Synthesis and biological study of some novel 4-[5-(4,6-disubstituted-2- thiomethylpyrimidyl)-4'-amino-1,2,4- triazol-3'-yl] thioacetyl-3-arylsydnones

Phosphorus, Sulfur and Silicon and the Related Elements

Volumn 182, Issue 6, 2007, Pages 1393-1401

  Kalluraya, Balakrishna ^a   Lingappa, B ^a,b   Nooji, Satheesh Rai ^a  

^a MANGALORE UNIVERSITY   (India)

^b Strides Research and Specialty Chemicals Ltd   (India)

Author keywords

Biological activity; Pyrimidine; Sydnone; Triazoles

Indexed keywords

EID: 34247547879     PISSN: 10426507     EISSN: 15635325     Source Type: Journal    
DOI: 10.1080/10426500601161049     Document Type: Article

References (24)

1. J. Wichmann, A. Geo, S. Koclzewskis M. Vincent, and T. Woletring, Bioorg. Med. Chem. Lett., 9, 1513 (1999).
2. E. R. El-Bendary, M. A. El-Sherbeny, and F. A. Badri, Bull. Chem. Farm., 137, 115 (1998).
3. G. Kirpal, U. S. Patent, 5,869,494;
4. Chem. Abstr., 130,163202 (1999).
5. K. Tsuji and H. Ishikawa, Bioorg. Med. Chem. Lett., 4, 160 (1994).
6. W. Lie, Y.Tin, and P. G Wang, Chemtech., 2, 23 (1999).
7. R. S. Varma, Green Chem., 1, 43 (1999).
8. M. Kidwai, R.Venkatraman, R. K. Garg, and K. R. Bhushan, J. Chem. Res., 5, 586 (2000).
9. C. O. Kappe, W. M. F. Fabian, and M. A. Semones, Tetrahedron. 53, 2803 (1997).
10. G. Lepetil and S. P. A. Fodar, German Patent., 2,424,670, (1974);
11. Chem. Abstr., 83, 20628 (1975).
12. G. E. Hardmann and F. G. Kathawala, U.S. Patent., 4,053,600, (1997);
13. Chem. Abstr., 88, 22970 (1978).
14. J. Mohan, G. S. R Anjaneyulu, and P. Vernia, Curr. Sci., 58, 1028 (1989).
15. P. G. Baraldi, B. Cacciari, and G. Spalluto, J. Med. Chem., 39, 1164 (1996).
16. P. G. Baraldi, F. Fruttarolo, M. A. Tabrizi, D. Preti, R. Romagnoli, H. El-Kashef, et al., J. Med. Chem., 46, 1229 (2003).
17. L. B. Kier and E. B.Roche, J. Pharm. Sci., 51, 149 (1967).
18. K. Balakrishna, R. Abdul, and B. David, Arch. Pharm. Med. Chem., 334, 263 (2001).
19. C. Y.Greeo, J. Tobias, and L. B. Kier, J. Heterocycl. Chem., 4, 160 (1967).
20. L. C. Garg and C. K. Atal, Indian J. Pharm., 31, 104 (1969).
21. (a) G. Donald, V. Robert, R. Berthold, and Herbert, E. Johnson, Org. Synthesis, 5, 703;
22. (b) Walter, France, and Richard Kraft, Chem. Ber., 86, 797 (1953).
23. W. Baker, W. D. Ollis, and V. D. Poole, J. Chem. Soc., 307 (1949).
24. R. Gruickshank, J. P. Duguid, B. P. Mornion, and R. H. A. Swain, Medicinal Micro-biology, Vol. 2, p. 190 (Churchill-Livingstone, New York, 1975).