Mechanistic study on hydration and drug release behavior of sodium alginate compacts

Drug Development and Industrial Pharmacy

Volumn 33, Issue 6, 2007, Pages 667-676

  Chan, Lai Wah ^a   Ching, Ai Ling ^a   Liew, Celine Valeria ^a   Heng, Paul Wan Sia ^a  

^a NATIONAL UNIVERSITY OF SINGAPORE   (Singapore)

Author keywords

Alginate; Anisotropy; Dimensional changes; Solvent penetration front; Viscosity

Indexed keywords

ALGINIC ACID; POLYMER; SOLVENT;

ANISOTROPY; ARTICLE; DRUG PENETRATION; DRUG RELEASE; DRUG SOLUBILITY; GEL; HYDRATION; MATRIX TABLET; PH; TABLET; TENSION; VISCOSITY;

ALGINATES; ANISOTROPY; CHEMISTRY, PHARMACEUTICAL; CHLORPHENIRAMINE; DELAYED-ACTION PREPARATIONS; DRUG CARRIERS; GLUCURONIC ACID; HEXURONIC ACIDS; HYDROGEN-ION CONCENTRATION; KINETICS; SOLUBILITY; TABLETS; VISCOSITY;

EID: 34447123239     PISSN: 03639045     EISSN: 15205762     Source Type: Journal    
DOI: 10.1080/03639040600943814     Document Type: Article

References (22)

1. Alderborn, G., & Nyström, C. (1984). Radial and axial tensile strength and strength variability of paracetamol tablets. Acta Pharm. Suec., 21, 1-8.
2. Brondsted, H., & Kopecek, J. (1992). pH-sensitive hydrogels. In Polyelectrolyte Gels: Properties, Preparation and Applications; Harland, R.S., & Prud'homme, R.K., Ed.; American Chemical Society: Washington, DC, 285-304.
3. Colombo, P., Bettini, R., Massimo, G., Catellani, P. L., & Peppas, N. A. (1995). Drug diffusion front movement is important in drugrelease control from swellable matrix tablets. J. Pharm. Sci., 84, 991-997.
4. Colombo, P., Catellani, P. L., Peppas, N. A., Maggi, L., & Conte, U. (1992). Swelling characteristics of hydrophilic matrices for controlled-release: new dimensionless number to describe the swelling and release behavior. Int. J. Pharm., 88, 99-109.
5. Gao, P., & Meury, R. H. (1996). Swelling of hydroxypropyl methylcellulose matrix tablets. 1. Characterization of swelling using a novel optical imaging method. J. Pharm. Sci., 85, 725-731.
6. Gao, P., Skoug, J. W., Nixon, P. R., Ju, T. R., Stemm, N. L., & Sung, K.-C. (1996). Swelling of hydroxypropyl methylcellulose matrix tablets. 2. Mechanistic study of the influence of formulation variables on matrix performance and drug release. J. Pharm. Sci., 85, 732-740.
7. Goldhoff, R. M. (1971). Creep recovery in heat resistant steels. In Advances in Creep Design, the A. E. Johnson Memorial Volume; Smith, A.I., & Nicolson, A.M., Eds.; Applied Science Publishers: London, 81-109.
8. Haug, A. (1964). Composition and properties of alginates. Thesis. Norweigian institute of Technology, Trondheim.
9. Hodsdon, A. C., Mitchell, J. R., Davies, M. C., & Melia, C. D. (1995). Structure and behavior in hydrophilic matrix sustained release dosage forms: 3. The influence of pH on the sustained-release performance and internal gel structure of sodium alginate matrices. J. Control. Release, 33, 143-152.
10. Kanjickal, D. G., & Lopina, S. T. (2004). Modeling of drug release from polymeric delivery systems-A review. Crit. Rev. Ther. Drug., 21, 345-386.
11. Kavanagh, N, & Corrigan, O. I. (2004). Swelling and erosion properties of hydroxypropylmethylcellulose (Hypromellose) matrices -influence of agitation rate and dissolution medium composition. Int. J. Pharm., 279, 141-152.
12. Liew, C. V., Chan, L. W., Ching, A. L., & Heng, P. W. S. (2006). Evaluation of sodium alginate as drug release modifier in matrix tablets. Int. J. Pharm., 309, 25-37.
13. Malveau, C., Baille, W. E., Zhu, X. X., & Marchessault, R. H. (2002). NMR imaging of high-amylose starch tablets. 2. Effect of tablet size. Biomacromolecules, 3, 1249-1254.
14. Moussa, I. S., Lenaerts, V., & Cartilier, L. H. (1998). Image analysis studies of water transport and dimensional changes occurring in the early stages of hydration in cross-linked amylase matrices, J. Control. Release, 52, 63-70.
15. Papadimitriou, E., Buckton, G., & Efentakis, M. (1993). Probing the mechanisms of swelling of hydroxypropylmethylcellulose matrices. Int. J. Pharm., 98, 57-62.
16. Rajabi-Siahboomi, A. R., Bowtell, R. W., Mansfield, P., Henderson, A., Davies, M. C., & Melia C. D. (1994). Structure and behaviour in hydrophilic matrix sustained release dosage forms: 2. NMR-imaging studies of dimensional changes in the gel layer and core of HPMC tablets undergoing hydration. J. Control. Release, 31, 121-128.
17. Roy, D. S., Rohera, B. D. (2002). Comparative evaluation of rate of hydration and matrix erosion of HEC and HPC and study of drug release from their matrices. Eur. J. Pharm. Sci., 16, 193-199.
18. Siepmann, J., & Peppas, N. A. (2000). Hydrophilic matrices for controlled drug delivery: an improved mathematical model to predict the resulting drug release kinetics (the "Sequential Layer" model). Pharm. Res., 17, 1290-1298.
19. Streubel, A., Siepmann, J., Peppas, N. A., Bodmeier, R. (2000). Bimodal drug release achieved with multi-layer matrix tablets: transport mechanisms and device design. J. Control. Release, 69, 455-468.
20. Tahara, K., Yamamoto, K., & Nishihata, T. (1995). Overall mechanism behind matrix sustained release tablets prepared with hydroxypropyl methylcellulose 2910. J. Control. Release, 35, 59-66.
21. The United States Pharmacopeia (2002). Chapters < 711 > and < 724 >, United States Pharmacopeial Convention, Inc.: Rockville, MD.
22. Wan, L. S. C., Heng, P. W. S., & Wong, L. F. (1995). Matrix swelling: a simple model describing extent of swelling of HPMC matrices. Int. J. Pharm., 116, 159-168.