447319963     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2007.05.099     Document Type: Article

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