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European Journal of Medicinal Chemistry

Volumn 42, Issue 2, 2007, Pages 175-197

New polyamine-sensitive inhibitors of the NMDA receptor: Syntheses and pharmacological evaluation

(6) Pöhler, Thomas a,c Schadt, Oliver c Niepel, Daniela a Rebernik, Patrick b Berger, Michael L b Noe, Christian R a,c

a UNIVERSITY OF VIENNA (Austria)

b MEDICAL UNIVERSITY OF VIENNA (Austria)

c GOETHE UNIVERSITY (Germany)

Author keywords

1,12 Diaminododecane; NMDA receptor; Polyamine inverse agonist; Spermine; Thiophene

Indexed keywords

AMIDE; AMINE; BENZENE; DIZOCILPINE; GUANIDINE DERIVATIVE; N METHYL DEXTRO ASPARTIC ACID RECEPTOR; N METHYL DEXTRO ASPARTIC ACID RECEPTOR BLOCKING AGENT; OCTYLAMINE; PIPERIDINE; POLYAMINE DERIVATIVE; SPERMINE; TROMETAMOL;

ALKYLATION; ANNULATION REACTION; ARTICLE; BRAIN MEMBRANE; CHEMICAL BOND; CLEMMENSEN REDUCTION; DEPROTECTION REACTION; DRUG POTENCY; DRUG RECEPTOR BINDING; DRUG SCREENING; DRUG SYNTHESIS; FRIEDEL CRAFTS REACTION; IC 50; METHYLATION; NONHUMAN; QUANTUM YIELD; RAT; REACTION ANALYSIS; STRUCTURE ACTIVITY RELATION; SUBSTITUTION REACTION;

ANIMALS; BRAIN; POLYAMINES; RADIOLIGAND ASSAY; RATS; RECEPTORS, N-METHYL-D-ASPARTATE; STRUCTURE-ACTIVITY RELATIONSHIP; THIOPHENES;

EID: 33847161755 PISSN: 02235234 EISSN: 17683254 Source Type: Journal
DOI: 10.1016/j.ejmech.2006.09.017 Document Type: Article

Times cited : (8)

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