SCOPUS 정보 검색 플랫폼

Chemistry Letters

Volumn 36, Issue 2, 2007, Pages 222-223

Synthesis of N-(3-Arylmethyl-2-oxo-2,3-dihydroimidazo[1,2-a]pyridin-3-yl) benzamides

(7) Tu, Shujiang a Zhang, Junyong a Jia, Runhong a Jiang, Bo a Zhang, Yan a Yao, Changsheng a Jiang, Hong a

a JIANGSU NORMAL UNIVERSITY (China)

Author keywords

[No Author keywords available]

Indexed keywords

EID: 34247208665 PISSN: 03667022 EISSN: None Source Type: Journal
DOI: 10.1246/cl.2007.222 Document Type: Article

Times cited : (5)

References (40)

1
- 0028803899
- J. Pastor, J. Siro, J. L. Garcia-Navio, M. M. Rodrigo, M. Ballesteros, J. Alvarez-Builla, Bioorg. Med. Chem. Lett. 1995, 5, 3043.
- (1995) Bioorg. Med. Chem. Lett , vol.5 , pp. 3043
- Pastor, J.¹ Siro, J.² Garcia-Navio, J.L.³ Rodrigo, M.M.⁴ Ballesteros, M.⁵ Alvarez-Builla, J.⁶

2
- 0028145156
- a) A. Elhakmaoui, A. Gueiffier, J.-C. Milhavet, Y. Blache, J.-P. Chapat, O. Chavignon, J.-C. Teulade, R. Snoeck, G. Andrei, E. De Clercq, Bioorg. Med. Chem. Lett. 1994, 16, 1937.
- (1994) Bioorg. Med. Chem. Lett , vol.16 , pp. 1937
- Elhakmaoui, A.¹ Gueiffier, A.² Milhavet, J.-C.³ Blache, Y.⁴ Chapat, J.-P.⁵ Chavignon, O.⁶ Teulade, J.-C.⁷ Snoeck, R.⁸ Andrei, G.⁹ De Clercq, E.¹⁰

3
- 8944242597
- b) A. Gueiffier, M. Lhassani, A. Elhakmaoui, R. Snoeck, G. Andrei, O. Chavignon, J.-C. Teulade, A. Kerbal, E. M. Essassi, J.-C. Debouzy, M. Witvrouw, Y. Blache, J. Baizarini, E. De Clercq, J.-P. Chapat, J. Med. Chem. 1996, 39, 2856.
- (1996) J. Med. Chem , vol.39 , pp. 2856
- Gueiffier, A.¹ Lhassani, M.² Elhakmaoui, A.³ Snoeck, R.⁴ Andrei, G.⁵ Chavignon, O.⁶ Teulade, J.-C.⁷ Kerbal, A.⁸ Essassi, E.M.⁹ Debouzy, J.-C.¹⁰ Witvrouw, M.¹¹ Blache, Y.¹² Baizarini, J.¹³ De Clercq, E.¹⁴ Chapat, J.-P.¹⁵

4
- 34247230541
- c) L. B. Townsend, J. C. Drach, WO 27 205, 1997;
- (1997) , vol.WO 27 , Issue.205
- Townsend, L.B.¹ Drach, J.C.²

5
- 34247226240
- Chem. Abstr. 1997, 127, 190983j.
- Chem. Abstr. 1997, 127, 190983j.

6
- 0032480898
- d) A. Gueiffier, S. Mavel, M. Lhassani, A. Elhakmaoui, R. Snoeck, G. Andrei, O. Chavignon, J.-C. Teulade, M. Witvrouw, J. Balzarini, E. De Clercq, J.-P. Chapat, J. Med. Chem. 1998, 41, 5108.
- (1998) J. Med. Chem , vol.41 , pp. 5108
- Gueiffier, A.¹ Mavel, S.² Lhassani, M.³ Elhakmaoui, A.⁴ Snoeck, R.⁵ Andrei, G.⁶ Chavignon, O.⁷ Teulade, J.-C.⁸ Witvrouw, M.⁹ Balzarini, J.¹⁰ De Clercq, E.¹¹ Chapat, J.-P.¹²

7
- 0035029042
- e) S. Mavel, J. L. Renou, C. Galtier, R. Snoeck, G. Andrei, J. Balzarini, E. De Clercq, A. Gueiffier, Arzneim.-Forsch. 2001, 51, 304;
- (2001) Arzneim.-Forsch , vol.51 , pp. 304
- Mavel, S.¹ Renou, J.L.² Galtier, C.³ Snoeck, R.⁴ Andrei, G.⁵ Balzarini, J.⁶ De Clercq, E.⁷ Gueiffier, A.⁸

8
- 34247185460
- Chem. Abstr. 2001, 135, 131730s.
- Chem. Abstr. 2001, 135, 131730s.

9
- 0017857779
- J. C. Teulade, G. Grassy, J. P. Girard, J. P. Chapat, M. Simeon De Buochberg, Eur. J. Med. Chem. 1978, 13, 271.
- (1978) Eur. J. Med. Chem , vol.13 , pp. 271
- Teulade, J.C.¹ Grassy, G.² Girard, J.P.³ Chapat, J.P.⁴ Simeon De Buochberg, M.⁵

10
- 0001666197
- a) L. Almirante, L. Polo, A. Mugnaini, E. Provinciali, P. Rugarli, A. Biancotti, A. Gamba, W. Murmann, J. Med. Chem. 1965, 8, 305.
- (1965) J. Med. Chem , vol.8 , pp. 305
- Almirante, L.¹ Polo, L.² Mugnaini, A.³ Provinciali, E.⁴ Rugarli, P.⁵ Biancotti, A.⁶ Gamba, A.⁷ Murmann, W.⁸

11
- 0038459397
- b) E. Abignente, F. Arena, E. Luraschi, C. Saturnino, F. Rossi, E. Lampa, M. Cazzola, E. Brandinelli, R. Marrazzo, E. Marmo, Rend. Atti Accad. Sci. Med. Chir. 1985, 139, 313;
- (1985) Rend. Atti Accad. Sci. Med. Chir , vol.139 , pp. 313
- Abignente, E.¹ Arena, F.² Luraschi, E.³ Saturnino, C.⁴ Rossi, F.⁵ Lampa, E.⁶ Cazzola, M.⁷ Brandinelli, E.⁸ Marrazzo, R.⁹ Marmo, E.¹⁰

12
- 34247190277
- Chem. Abstr. 1986, 105, 126822z.
- Chem. Abstr. 1986, 105, 126822z.

13
- 0000010130
- c) E. Abignente, Actual. Chim. Ther. 1991, 18, 193;
- (1991) Actual. Chim. Ther , vol.18 , pp. 193
- Abignente, E.¹

14
- 34247263967
- Chem. Abstr. 1991, 115, 256028n.
- Chem. Abstr. 1991, 115, 256028n.

15
- 0038797118
- G. Bartholini, L.E.R.S. Monogr. Ser. 1993, 8, 1;
- (1993) L.E.R.S. Monogr. Ser , vol.8 , pp. 1
- Bartholini, G.¹

16
- 34247208728
- Chem. Abstr. 1996, 124, 164079n.
- Chem. Abstr. 1996, 124, 164079n.

17
- 34247275364
- K. Fuchs, M. Romig, K. Mendia, H. Briem, K. Fechteler, WO 14 313, 2002;
- (2002) , vol.WO 14 , Issue.313
- Fuchs, K.¹ Romig, M.² Mendia, K.³ Briem, H.⁴ Fechteler, K.⁵

18
- 34247262196
- Chem. Abstr. 2002, 136, 183824r.
- Chem. Abstr. 2002, 136, 183824r.

19
- 15444356141
- Y. Abe, H. Kayakiri, S. Satoh, T. Inoue, Y. Sawada, K. Imai, N. Inamura, M. Asano, C. Hatori, A. Katayama, T. Oku, H. Tanaka, J. Med. Chem. 1998, 41, 564.
- (1998) J. Med. Chem , vol.41 , pp. 564
- Abe, Y.¹ Kayakiri, H.² Satoh, S.³ Inoue, T.⁴ Sawada, Y.⁵ Imai, K.⁶ Inamura, N.⁷ Asano, M.⁸ Hatori, C.⁹ Katayama, A.¹⁰ Oku, T.¹¹ Tanaka, H.¹²

20
- 0037008399
- Y. Yamaguchi, T. Matsuno, S. Kawashima, Brain Res. 2002, 945, 259.
- (2002) Brain Res , vol.945 , pp. 259
- Yamaguchi, Y.¹ Matsuno, T.² Kawashima, S.³

21
- 0028124660
- C. Moog, A. Wick, P. Le Ber, A. Kim, A.-M. Aubertin, Antiviral Res. 1994, 24, 275.
- (1994) Antiviral Res , vol.24 , pp. 275
- Moog, C.¹ Wick, A.² Le Ber, P.³ Kim, A.⁴ Aubertin, A.-M.⁵

22
- 0025579881
- S. Z. Langer, S. Arbilla, J. Benavides, B. Scatton, Adv. Biochem. Psychopharmacol. 1990, 46, 61.
- (1990) Adv. Biochem. Psychopharmacol , vol.46 , pp. 61
- Langer, S.Z.¹ Arbilla, S.² Benavides, J.³ Scatton, B.⁴

23
- 0000972531
- a) E. S. Hand, W. W. Paudler, J. Org. Chem. 1978, 43, 2900.
- (1978) J. Org. Chem , vol.43 , pp. 2900
- Hand, E.S.¹ Paudler, W.W.²

24
- 0004193779
- b) R. Rydzkowski, D. Blondeau, H. Sliwa, Tetrahedron Lett. 1985, 26, 2571.
- (1985) Tetrahedron Lett , vol.26 , pp. 2571
- Rydzkowski, R.¹ Blondeau, D.² Sliwa, H.³

25
- 0032922157
- c) S. Löber, H. Hübner, P. Gmeiner, Bioorg. Med. Chem. Lett. 1999, 9, 97.
- (1999) Bioorg. Med. Chem. Lett , vol.9 , pp. 97
- Löber, S.¹ Hübner, H.² Gmeiner, P.³

26
- 0032993092
- d) H. Tomoda, T. Hirano, S. Saito, T. Mutai, K. Araki, Bull. Chem. Soc. Jpn. 1999, 72, 1327.
- (1999) Bull. Chem. Soc. Jpn , vol.72 , pp. 1327
- Tomoda, H.¹ Hirano, T.² Saito, S.³ Mutai, T.⁴ Araki, K.⁵

27
- 0035102259
- e) T. Ikemoto, M. Wakimasu, Heterocycles 2001, 55, 99.
- (2001) Heterocycles , vol.55 , pp. 99
- Ikemoto, T.¹ Wakimasu, M.²

28
- 85004878700
- A. J. Hubert, H. Reimlinger, Chem. Ber. 1970, 103, 3811.
- (1970) Chem. Ber , vol.103 , pp. 3811
- Hubert, A.J.¹ Reimlinger, H.²

29
- 84986479965
- H. Galons, I. Bergerat, C. Combet Farnoux, M. Miocque, Synthesis 1982, 1103.
- (1982) Synthesis , pp. 1103
- Galons, H.¹ Bergerat, I.² Combet Farnoux, C.³ Miocque, M.⁴

30
- 84984396969
- H.-J. Knölker, R. Boese, R. Hitzemann, Chem. Ber. 1990, 123, 327.
- (1990) Chem. Ber , vol.123 , pp. 327
- Knölker, H.-J.¹ Boese, R.² Hitzemann, R.³

31
- 0011434977
- M. P. Groziak, S. R. Wilson, G. L. Clauson, N. J. Leonard, J. Am. Chem. Soc. 1986, 108, 8002.
- (1986) J. Am. Chem. Soc , vol.108 , pp. 8002
- Groziak, M.P.¹ Wilson, S.R.² Clauson, G.L.³ Leonard, N.J.⁴

32
- 26844563013
- K. Groebke, L. Weber, F. Mehlin, Synlett 1998, 661.
- (1998) Synlett , pp. 661
- Groebke, K.¹ Weber, L.² Mehlin, F.³

33
- 34247215715
- L. Cai, C. Brouwer, K. Sinclair, J. Cuevas, V. W. Pike, Synthesis 2006, 113.
- (2006) Synthesis , pp. 113
- Cai, L.¹ Brouwer, C.² Sinclair, K.³ Cuevas, J.⁴ Pike, V.W.⁵

34
- 0347024178
- and references therein
- A. V. Dolzhenko, N. V. Kolotova, V. O. Kozminykh, W. Chui, P. W. S. Heng, V. N. Khrustalev, Heterocycles 2004, 63, 55, and references therein.
- (2004) Heterocycles , vol.63 , pp. 55
- Dolzhenko, A.V.¹ Kolotova, N.V.² Kozminykh, V.O.³ Chui, W.⁴ Heng, P.W.S.⁵ Khrustalev, V.N.⁶

35
- 0001565605
- C. Plorac, M. Baudy-noćh, A. Robert, Tetrahedron 1990, 46, 445.
- (1990) Tetrahedron , vol.46 , pp. 445
- Plorac, C.¹ Baudy-noćh, M.² Robert, A.³

36
- 28344438335
- a) S. Tu, T. Li, F. Shi, Q. Wang, J. Zhang, J. Xu, X. Zhu, X. Zhang, S. Zhu, D. Shi, Synthesis 2005, 3045.
- (2005) Synthesis , pp. 3045
- Tu, S.¹ Li, T.² Shi, F.³ Wang, Q.⁴ Zhang, J.⁵ Xu, J.⁶ Zhu, X.⁷ Zhang, X.⁸ Zhu, S.⁹ Shi, D.¹⁰

37
- 33748968361
- b) S. J. Tu, B. Jiang, R. H. Jia, J. Y. Zhang, Y. Zhang, C. S. Yao, F. Shi, Org. Biomol. Chem. 2006, 4, 3664.
- (2006) Org. Biomol. Chem , vol.4 , pp. 3664
- Tu, S.J.¹ Jiang, B.² Jia, R.H.³ Zhang, J.Y.⁴ Zhang, Y.⁵ Yao, C.S.⁶ Shi, F.⁷

38
- 33750154643
- c) S. J. Tu, B. Jiang, J. Y. Zhang, R. H. Jia, Y. Zhang, C. S. Yao, Org. Biomol. Chem. 2006, 4, 3980.
- (2006) Org. Biomol. Chem , vol.4 , pp. 3980
- Tu, S.J.¹ Jiang, B.² Zhang, J.Y.³ Jia, R.H.⁴ Zhang, Y.⁵ Yao, C.S.⁶

39
- 0038044688
- S. J. Tu, H. Jiang, Q. Y. Zhuang, C. B. Miao, D. Q. Shi, X. S. Wang, Y. Gao, Chin. J. Org. Chem. 2003, 23, 491.
- (2003) Chin. J. Org. Chem , vol.23 , pp. 491
- Tu, S.J.¹ Jiang, H.² Zhuang, Q.Y.³ Miao, C.B.⁴ Shi, D.Q.⁵ Wang, X.S.⁶ Gao, Y.⁷

40
- 34247239456
- General procedures for the synthesis of 3 are as follows: A mixture of 4-arylidene-2-phenyl-5(4H)-oxazolones (1, 1 mmol) and pyridin-2-amine (2, 1 mmol) was added to a 10-mL reaction vessel of the monomodal Emrys™ Creator microwave synthesizer and allowed to react under microwave irradiation at 240 W power and 120°C in ethylene glycol (2 mL) for 4-7 min. The reaction mixture was cooled to room temperature, then poured into water (50 mL, filtered to give crude product, which was further purified by recrystallization from EtOH (3a-31, Compound 3e: IR (KBr, 3241, 3014, 2987, 1679, 1664, 1567, 1532, 868, 809, 786, 724, 591 cm-1; 1H NMR (DMSO-d6, δ, ppm, δ 9.69 (s, 1H, NH, 8.30 (d, 1H, J, 6.4Hz, ArH, 8.04 (d, 2H, J, 8.4 Hz, ArH, 7.92 (d, 2H, J, 7.6 Hz, ArH, 7.65-7.52 (m, 4H, ArH, 7.15 (d, 2H, 7, 8.4 Hz, ArH, 6.82-6.74 (m, 2H, ArH, 3.69 (d, 1H, J, 13.2 Hz, CH2, 3.46 d, 1H, J, 13.2 Hz, CH2
- 4: C, 64.94; H, 4.15; N, 14.43%. Found: C, 65.12; H, 4.20; N, 14.28%.

* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.