Caco-2 cell permeability and stability of two d-glucopyranuronamide conjugates of thyrotropin-releasing hormone

Bioorganic and Medicinal Chemistry

Volumn 15, Issue 14, 2007, Pages 4946-4950

  Wessling, Susanne T ^a   Ross, Benjamin P ^a   Koda, Yasuko ^a   Blanchfield, Joanne T ^a   Toth, Istvan ^a  

^a UNIVERSITY OF QUEENSLAND   (Australia)

Author keywords

Caco 2 cells; Drug delivery; Lipoamino acids; Sugar conjugation; TRH

Indexed keywords

2 AMINOOCTANOIC ACID GLUTAMINYLHISTIDYLPROLINE DEXTRO GLUCOPYRANURONAMIDE; PROTIRELIN DERIVATIVE; PYROGLUTAMYLHISTIDYLPROLINE DEXTRO GLUCOPYRANURONAMIDE; UNCLASSIFIED DRUG;

AMINO TERMINAL SEQUENCE; ARTICLE; CELL MEMBRANE PERMEABILITY; CELL STRAIN CACO 2; CONTROLLED STUDY; DRUG HALF LIFE; DRUG PENETRATION; DRUG STABILITY; HUMAN; HUMAN CELL; IN VITRO STUDY; INTESTINE EPITHELIUM CELL; LIPOPHILICITY; MONOLAYER CULTURE;

AMIDES; CACO-2 CELLS; CELL MEMBRANE PERMEABILITY; GLUCURONATES; HUMANS; MOLECULAR STRUCTURE; THYROTROPIN-RELEASING HORMONE;

EID: 34249658940     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmc.2007.04.042     Document Type: Article

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