-
3
-
-
0030738669
-
-
S. E. de Sousa, P. O'Brien and P. Poumellec, Tetrahedron: Asymmetry, 1997, 8, 2613.
-
(1997)
Tetrahedron: Asymmetry
, vol.8
, pp. 2613
-
-
De Sousa, S.E.1
O'Brien, P.2
Poumellec, P.3
-
4
-
-
0001762573
-
-
(a) R. Shirai, M. Tanaka and K. Koga, J. Am. Chem. Soc., 1986, 108, 543;
-
(1986)
J. Am. Chem. Soc.
, vol.108
, pp. 543
-
-
Shirai, R.1
Tanaka, M.2
Koga, K.3
-
5
-
-
0001704054
-
-
(b) H. Kim, R. Shirai, H. Kawasaki, M. Nakajima and K. Koga, Heterocycles, 1990, 30, 307;
-
(1990)
Heterocycles
, vol.30
, pp. 307
-
-
Kim, H.1
Shirai, R.2
Kawasaki, H.3
Nakajima, M.4
Koga, K.5
-
6
-
-
0030906129
-
-
(c) R. Shirai, D. Sato, K. Aoki, M. Tanaka, H. Kawasaki and K. Koga, Tetrahedron, 1997, 53, 5963.
-
(1997)
Tetrahedron
, vol.53
, pp. 5963
-
-
Shirai, R.1
Sato, D.2
Aoki, K.3
Tanaka, M.4
Kawasaki, H.5
Koga, K.6
-
10
-
-
0028910707
-
-
(b) D. Bhuniya, A. DattaGupta and V. K. Singh, Tetrahedron Lett., 1995, 36, 2847.
-
(1995)
Tetrahedron Lett.
, vol.36
, pp. 2847
-
-
Bhuniya, D.1
DattaGupta, A.2
Singh, V.K.3
-
11
-
-
0000803525
-
-
D. Bhuniya, A. DattaGupta and V. K. Singh, J. Org. Chem., 1996, 61, 6108.
-
(1996)
J. Org. Chem.
, vol.61
, pp. 6108
-
-
Bhuniya, D.1
DattaGupta, A.2
Singh, V.K.3
-
12
-
-
0030580414
-
-
For a review, see: D. M. Hodgson, A. R. Gibbs and G. P. Lee, Tetrahedron, 1996, 52, 14 361.
-
(1996)
Tetrahedron
, vol.52
, pp. 14361
-
-
Hodgson, D.M.1
Gibbs, A.R.2
Lee, G.P.3
-
15
-
-
0027411133
-
-
B. E. Rossiter, M. Eguchi, G. Miao, N. M. Swingle, A. E. Hernandez, E. Fluckiger, D. Vickers, R. G. Patterson and K. V. Reddy, Tetrahedron, 1993, 49, 965.
-
(1993)
Tetrahedron
, vol.49
, pp. 965
-
-
Rossiter, B.E.1
Eguchi, M.2
Miao, G.3
Swingle, N.M.4
Hernandez, A.E.5
Fluckiger, E.6
Vickers, D.7
Patterson, R.G.8
Reddy, K.V.9
-
18
-
-
0026031238
-
-
(a) G. F. Costello, R. James, J. S. Shaw, A. M. Slater and N. C. Stutchbury, J. Med. Chem., 1991, 34, 181;
-
(1991)
J. Med. Chem.
, vol.34
, pp. 181
-
-
Costello, G.F.1
James, R.2
Shaw, J.S.3
Slater, A.M.4
Stutchbury, N.C.5
-
19
-
-
0026344565
-
-
(b) J. J. Barlow, T. P. Blackburn, G. F. Costello, R. James, D. J. Le Count, B. G. Main, R. J. Pearce, K. Russell and J. S. Shaw, J. Med. Chem., 1991, 34, 3149.
-
(1991)
J. Med. Chem.
, vol.34
, pp. 3149
-
-
Barlow, J.J.1
Blackburn, T.P.2
Costello, G.F.3
James, R.4
Le Count, D.J.5
Main, B.G.6
Pearce, R.J.7
Russell, K.8
Shaw, J.S.9
-
20
-
-
0028304348
-
-
(a) A.-C. Chang, A. E. Takemori and P. S. Portoghese, J. Med. Chem., 1994, 37, 1547;
-
(1994)
J. Med. Chem.
, vol.37
, pp. 1547
-
-
Chang, A.-C.1
Takemori, A.E.2
Portoghese, P.S.3
-
21
-
-
0028000959
-
-
(b) S. A. Weerawarna, R. D. Davis and W. L. Nelson, J. Med. Chem., 1994, 37, 2856;
-
(1994)
J. Med. Chem.
, vol.37
, pp. 2856
-
-
Weerawarna, S.A.1
Davis, R.D.2
Nelson, W.L.3
-
22
-
-
0028590201
-
-
(c) A.-C. Chang, A. E. Takemori, W. H. Ojala, W. B. Gleason and P. S. Portoghese, J. Med. Chem., 1994, 37, 4490;
-
(1994)
J. Med. Chem.
, vol.37
, pp. 4490
-
-
Chang, A.-C.1
Takemori, A.E.2
Ojala, W.H.3
Gleason, W.B.4
Portoghese, P.S.5
-
23
-
-
0029037439
-
-
(d) G. A. Pinna, E. Gavini, G. Cignarella, S. Scolastico and P. Fadda, Eur. J. Med. Chem., 1995, 30, 515.
-
(1995)
Eur. J. Med. Chem.
, vol.30
, pp. 515
-
-
Pinna, G.A.1
Gavini, E.2
Cignarella, G.3
Scolastico, S.4
Fadda, P.5
-
25
-
-
24244444143
-
-
(Pfizer Inc.) 1996, JP-00820
-
F. Ito (Pfizer Inc.) 1996, JP-00820 (Chem. Abstr., 1996, 125, 86 487y).
-
(1996)
Chem. Abstr.
, vol.125
-
-
Ito, F.1
-
26
-
-
0028291746
-
-
R. Shirai, K. Aoki, D. Sato, H.-D. Kim, M. Murakata, T. Yasukata and K. Koga, Chem. Pharm. Bull., 1994, 42, 690.
-
(1994)
Chem. Pharm. Bull.
, vol.42
, pp. 690
-
-
Shirai, R.1
Aoki, K.2
Sato, D.3
Kim, H.-D.4
Murakata, M.5
Yasukata, T.6
Koga, K.7
-
27
-
-
0026353381
-
-
Racemisation during reactions of N-protected phenylglycine-derivatives is well documented. See for example: J.-N. Denis, A. Correa and A. E. Greene, J. Org. Chem., 1991, 56, 6939.
-
(1991)
J. Org. Chem.
, vol.56
, pp. 6939
-
-
Denis, J.-N.1
Correa, A.2
Greene, A.E.3
-
28
-
-
0347238854
-
-
(a) R. K. Dieter, B. Lagu, J. W. Dieter, N. Deo and W. T. Pennington, Synlett, 1990, 109;
-
(1990)
Synlett
, pp. 109
-
-
Dieter, R.K.1
Lagu, B.2
Dieter, J.W.3
Deo, N.4
Pennington, W.T.5
-
29
-
-
0026572789
-
-
(b) R. K. Dieter, N. Deo, B. Lagu and J. W. Dieter, J. Org. Chem., 1992, 57, 1663.
-
(1992)
J. Org. Chem.
, vol.57
, pp. 1663
-
-
Dieter, R.K.1
Deo, N.2
Lagu, B.3
Dieter, J.W.4
-
30
-
-
0030734433
-
-
For examples of aziridinium ion intermediates in synthesis, see: (a) Q. Liu, A. P. Marchington and C. M. Rayner, Tetrahedron, 1997, 53, 15 729;
-
(1997)
Tetrahedron
, vol.53
, pp. 15729
-
-
Liu, Q.1
Marchington, A.P.2
Rayner, C.M.3
-
31
-
-
33748664816
-
-
(b) Q. Liu, A. P. Marchington, N. Boden and C. M. Rayner, J. Chem. Soc., Perkin Trans. 1, 1997; 511;
-
(1997)
J. Chem. Soc., Perkin Trans. 1
, pp. 511
-
-
Liu, Q.1
Marchington, A.P.2
Boden, N.3
Rayner, C.M.4
-
34
-
-
0028104847
-
-
(e) P. Gmeiner, D. Junge and A. Kärtner, J. Org. Chem., 1994, 59, 6766;
-
(1994)
J. Org. Chem.
, vol.59
, pp. 6766
-
-
Gmeiner, P.1
Junge, D.2
Kärtner, A.3
-
35
-
-
0000149768
-
-
(f) J. Freedman, M. J. Vaal and E. W. Huber, J. Org. Chem., 1991, 56, 670;
-
(1991)
J. Org. Chem.
, vol.56
, pp. 670
-
-
Freedman, J.1
Vaal, M.J.2
Huber, E.W.3
-
36
-
-
0024544606
-
-
(g) D. R. Williams, D. L. Brown and J. W. Benbow, J. Am. Chem. Soc., 1989, 111, 1923;
-
(1989)
J. Am. Chem. Soc.
, vol.111
, pp. 1923
-
-
Williams, D.R.1
Brown, D.L.2
Benbow, J.W.3
-
37
-
-
0023744270
-
-
(h) T. Rosen, S. W. Fesik, D. T. W. Chu and A. G. Pernet, Synthesis, 1988, 40;
-
(1988)
Synthesis
, pp. 40
-
-
Rosen, T.1
Fesik, S.W.2
Chu, D.T.W.3
Pernet, A.G.4
-
41
-
-
33748636864
-
-
(R)- and (S)-styrene oxide are available from the Aldrich Chemical Company
-
(R)- and (S)-styrene oxide are available from the Aldrich Chemical Company.
-
-
-
-
42
-
-
0001274664
-
-
S. Miyano, L. D.-L. Lu, S. M. Viti and K. B. Sharpless, J. Org. Chem., 1985, 50, 4350.
-
(1985)
J. Org. Chem.
, vol.50
, pp. 4350
-
-
Miyano, S.1
Lu, L.D.-L.2
Viti, S.M.3
Sharpless, K.B.4
-
44
-
-
0003084239
-
-
A. Toshimitsu, C. Hirosawa and K. Tamao, J. Chem. Soc., Chem. Commun., 1989, 530.
-
(1989)
J. Chem. Soc., Chem. Commun.
, pp. 530
-
-
Toshimitsu, A.1
Hirosawa, C.2
Tamao, K.3
-
45
-
-
0028041025
-
-
A. Toshimitsu, C. Hirosawa and K. Tamao, Tetrahedron, 1994, 50, 8997.
-
(1994)
Tetrahedron
, vol.50
, pp. 8997
-
-
Toshimitsu, A.1
Hirosawa, C.2
Tamao, K.3
-
46
-
-
33748650521
-
-
Dr Simon A. Osborne, personal communication
-
Dr Simon A. Osborne, personal communication.
-
-
-
-
47
-
-
33748659422
-
-
(R)- and (S)-phenylglycinol are commercially available from Lancaster Synthesis
-
(R)- and (S)-phenylglycinol are commercially available from Lancaster Synthesis.
-
-
-
-
48
-
-
85026861700
-
-
2O), we have prepared 3.26 g of (R)-phenylglycinol (73% yield): M. A. Tschantz, L. E. Burgess and A. I. Meyers, Org. Synth., 1996, 73, 221.
-
(1996)
Org. Synth.
, vol.73
, pp. 221
-
-
Tschantz, M.A.1
Burgess, L.E.2
Meyers, A.I.3
-
49
-
-
37049083984
-
-
M. Meguro, N. Asao and Y. Yamamoto, J. Chem. Soc., Perkin Trans. 1, 1994, 2597.
-
(1994)
J. Chem. Soc., Perkin Trans. 1
, pp. 2597
-
-
Meguro, M.1
Asao, N.2
Yamamoto, Y.3
-
50
-
-
0030200768
-
-
E. Brown, A. Lézé and J. Touet, Tetrahedron: Asymmetry, 1996, 7, 2029.
-
(1996)
Tetrahedron: Asymmetry
, vol.7
, pp. 2029
-
-
Brown, E.1
Lézé, A.2
Touet, J.3
-
51
-
-
0025753973
-
-
E. Brown, A. Penfornis, J. Bayma and J. Touet, Tetrahedron: Asymmetry, 1991, 2, 339.
-
(1991)
Tetrahedron: Asymmetry
, vol.2
, pp. 339
-
-
Brown, E.1
Penfornis, A.2
Bayma, J.3
Touet, J.4
-
53
-
-
0031019992
-
-
J. Juárez, D. Gnecco, A. Galindo, R. G. Enríquez, C. Marazano and W. F. Reynolds, Tetrahedron: Asymmetry, 1997, 8, 203.
-
(1997)
Tetrahedron: Asymmetry
, vol.8
, pp. 203
-
-
Juárez, J.1
Gnecco, D.2
Galindo, A.3
Enríquez, R.G.4
Marazano, C.5
Reynolds, W.F.6
-
54
-
-
0002714675
-
-
W. C. Still, M. Kahn and A. Mitra, J. Org. Chem., 1978, 43, 2923.
-
(1978)
J. Org. Chem.
, vol.43
, pp. 2923
-
-
Still, W.C.1
Kahn, M.2
Mitra, A.3
|