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Volumn 9, Issue 10, 2007, Pages 2039-2042

Chemoselective amination of 5-bromo-2-chloro-3-fluoropyridine

Author keywords

[No Author keywords available]

Indexed keywords

5 BROMO 2 CHLORO 3 FLUOROPYRIDINE; 5-BROMO-2-CHLORO-3-FLUOROPYRIDINE; BROMIDE; CHLORIDE; FLUORINE; HALOGENATED HYDROCARBON; PYRIDINE; PYRIDINE DERIVATIVE; UNCLASSIFIED DRUG;

EID: 34249295533     PISSN: 15237060     EISSN: None     Source Type: Journal    
DOI: 10.1021/ol070695     Document Type: Article
Times cited : (14)

References (16)
  • 6
    • 32644435758 scopus 로고    scopus 로고
    • For other examples of selective animation of polyhalo substrates, see: a
    • For other examples of selective animation of polyhalo substrates, see: (a) Peng, Z.; Journet, M.; Humphrey, G. Org. Lett. 2006, 8, 395.
    • (2006) Org. Lett , vol.8 , pp. 395
    • Peng, Z.1    Journet, M.2    Humphrey, G.3
  • 11
    • 34249276421 scopus 로고    scopus 로고
    • For an example of carbanion addition to le at elevated temperatures, see WO2005005398.
    • For an example of carbanion addition to le at elevated temperatures, see WO2005005398.
  • 14
    • 0035799878 scopus 로고    scopus 로고
    • For an analogous result with 2-chloro-5-iodopyridine and a biscarbene ligand, see
    • For an analogous result with 2-chloro-5-iodopyridine and a biscarbene ligand, see: Cheng, J.; Trudell, M. L. Org. Lett. 2001, 3, 1371.
    • (2001) Org. Lett , vol.3 , pp. 1371
    • Cheng, J.1    Trudell, M.L.2
  • 15
    • 0034740448 scopus 로고    scopus 로고
    • a values are in the following rank order: piperidine (11.24) > [1,4]-oxazepine > phenyl piperazine > morpholine > bis(2-methoxyethyl)amine (8.67).
    • a values are in the following rank order: piperidine (11.24) > [1,4]-oxazepine > phenyl piperazine > morpholine > bis(2-methoxyethyl)amine (8.67).
  • 16
    • 12144276704 scopus 로고    scopus 로고
    • For an example of nucleophilic substitution of 3-fluoropyridine with imidazole, see
    • For an example of nucleophilic substitution of 3-fluoropyridine with imidazole, see: Denton, T.; Zhang, X.; Cashman, J. J. Med. Chem. 2005, 48, 224.
    • (2005) J. Med. Chem , vol.48 , pp. 224
    • Denton, T.1    Zhang, X.2    Cashman, J.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.