Antibacterial and antifungal activity of acyclic and macrocyclic uracil derivatives with quaternized nitrogen atoms in spacers

European Journal of Medicinal Chemistry

Volumn 41, Issue 9, 2006, Pages 1093-1101

  Semenov, V E ^a   Voloshina, A D ^a   Toroptzova, E M ^a   Kulik, N V ^a   Zobov, V V ^a   Giniyatullin, R K ^a   Mikhailov, A S ^a   Nikolaev, A E ^a   Akamsin, V D ^a   Reznik, V S ^a  

^a A E ARBUZOV INSTITUTE OF ORGANIC AND PHYSICAL CHEMISTRY   (Russian Federation)

Author keywords

Antibacterial activity; Antifungal activity; Pyrimidinophanes; Quaternization; Toxicity; Uracils

Indexed keywords

CARBENE; CARBONYL DERIVATIVE; MACROCYCLIC COMPOUND; NITROGEN; PYRIDINE DERIVATIVE; URACIL DERIVATIVE; ANTIFUNGAL AGENT; ANTIINFECTIVE AGENT; DRUG DERIVATIVE; URACIL;

ANIMAL EXPERIMENT; ANTIBACTERIAL ACTIVITY; ANTIFUNGAL ACTIVITY; ARTICLE; ASPERGILLUS NIGER; BACILLUS SUBTILIS; CONTROLLED STUDY; DAPHNIA; DRUG CONFORMATION; DRUG DETERMINATION; DRUG STRUCTURE; ESCHERICHIA COLI; FUNGICIDAL ACTIVITY; GRAM NEGATIVE BACTERIUM; GRAM POSITIVE BACTERIUM; LETHAL DOSE; MICROBIAL ACTIVITY; MINIMUM INHIBITORY CONCENTRATION; MOUSE; NONHUMAN; PSEUDOMONAS AERUGINOSA; STAPHYLOCOCCUS AUREUS; STRUCTURE ANALYSIS; TRICHOPHYTON MENTAGROPHYTES; ANIMAL; CHEMICAL STRUCTURE; CHEMISTRY; DEUTEROMYCETES; DRUG EFFECT; ISOMERISM; STRUCTURE ACTIVITY RELATION; SYNTHESIS;

ANIMALS; ANTI-BACTERIAL AGENTS; ANTIFUNGAL AGENTS; DAPHNIA; GRAM-NEGATIVE BACTERIA; GRAM-POSITIVE BACTERIA; ISOMERISM; MACROCYCLIC COMPOUNDS; MICE; MITOSPORIC FUNGI; MOLECULAR STRUCTURE; NITROGEN; STRUCTURE-ACTIVITY RELATIONSHIP; URACIL;

EID: 33748451272     PISSN: 02235234     EISSN: 17683254     Source Type: Journal    
DOI: 10.1016/j.ejmech.2006.03.030     Document Type: Article

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