Synthesis and biological evaluation of new GnRH analogues on pituitary and breast cancer cells

International Journal of Peptide Research and Therapeutics

Volumn 13, Issue 1-2, 2007, Pages 143-149

  Zompra, Aikaterini A ^a   Magafa, Vassiliki ^a   Chryssanthi, Dimitra G ^a   Lamari, Fotini N ^a   Spyroulias, Georgios A ^a   Maina, Theodosia ^b   Nock, Berthold A ^b   Karamanos, Nikos K ^a   Cordopatis, Paul ^a  

^a UNIVERSITY OF PATRAS   (Greece)

^b INSTITUTE OF NANOSCIENCE AND NANOTECHNOLOGY   (Greece)

Author keywords

Breast cancer; GnRH; Leuprolide analogues; LHRH; Pituitary binding; Proliferation

Indexed keywords

2 AMINO 2 METHYLPROPIONIC ACID; 2 AMINO 4 PYRROLIDINOTHIENO[2,3 D]PYRIMIDINE 6 CARBOXYLIC ACID; ALANINE; CARBOXYLIC ACID DERIVATIVE; GLYCINE; GONADORELIN; GONADORELIN AGONIST; GONADORELIN DERIVATIVE; GONADORELIN RECEPTOR; LEUCINE; LEUPRORELIN; LYSINE; UNCLASSIFIED DRUG;

AMINO ACID ANALYSIS; AMINO ACID SEQUENCE; AMINO ACID SUBSTITUTION; AMINO TERMINAL SEQUENCE; ANIMAL CELL; ANTINEOPLASTIC ACTIVITY; ARTICLE; BINDING AFFINITY; BREAST ADENOCARCINOMA; BREAST CANCER; CANCER CELL; CANCER CELL CULTURE; CARBOXY TERMINAL SEQUENCE; CELL MEMBRANE; CELL PROLIFERATION; CELL STRAIN MCF 7; COVALENT BOND; DRUG EFFECT; DRUG POTENCY; DRUG SYNTHESIS; HUMAN; HUMAN CELL; MEMBRANE BINDING; MITOSIS INHIBITION; MOUSE; NONHUMAN; PROTEIN MODIFICATION; STRUCTURE ACTIVITY RELATION;

EID: 34249986876     PISSN: 15733149     EISSN: 15733904     Source Type: Journal    
DOI: 10.1007/s10989-006-9057-9     Document Type: Article

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