Selection of new chromogenic substrates of serine proteinases using combinatorial chemistry methods

Combinatorial Chemistry and High Throughput Screening

Volumn 10, Issue 3, 2007, Pages 171-180

  Wysocka, Magdalena ^a   Kwiatkowska, Bozena ^a   Rzadkiewicz, Marek ^a   Lesner, Adam ^a   Rolka, Krzysztof ^a  

^a UNIVERSITY OF GDA SK   (Poland)

Author keywords

Chromogenic substrates; p nitroanilides; Peptide library; Serine proteinase

Indexed keywords

5 AMINO 2 NITROBENZOIC ACID; AMIDE; BENZOIC ACID DERIVATIVE; CHROMOGENIC SUBSTRATE; CHYMOTRYPSIN A; LEUKOCYTE ELASTASE; PEPTIDE LIBRARY; SERINE PROTEINASE; TETRAPEPTIDE; UNCLASSIFIED DRUG;

AMINO ACID SEQUENCE; AMINO TERMINAL SEQUENCE; ARTICLE; CARBOXY TERMINAL SEQUENCE; CHROMATOPHORE; COMBINATORIAL CHEMISTRY; ENZYME MECHANISM; ENZYME SUBSTRATE; KINETICS; PEPTIDE SYNTHESIS; PHYSICAL CHEMISTRY; PRIORITY JOURNAL; SYNTHESIS;

ANIMALS; CATTLE; CHROMOGENIC COMPOUNDS; CHYMOTRYPSIN; COMBINATORIAL CHEMISTRY TECHNIQUES; HUMANS; LEUKOCYTE ELASTASE; OLIGOPEPTIDES; PEPTIDE LIBRARY; SERINE ENDOPEPTIDASES; SUBSTRATE SPECIFICITY;

BOVINAE;

EID: 33947287859     PISSN: 13862073     EISSN: None     Source Type: Journal    
DOI: 10.2174/138620707780126714     Document Type: Article

References (27)

1. Erlanger, B.F.; Kokovsky, N.; Cohen, W. Arch. Biochem. Biophys., 1961, 95, 271.
2. Polanowska, J.; Krokoszynska, I.; Czapinska, H.; Watorek, W.; Dadlez, M.; Otlewski, J. Biochim. Biophys. Acta, 1998, 1386, 189.
3. Hsieh, M.L.; Tseng, M.J.; Tseng, M.C.; Chu, Y.H. Anal. Biochem., 2006, 354, 104.
4. Lu, W.; Apostol, I.; Qasim, M.A.; Warne, N.; Wynn, R.; Zhang, W.L.; Anderson, S.; Chiang, Y.W.; Ogin, E.; Rothberg, I.; Ryan, K.; Laskowski, M. Jr. J. Mol. Biol., 1997, 266, 441.
5. Lesner, A.; Brzozowski, K.; Kupryszewski, G; Rolka, K. Biochem. Biophys. Res. Commun., 2000, 269, 81.
6. Rano, T.A.; Timkey, T.; Peterson, E.P.; Rotonda, J.; Nicholson, D.W.; Becker, J.W.; Chapman, K.T.; Thornberry, N.A. Chem. Biol., 1997, 4, 149.
7. Matsumura, M.; Bhatt, A.S.; Andress, D.; Clegg, N.; Takayama, T.K.; Craik, C.S.; Nelson, P.S. Prostate, 2005, 62, 1.
8. Mathieu, M.A.; Bogyo, M.; Caffrey, C.R.; Choe, Y.; Lee, J.; Chapman, H.; Sajid, M.; Craik, C.S.; McKerrow, J.H. Mol. Biochem. Parasitol., 2002, 121, 99.
9. Beyer, B.B.; Johnson, J.V.; Chung, A.Y.; Li., T.; Madabushi, A; Agbandje-McKenna, M.; McKenna, R.; Dame, J.B.; Dunn, B.M. Biochemistry, 2005, 44, 1768.
10. Kaspari, A.; Schierhorn, A.; Schutkowski, M. Int. J. Pept. Protein Res., 1996, 48, 486.
11. Schutkowski, M.; Mrestani-Klaus, C.; Neubert, K. Int. J. Peptide Protein Res., 1995, 45, 257.
12. Hojo, K.; Maeda, M.; Iguchi, S.; Smith, T.; Okamoto, H.; Kawasaki, K. Chem. Pharm. Bull., 2000, 48, 1740.
13. Zabłotna, E.; Dysasz, H.; Lesner, A.; Jaśkiewicz, A.; Kaźmierczak, K; Miecznikowska, H.; Rolka, K. Biochem. Biophys. Res. Commun., 2004, 319, 185.
14. Kaźmierczak, K.; Zabłotna, E.; Jaśkiewicz, A.; Miecznikowska, H.; Rolka, K. Biochem. Biophys. Res. Commun., 2003, 310, 811.
15. Hougten, R.H.; Pinilla, C.; Blondelle, S.E.; Appel, J.R.; Dooley, C.T.; Cuervo J.H. Nature, 1991, 354, 84.
16. Sole, N.A.; Barany, G. J. Org. Chem., 1992, 57, 5399.
17. Furka, A.; Sebestyn, F.; Asgedom, M.; Dib, G. Int. J. Peptide Prot. Res., 1991, 37, 487.
18. Ostresh, J.M.; Blondelle, S.E.; Dorner, B.; Houghten, R.A. Methods Enzymol., 1996, 267, 220.
19. Furlong, S.T.; Mauger, R.C.; Strimpler, A.M.; Liu, Y.P.; Morris, F.X.; Edwards, P.D. Bioorg. Med. Chem., 2002, 10, 3637.
20. Lesner, A.; Kupryszewski, G.; Rolka, K. Biochem. Biophys. Res. Commun., 2001, 285, 1350.
21. Schellenberger, V.; Braune, K.; Hofmann, H.-J.; Jakubke, H.-D. Eur. J. Biochem., 1991, 199, 623.
22. Laskowski Jr M.; Kato I. Annu. Rev. Biochem., 1980, 49, 593.
23. Brauer, A.B.; Nievo, M.; Mcbride, J.D.; Leatherbarrow, R.J. J. Biomol. Struct. Dyn., 2003, 20, 645.
24. Harris, J.L., Bradley, J.B., Leonetii, F., Mahrus, S., Ellman, A., Craik, C.S. Proc. Natl. Acad. Sci. USA, 2000, 97, 7754.
25. Wesolowska, O, Krokoszynska, I, Krowarsch, D, Otlewski, J. Biochim. Biophys. Acta, 2001, 1545, 78.
26. Nakajima, K., Powers, J.C., Ashe, B.M., Zimmerman M. J. Biol. Chem., 1979, 254, 4027.
27. Bode, W.; Meyer, E. Jr.; Powers, J.C. Biochemistry, 1989, 28, 1951.