Duplexed, bead-based competitive assay for inhibitors of protein kinases

Cytometry Part A

Volumn 71, Issue 7, 2007, Pages 451-459

  Simons, Peter C ^a,b   Young, Susan M ^a,b   Gibaja, Veronica ^c   Lee, Wen Cherng ^c   Josiah, Serene ^c   Edwards, Bruce S ^a,b   Sklar, Larry A ^a,b,d  

^a UNIVERSITY OF NEW MEXICO HEALTH SCIENCES CENTER   (United States)

^b UNIVERSITY OF NEW MEXICO   (United States)

^c BIOGEN   (United States)

^d UNIVERSITY OF NEW MEXICO SCHOOL OF MEDICINE   (United States)

Author keywords

ALK4; ALK5; Bead based; High throughput; Kinase inhibitor; Protein kinase

Indexed keywords

ACTIVIN RECEPTOR LIKE KINASE 4; ADENOSINE TRIPHOSPHATE; FLUORESCENT KINASE LIGAND; HEXAHISTIDINE; NICKEL; PROTEIN KINASE; PROTEIN KINASE INHIBITOR; TRANSFORMING GROWTH FACTOR BETA RECEPTOR 1; UNCLASSIFIED DRUG;

ARTICLE; BINDING AFFINITY; BINDING SITE; BRIGHTNESS; ENZYME ACTIVITY; ENZYME ASSAY; ENZYME BINDING; ENZYME INHIBITION; ENZYME PURIFICATION; FLOW CYTOMETRY; FLUORESCENCE POLARIZATION; PRIORITY JOURNAL; PROTEIN EXPRESSION; SIGNAL TRANSDUCTION;

ACTIVIN RECEPTORS, TYPE I; ADENOSINE TRIPHOSPHATE; BINDING, COMPETITIVE; FLOW CYTOMETRY; GREEN FLUORESCENT PROTEINS; HISTIDINE; HUMANS; LIGANDS; MICROSPHERES; NICKEL; OLIGOPEPTIDES; PROTEIN BINDING; PROTEIN KINASE INHIBITORS; RECEPTORS, TRANSFORMING GROWTH FACTOR BETA; RECOMBINANT PROTEINS;

EID: 34447129552     PISSN: 15524922     EISSN: 15524930     Source Type: Journal    
DOI: 10.1002/cyto.a.20398     Document Type: Article

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